Enzyme Substrates / Activators
Products for Enzyme Substrates / Activators
- Cat.No. Product Name Information
-
GC41698
(D)2-Rh 110 (trifluoroacetate salt)
D2R, (Asp)2-Rhodamine 110, Rhodamine 110 bis-(L-aspartic acid amide)
(D)2-Rh 110 is a fluorogenic caspase substrate. -
GC40121
(Z-DEVD)2-Rh 110 (trifluoroacetate salt)
(Z-Asp-Glu-Val-Asp)2-Rhodamine 110
(Z-DEVD)2-Rh 110 is a fluorogenic substrate for caspase-3. -
GC41742
(Z-IETD)2-Rh 110 (trifluoroacetate salt)
(Z-Ile-Glu-Thr-Asp)2-R110, Rhodamine 110 bis-(N-CBZ-IETD)2
(Z-IETD)2-Rh 110 is a fluorogenic substrate for caspase-8. -
GC90815
2',3'-cyclic NADP+ (sodium salt)
A substrate for CNP
-
GC15945
2B-(SP)
Selective phosphopeptide substrate for glycogen synthase kinase-3 (GSK-3)
-
GC42450
4-Methylumbelliferyl-α-L-Iduronide 2-sulfate (sodium salt)
4Methylumbelliferyl-α-L-Idopyranosiduronic Acid 2-sulfate, 4-MU-α-IdoA 2-sulfate
4-Methylumbelliferyl-α-L-iduronide 2-sulfate (4-MU-α-IdoA 2-sulfate) is a fluorogenic substrate of α-L-iduronidase that has been used in an assay to detect Hurler syndrome. -
GC19852
4-Methylumbelliferyl-α-D-glucopyranoside
4-Methylumbelliferyl-α-D-Glucose, 4-Methylumbelliferyl-α-D-Glucoside, 4-MU-α-D-Glucopyranoside
-
GC90796
5-(3-Aminoallyl)-2'-deoxyuridine-5'-O-triphosphate (sodium salt)
An amine-modified nucleotide
-
GC48435
5-Bromo-4-chloro-3-indolyl-β-D-Glucuronide (cyclohexylammonium salt hydrate)
BCIG, X-GLUC
-
GC20169
5-Bromo-4-Chloro-3-Indolyl-Alpha-D-Galactopyranoside
Rarechem AH BS 0009; X-Alpha-Gal; X-Alpha-D-Gal; X-Alpha-D-GalACTOSIDE; X-A-Gal; 5-Bromo-4-Chloro-3-Indoxyl-Alpha-D-GalACTOPYRANOSIDE; Alpha-X-Gal; 5-Bromo-4-Chloro-3-Indolyl-Alp
-
GC52499
Abz-Ala-Pro-Glu-Glu-Ile-Met-Arg-Arg-Gln-EDDnp (trifluoroacetate salt)
A sensitive substrate for neutrophil elastase
-
GC42687
Ac-DMQD-AMC (trifluoroacetate salt)
Ac-Asp-Met-Gln-Asp-AMC, Ac-Asp-Met-Gln-Asp-7-amino-4-methylcoumarin
Ac-DMQD-AMC is a fluorogenic substrate for caspase-3. -
GC42706
Ac-IEPD-AMC (trifluoroacetate salt)
Acetyl-Ile-Glu-Pro-Asp-7-amino-4-Methylcoumarin, Ac-Ile-Glu-Pro-Asp-AMC
Ac-IEPD-AMC is a fluorogenic substrate for granzyme B. -
GC40152
Ac-IEPD-pNA (trifluoroacetate salt)
Ac-Ile-Glu-Pro-Asp-p-nitroanilide, Caspase-8 Chromogenic Substrate, Granzyme B Substrate VIII
Ac-IEPD-pNA is a colorimetric substrate for granzyme B and caspase-8. -
GC42708
Ac-LEHD-AFC (trifluoroacetate salt)
N-Acetyl-Leu-Glu-His-Asp-7-amino-4-Trifluoromethylcoumarin, Caspase-9 substrate (Fluorogenic)
Ac-LEHD-AFC is a fluorogenic substrate that can be cleaved by caspase-4, -5, and -9. -
GC46791
Ac-LEHD-pNA (trifluoroacetate salt)
Ac-Leu-Glu-His-Asp-pNA, Caspase-9 Chromogenic Substrate I
A neuropeptide with diverse biological activities -
GC45683
Ac-QQQ-AMC (hydrochloride)
Ac-Gln-Gln-Gln-AMC, Ac-Gln-Gln-Gln-7-amino-4-methylcoumarin, Ac-L-Gln-L-Gln-L-Gln-AMC
