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Cancer Biology

Products for  Cancer Biology

  1. Cat.No. Nombre del producto Información
  2. GC47054 CAY10748 A STING agonist CAY10748  Chemical Structure
  3. GC47064 CAY10770 An inhibitor of CYP4Z1 CAY10770  Chemical Structure
  4. GC47066 CAY10777 An antiproliferative agent CAY10777  Chemical Structure
  5. GC91432 CAY10799

    Di-tert-butyl (((S)-1-(tert-butoxy)-3-(4-hydroxyphenyl)-1-oxopropan-2-yl)carbamoyl)-L-glutamate

    CAY10799 es un precursor en la síntesis de ligandos y sondas fluorescentes del antígeno de membrana específico de próstata (PSMA) que se han utilizado en la detección de PSMA en células LNCaP y PC3.

    CAY10799  Chemical Structure
  6. GC43207 Caylin-1 Nutlin-3 is an activator of p53 that functions by inhibiting the interaction of p53 with MDM2, a negative regulator of p53 activity. Caylin-1  Chemical Structure
  7. GC43208 Caylin-2 Nutlin-3 is an activator of p53 that functions by inhibiting the interaction of p53 with MDM2, a negative regulator of p53 activity. Caylin-2  Chemical Structure
  8. GC49664 CB-1158

    INCB 01158, Numidargistat

    An arginase inhibitor CB-1158  Chemical Structure
  9. GP10098 Cdk2/Cyclin Inhibitory Peptide I

    H2N-Tyr-Gly-Arg-Lys-Lys-Arg-Arg-Gln-Arg-Arg-Arg-Gly-Pro-Val-Lys-Arg-Arg-Leu-Phe-Gly-OH

    Cdk2/Cyclin Inhibitory Peptide I  Chemical Structure
  10. GC16722 CE3F4 CE3F4 es un antagonista selectivo de la proteÍna de intercambio activada directamente por cAMP (Epac1), con IC50 de 10,7 μM y 66 μM para Epac1 y Epac2(B), respectivamente. CE3F4  Chemical Structure
  11. GC65347 Ceanothic acid El Ácido ceanÓtico (Ácido emÓlico) es un homÓlogo del anillo A del Ácido betulÍnico. El Ácido ceanÓtico inhibe las células OVCAR-3, HeLa y FS-5 con una supervivencia celular del 68 %, 65 % y 81 %, respectivamente. Ceanothic acid  Chemical Structure
  12. GC45716 Cerevisterol Cerevisterol es un esteroide aislado de los cuerpos fructÍferos de Agaricus blazei. Cerevisterol  Chemical Structure
  13. GC43244 Chlorin e6

    Ce6

    Chlorin e6 (Ce6) es un fotosensibilizador de segunda generación. Chlorin e6  Chemical Structure
  14. GC91297 Cholesterol-Doxorubicin

    Una forma de prodroga de doxorrubicina.

    Cholesterol-Doxorubicin  Chemical Structure
  15. GC43258 Cholesteryl Hemisuccinate

    Cholesteryl hydrogen succinate

    Cholesteryl Hemisuccinate is an acidic cholesterol ester with hepatoprotective and anticancer activities. Cholesteryl Hemisuccinate  Chemical Structure
  16. GC18290 Chrysomycin A

    Albacarcin V, NSC 613946, Virenomycin V

    Chrysomycin A is an antibiotic isolated from a strain of Streptomyces. Chrysomycin A  Chemical Structure
  17. GC12948 CID-1067700

    ML-282

    CID-1067700 (ML282) es un inhibidor de pan GTPasa e inhibe competitivamente el Ras relacionado en el cerebro 7 (Rab7) con una Ki de 13 nM. CID-1067700  Chemical Structure
  18. GC41578 cis-10-Heptadecenoic Acid

    (Z)-Heptadec-10-enoic acid

    cis-10-Heptadecenoic acid is a C17:1 monounsaturated fatty acid that is a minor constituent of ruminant fats.