A neuropeptide with diverse biological activities -
GC42712
Ac-RLR-AMC (trifluoroacetate salt)
Ac-Arg-Leu-Arg-AMC, Ac-Arg-Leu-Arg-7-amino-4-Methylcoumarin
Ac-RLR-AMC is a fluorogenic substrate for the 26S proteasome. -
GC52372
Ac-VDVAD-AFC (trifluoroacetate salt)
N-Acetyl-Val-Asp-Val-Ala-Asp-AFC, N-Acetyl-Val-Asp-Val-Ala-Asp-7-amino-4-Trifluoromethylcoumarin, Caspase-2 Substrate (Fluorogenic)
A fluorogenic substrate for caspase-2 -
GC42716
Ac-VDVAD-pNA (trifluoroacetate salt)
Ac-Val-Asp-Val-Ala-Asp-pNA, Caspase-2 Chromogenic Substrate, acetyl-Val-Asp-Val-Ala-Asp-p-nitroanilide, acetyl-VDVAD-p-nitroanilide
Ac-VDVAD-pNA is a colorimetric substrate for caspase-2. -
GC40162
Ac-VEID-pNA (trifluoroacetate salt)
Ac-Val-Glu-Ile-Asp-pNA, Ac-Val-Glu-Ile-Asp-p-nitroanilide, Caspase-6 Chromogenic Substrate
Ac-VEID-pNA is a substrate for caspase-6. -
GC40124
Ac-WEAD-AMC (trifluoroacetate salt)
Ac-Trp-Glu-Ala-Asp-AMC
Ac-WEAD-AMC is a fluorogenic substrate for caspase-1 and caspase-4. -
GC42719
Ac-WEAD-pNA (trifluoroacetate salt)
Ac-Trp-Glu-Ala-Asp-pNA, Ac-Trp-Glu-Ala-Asp-p-nitroanilide, Caspase-1 and Caspase-4 Chromogenic Substrate
Ac-WEAD-pNA is a colorimetric substrate for caspase-1 and caspase-4. -
GC46796
Ac-WEHD-AFC (trifluoroacetate salt)
N-Acetyl-Trp-Glu-His-Asp-7-amino-4-Trifluoromethylcoumarin, Caspase1 Substrate (Fluorogenic), Caspase5 Substrate (Fluorogenic)
A neuropeptide with diverse biological activities -
GC52443
Akt Substrate (trifluoroacetate salt)
RPRAATF
An Akt peptide substrate -
GC15822
Akt/SKG Substrate Peptide
substrate for Akt/PKB
-
GC12160
AKTide-2T
Peptide substrate for Akt/PKB
-
GC52361
AMARA Peptide (trifluoroacetate salt)
AMARAASAAALARRR-OH, H-Ala-Met-Ala-Arg-Ala-Ala-Ser-Ala-Ala-Ala-Leu-Ala-Arg-Arg-Arg-OH
A peptide substrate for AMPK -
GC42876
Autocamtide 2 (trifluoroacetate salt)
Autocamtide 2 is a peptide substrate for calcium/calmodulin-dependent protein kinase (CaMK) and CaMKII.
-
GC90276
Boc-LRR-AMC (trifluoroacetate salt)
A fluorogenic substrate for trypsin-like activity of the 26S proteasome or 20S proteolytic core
-
GC52488
Bz-FVR-AMC (trifluoroacetate salt)
Benzoyl-Phe-Val-Arg-AMC, Thrombin Fluorogenic Substrate III
A fluorogenic peptide substrate -
GC52360
Chymotrypsin Substrate I, Colorimetric (trifluoroacetate salt)
Suc-GGF-pNA, Suc-Gly-Gly-Phe-pNA, Suc-Gly-Gly-Phe-p-Nitroanilide
A colorimetric chymotrypsin substrate -
GC52387
Crosstide (trifluoroacetate salt)
Gly-Arg-Pro-Arg-Thr-Ser-Ser-Phe-Ala-Glu-Gly-OH, GRPRTSSFAEG-OH
A peptide substrate for Akt -
GC47164
Dabcyl-GABA-PQGL-Glu(EDANS)-AK-NH2, (trifluoroacetate salt)
MMP Fluorogenic Substrate III
A neuropeptide with diverse biological activities -
GC43369
Dabcyl-GABA-RPKPVE-Nva-WR-Glu(EDANS)-AK-NH2 (trifluoroacetate salt)
Dabcyl-GABA-RPKPVE-Nva-WR-Glu(EDANS)-AK-NH2 is a fluorogenic substrate for matrix metalloproteinase-3 (MMP-3).
-
GC43370
Dabcyl-RGVVNASSRLA-EDANS (trifluoroacetate salt)
Fluorogenic Human CMV Protease Substrate
Dabcyl-RGVVNASSRLA-EDANS is a fluorogenic substrate for human cytomegalovirus (HCMV) protease. -
GC43451
Dieosinediglutathione
DiEGSSG
Dieosinediglutathione is the product of glutathione disulfide and eosin isothiocyanate which has been purified and lyophilized. -
GC43542
Dnp-GPLGMRGL-NH2 (trifluoroacetate salt)
Dnp-Gly-Pro-Leu-Gly-Met-Arg-Gly-Leu-NH2, Matrix Metalloproteinase-13 Substrate, MMP-13 Substrate
Dnp-GPLGMRGL-NH2 is a peptide substrate for matrix metalloproteinase-13 (MMP-13) with a kcat/Km value of 4,200,000 M-1s-1. -
GC43544
Dnp-P-Cha-Abu-Cys(Me)-HA-K(Nma)-NH2
Dnp-Pro-Cha-Abu-Cys(Me)-His-Ala-Lys(Nma)-NH2, Matrix Metalloproteinase-1 Fluorogenic Substrate III, MMP-1 Fluorogenic Substrate III
Dnp-P-Cha-Abu-Cys(Me)-HA-K(Nma)-NH2 is a fluorogenic substrate for matrix metalloproteinase-1 (MMP-1) and MMP-9. -
GC43548
Dnp-PLG-Cys(Me)-HA-DArg-NH2 (trifluoroacetate salt)
Dnp-Pro-Leu-Gly-Cys(Me)-His-Ala-DArg-NH2, Matrix Metalloproteinase-1 Substrate II, MMP-1 Substrate II
Dnp-PLG-Cys(Me)-HA-DArg-NH2 is a peptide substrate for matrix metalloproteinase-1 (MMP-1). -
GC43549
Dnp-PLGLWA-DArg-NH2 (trifluoroacetate salt)
Dnp-PLGLWA-DArg-NH2 is a fluorogenic substrate for matrix metalloproteinase-1 (MMP-1), MMP-2, MMP-7, and MMP-9.
-
GC43667
FITC-C6-PLALWAR-Lys(Biotin)-NH2 (trifluoroacetate salt)
FITC-C6-Pro-Leu-Ala-Leu-Trp-Ala-Arg-Lys(Biotin)-NH2, MMP-1/MMP-2/MMP-3 Fluorogenic Substrate
FITC-C6-PLALWAR-Lys(Biotin)-NH2 is a substrate for matrix metalloproteinase-1 (MMP-1), MMP-2, and MMP-3 that can be sequestered by streptavidin via its biotin group. -
GC43668
FITC-C6-YVADAP-K(Dnp) (trifluoroacetate salt)
FITC-C6-Tyr-Val-Ala-Asp-Ala-Pro-Lys(Dnp)-OH
FITC-C6-YVADAP-K(Dnp) is a caspase-1 fluorogenic substrate. -
GC43815
Heptanoyl thio-PC
Thioester analogs of glycerophospholipids, in combination with Ellman's reagent, are convenient colorimetric substrates for the measurement of phospholipase (PL) activity.
-
GC44130
Mca-EVKMDAEF-K(Dnp)-NH2 (ammonium salt)
β-Secretase Fluorogenic Substrate
Mca-EVKMDAEF-K(Dnp)-NH2 is a fluorogenic substrate for β-secretase. -
GC44131
Mca-HQKLVFFA-K(Dnp)-NH2 (trifluoroacetate salt)
α-Secretase Fluorogenic Substrate
Mca-HQKLVFFA-K(Dnp)-NH2 is a fluorogenic substrate for α-secretase. -
GC90559
Mca-KPLGL-Dap(Dnp)-AR-NH2 (trifluoroacetate salt)
A fluorogenic substrate for MMPs
-
GC40120
Mca-LEVDGW-K(Dnp)-NH2 (trifluoroacetate salt)
Mca-Leu-Glu-Val-Asp-Gly-Trp-Lys(Dnp)-NH2
Mca-LEVDGW-K(Dnp)-NH2 is a fluorogenic substrate for caspase-4. -
GC47605
Mca-P-Cha-G-Nva-HA-Dap(Dnp)-NH2 (trifluoroacetate salt)
Mca-Pro-Cha-Gly-Nva-His-Ala-Dap(DNP)-NH2
A neuropeptide with diverse biological activities -
GC44133
Mca-PLA-Nva-Dap(Dnp)-AR-NH2 (trifluoroacetate salt)
Matrix Metalloproteinase-2 Fluorogenic Substrate, Mca-Pro-Leu-Ala-Nva-Dap(Dnp)-Ala-Arg-NH2, MMP-2 Fluorogenic Substrate
Mca-PLA-Nva-Dap(Dnp)-AR-NH2 is a fluorogenic substrate for matrix metalloproteinase-2 (MMP-2). -