    cis-10-Heptadecenoic Acid  Chemical Structure
  19. GC41587 cis-Vaccenic Acid

    C18:1 n-7, C18:1(11Z), cis-11-Octadecenoic Acid

    El Ácido cis-vaccénico, el extracto antiviral del capsulato de Rhodopseudomonas y el componente activo predominante del capsulato de Rhodopseudomonas, actÚa como un potencial inductor de la hemoglobina fetal. cis-Vaccenic Acid  Chemical Structure
  20. GC52367 Citrullinated Vimentin (G146R) (R144 + R146) (139-159)-biotin Peptide

    Biotin-GQGKS(Cit)L(Cit)DLYEEEMRELRRQ, Biotin-GQGKSXLXDLYEEEMRELRRQ (X=Citrulline), Citrullinated VIM (G146R) (R144 + R146)-biotin

    A biotinylated and citrullinated mutant vimentin peptide Citrullinated Vimentin (G146R) (R144 + R146) (139-159)-biotin Peptide  Chemical Structure
  21. GC52370 Citrullinated Vimentin (R144) (139-159)-biotin Peptide

    Biotin-GQGKS(Cit)LGDLYEEEMRELRRQ, Biotin-GQGKSXLGDLYEEEMRELRRQ (X=Citrulline), Citrullinated VIM (R144)-biotin

    A biotinylated and citrullinated vimentin peptide Citrullinated Vimentin (R144) (139-159)-biotin Peptide  Chemical Structure
  22. GC47109 Clotrimazole-d5 An internal standard for the quantification of clotrimazole Clotrimazole-d5  Chemical Structure
  23. GC47117 Colchicine-d6 La colchicina-d6 es la colchicina marcada con deuterio. La colchicina es un inhibidor de la tubulina y un agente disruptor de los microtÚbulos. La colchicina inhibe la polimerizaciÓn de microtÚbulos con una IC50 de 3 nM. La colchicina también es un antagonista competitivo de los receptores de glicina α3 (GlyR). Colchicine-d6  Chemical Structure
  24. GC43299 Collismycin A

    SF 2738A

    Collismycin A is a bacterial metabolite originally isolated from Streptomyces that has diverse biological activities, including antibacterial, antiproliferative, and neuroprotective properties. Collismycin A  Chemical Structure
  25. GC52018 COTC

    2-Crotonyloxymethyl-(4R,5R,6R)-4,5,6-trihydroxycyclohex-2-enone

    A bacterial metabolite with anticancer activity COTC  Chemical Structure
  26. GC49569 CP 226,269 A dopamine D4 receptor agonist CP 226,269  Chemical Structure
  27. GC49059 CP94

    CGP 46700, 1,2-Diethyl-3-hydroxypyridin-4-one, EL1Net, 1,2-diethyl HP

    An iron chelator CP94  Chemical Structure
  28. GC62215 CRT0273750 CRT0273750 es un inhibidor de la autotaxina (ATX) y modula los niveles de LPA en plasma (IC50 = 0,014 μM). CRT0273750 se puede utilizar en modelos de cÁncer dependientes de ATX/LPA. CRT0273750  Chemical Structure
  29. GC49557 Cu-GTSM

    CuII(gtsm), copper-GTSM

    A copper-containing compound with diverse biological activities Cu-GTSM  Chemical Structure
  30. GC47137 Cy5-SE (triethylamine salt)

    Sulfo-Cy5

    La sal de trietilamina Cy5-SE (Cy5 NHS Ester) es un colorante reactivo para el etiquetado de grupos amino en péptidos, proteínas y oligonucleótidos. Cy5-SE (triethylamine salt)  Chemical Structure
  31. GP10048 Cyclin D1