GC47606
Mca-PLGL-Dap(Dnp)-AR-NH2 (trifluoroacetate salt)
Mca-Pro-Leu-Gly-Leu-Dap(Dnp)-Ala-Arg-NH2, 7-Methoxycoumarin-4-acetyl-P-L-G-L-β-(2,4-dinitrophenylamino)A-R amide
A neuropeptide with diverse biological activities -
GC44134
Mca-PLGL-Dpa-AR-NH2 (trifluoroacetate salt)
Matrix Metalloproteinase-2/Matrix Metalloproteinase-7 Fluorogenic Substrate, Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2, MMP-2/MMP-7 Fluorogenic Substrate
Mca-PLGL-Dpa-AR-NH2 is a fluorogenic substrate for matrix metalloproteinase-2 (MMP-2) and MMP-7. -
GC90538
Mca-RPPGFSAFK(Dnp)-OH (trifluoroacetate salt)
A fluorogenic substrate for ECE-1
-
GC44135
Mca-VDQMDGW-K(Dnp)-NH2 (ammonium salt)
Caspase-3 Fluorogenic Substrate V
Mca-VDQMDGW-K(Dnp)-NH2 is a substrate for caspase-3. -
GC47607
Mca-YVADAP-K(Dnp)-OH (trifluoroacetate salt)
Caspase-1 Fluorogenic Substrate V, Mca-Tyr-Val-Ala-Asp-Ala-Pro-Lys(DNP)-OH, Mca-YVADAP-Lys(Dnp)-OH, (7-Methoxycoumarin-4-yl)acetyl-YVADAPK(2,4-dinitrophenyl)-OH
A neuropeptide with diverse biological activities -
GC90529
Myelin Basic Protein Peptide (mouse, bovine) (trifluoroacetate salt)
A peptide substrate for PKC
-
GC45531
N-α-Benzoyl-L-Arginine ethyl ester (hydrochloride)
BAEE, Bz-Arg-OEt, NSC 86159
-
GC48415
N-Cbz-Gly-Pro-Gly-Gly-Pro-Ala-OH (trifluoroacetate salt)
N-ZGPGGPA-OH
-
GC10797
N1,N11-Diethylnorspermine tetrahydrochloride
spermidine/spermine N1-acetyltransferase inducer
-
GC47947
Phenolphthalein β-D-Glucuronide (hydrate)
Phenolphthalein β-Glucuronide
A neuropeptide with diverse biological activities -
GC16503
Phospho-Glycogen Synthase Peptide-2 (substrate)
substrate for glycogen synthase kinase-3 (GSK-3)
-
GC44936
Sphingosine-1-Phosphate Lyase Fluorogenic Substrate
RBM13, S1P Lyase Fluorogenic Substrate
S1P lyase fluorogenic substrate is a substrate of S1P lyase, leading to the production of the fluorescent product umbelliferone (7-hydroxycoumarin) under appropriate conditions. -
GC45572
Suc-YVAD-pNA
Caspase-1 and Caspase-4 Chromogenic Substrate, Suc-Tyr-Val-Ala-Asp-p-nitroanilide
-
GC45036
Thioarginine (hydrobromide)
L-Arginine serves as a common substrate for both nitric oxide synthase (NOS) and arginase in the cell.
-
GC48390
Z-LRGG-AMC (trifluoroacetate salt)
Z-Leu-Arg-Gly-Gly-AMC, Z-Leu-Arg-Gly-Gly-7-amino-4-methylcoumarin
-
GC45190
Z-VDVAD-AFC (trifluoroacetate salt)
Z-Val-Asp-Val-Ala-Asp-AFC, Z-Val-Asp-Val-Ala-Asp-7-amino-4-trifluormethylcoumarin
Z-VDVAD-AFC is a fluorogenic substrate for caspase-2. -
GC45191
Z-VDVAD-pNA (trifluoroacetate salt)
Z-VDVAD-p-nitroanilide, Z-Val-Asp-Val-Ala-Asp-pNA, Z-Val-Asp-Val-Ala-Asp-p-nitroanilide
Z-VDVAD-pNA is a colorimetric substrate for caspase-2. -
GC40150
Z-VEID-AFC (trifluoroacetate salt)
Z-Val-Glu-Ile-Asp-AFC, Z-Val-Glu-Ile-Asp-7-amino-4-trifluormethylcoumarin
Z-VEID-AFC is a fluorogenic substrate for caspase-6. -
GC40153
Z-YVAD-AFC (trifluoroacetate salt)
Z-Tyr-Val-Ala-Asp-AFC, Z-Tyr-Val-Ala-Asp-7-amino-4-trifluoromethylcoumarin, Z-YVAD-7-amino-4-trifluoromethylcoumarin
Z-YVAD-AFC is a fluorogenic substrate for caspase-1.