    H2N-Leu-Leu-Gly-Ala-Thr-Cys-Met-Phe-Val-OH

    G1/S-specific cyclin-D1 (H2N-Leu-Leu-Gly-Ala-Thr-Cys-Met-Phe-Val-OH) is a protein that in humans is encoded by the CCND1 gene. Cyclin D1  Chemical Structure
  32. GP10038 Cyclin dependent kinase inhibitor 2A - Tumor Suppressor

    H2N-Met-Val-Arg-Arg-Phe-Leu-Val-Thr-Leu-Arg-Ile-Arg-Arg-Ala-Cys-Gly-Pro-Pro-Arg-Val-OH

    Cyclin dependent kinase inhibitor 2A (CDKN2A, p16Ink4A) (H2N-Met-Val-Arg-Arg-Phe-Leu-Val-Thr-Leu-Arg-Ile-Arg-Arg-Ala-Cys-Gly-Pro-Pro-Arg-Val-OH), also known as multiple tumor suppressor 1 (MTS-1), is a tumor suppressor protein, which in humans is encoded by the CDKN2A gene.

    Cyclin dependent kinase inhibitor 2A - Tumor Suppressor  Chemical Structure
  33. GC43342 Cyclo(L-Leu-L-Pro)

    Maculosin 6

    Cyclo(L-Leu-L-Pro) is a diketopiperazine metabolite that has been isolated from various bacterial and fungal species including Streptomyces. Cyclo(L-Leu-L-Pro)  Chemical Structure
  34. GC49707 Cyclo(RGDfC) (trifluoroacetate salt)

    c(RGDfC), cyclo(Arg-Gly-Asp-D-Phe-Cys)

    A cyclic pentapeptide Cyclo(RGDfC) (trifluoroacetate salt)  Chemical Structure
  35. GC49709 cyclo(RGDyC) (trifluoroacetate salt)

    c(RGDyC), cyclo(Arg-Gly-Asp-D-Tyr-Cys)

    A cyclic pentapeptide cyclo(RGDyC) (trifluoroacetate salt)  Chemical Structure
  36. GP10143 Cytochrome c - pigeon (88-104)

    H2N-Lys-Ala-Glu-Arg-Ala-Asp-Leu-Ile-Ala-Tyr-Leu-Lys-Gln-Ala-Thr-Ala-Lys-OH

    Cytochrome c - pigeon (88-104)  Chemical Structure
  37. GP10007 Cytochrome c fragment (93-108)

    H2N-Ala-Asn-Glu-Arg-Ala-Asp-Leu-Ile-Ala-Tyr-Leu-Lys-Gln-Ala-Thr-Lys-OH

    Initiates apoptosis

    Cytochrome c fragment (93-108)  Chemical Structure
  38. GP10141 Cytochrome P450 CYP1B1 (190-198) [Homo sapiens]

    H2N-Phe-Leu-Asp-Pro-Arg-Pro-Leu-Thr-Val-OH

    Cytochrome P450 CYP1B1 (190-198) [Homo sapiens]  Chemical Structure
  39. GC43361 Cytostatin (sodium salt) Cytostatin is a natural antitumor inhibitor of cell adhesion to extracellular matrix, blocking adhesion of B16 melanoma cells to laminin and collagen type IV in vitro (IC50s = 1.3 and 1.4 μg/ml, respectively) and B16 cells metastatic activity in mice. Cytostatin (sodium salt)  Chemical Structure
  40. GC91419 CYY292

    CYY292 es un inhibidor de PDGFRα, PDGFRβ, FGFR1, -2 y -3 (IC50s = 5.35, 4.6, 28, 28 y 78 nM respectivamente).

    CYY292  Chemical Structure
  41. GC43368 D,L-1′-Acetoxychavicol Acetate

    ACA, 1'-Acetoxychavicol Acetate, Galangal Acetate

    D,L-1′-Acetoxychavicol acetate is a natural compound first isolated from the rhizomes of ginger-like plants. D,L-1′-Acetoxychavicol Acetate  Chemical Structure
  42. GC43504 D-myo-Inositol-1,2,3,4,5,6-hexaphosphate (sodium salt)

    IP6, Phytic Acid

    El Ácido fÍtico (hexafosfato de inositol) hexasÓdico es un compuesto de almacenamiento de fÓsforo de semillas y granos de cereales. D-myo-Inositol-1,2,3,4,5,6-hexaphosphate (sodium salt)  Chemical Structure
  43. GC47168 Daidzein-d4 An internal standard for the quantification of daidzein Daidzein-d4  Chemical Structure
  44. GC60121 Dasatinib D8

    Sprycel-d8

    Dasatinib D8 es un Dasatinib marcado con deuterio. Dasatinib es un inhibidor dual de la tirosina quinasa de la familia Bcr-Abl y Src. Dasatinib D8  Chemical Structure
  45. GC48581 Daunorubicinone

    (+)-Daunomycinone, NSC 109531

    An aglycone form of daunorubicin Daunorubicinone  Chemical Structure
  46. GC40697 DDA

    Decadienealdehyde, trans2,4Decadien1al

    DDA es un producto de peroxidaciÓn lipÍdica del Ácido linoleico. DDA  Chemical Structure
  47. GC43390 Deacetylravidomycin Deacetylravidomycin is a microbial metabolite that has been found in Streptomyces and has light-dependent antibiotic and anticancer activities. Deacetylravidomycin  Chemical Structure
  48. GC43391 Decanoic Acid (sodium salt)

    C10:0, Capric Acid, Decylic Acid

    Decanoic acid is a saturated medium-chain fatty acid that contains 10 carbons. Decanoic Acid (sodium salt)  Chemical Structure
  49. GC45815 Decanoic Acid-d19

    Capric Acid-d19, Decylic Acid-d19

    An internal standard for the quantification of decanoic acid Decanoic Acid-d19  Chemical Structure
  50. GC46127 Decanoic Acid-d2

    C10:0-d2, Capric Acid-d2, Decylic Acid-d2

    An internal standard for the quantification of decanoic acid Decanoic Acid-d2  Chemical Structure
  51. GC45722 Decanoic Acid-d3

    Capric Acid-d3, Decylic Acid-d3

    An internal standard for the quantification of decanoic acid Decanoic Acid-d3  Chemical Structure
  52. GC40230 Deferasirox-d4 Deferasirox-d4 es el deuterio etiquetado como Deferasirox. El deferasirox (ICL 670) es un quelante de hierro disponible por vÍa oral que se utiliza para el tratamiento de la sobrecarga transfusional de hierro. Deferasirox-d4  Chemical Structure
  53. GC52316 Deferitrin

    GT-56-252, (S)-4'-Hydroxydesazadesferrithiocin

    An iron chelator and derivative of desferrithiocin Deferitrin  Chemical Structure
  54. GC43407 Demethylwedelolactone Demethylwedelolactone (DWL) is a coumestan, originally isolated from E. Demethylwedelolactone  Chemical Structure
  55. GC40654 Deoxyviolacein Deoxyviolacein is a bacterial metabolite and byproduct in the biosynthesis of the bisindole alkaloid violacein that has anticancer, antibacterial, and antifungal properties. Deoxyviolacein  Chemical Structure
  56. GC47211 Dichlorvos

    DDVP, Dichlorovinyl Dimethyl Phosphate, NSC 6738

    An organophosphate insecticide Dichlorvos  Chemical Structure
  57. GC49293 Dichlorvos-d6

    DDVP-d6, Dichlorovinyl Dimethyl Phosphate-d6

    An internal standard for the quantification of dichlorvos Dichlorvos-d6  Chemical Structure
  58. GC47215 Dienogest-d8 An internal standard for the quantification of dienogest Dienogest-d8  Chemical Structure
  59. GC52194 Dimethylamino Parthenolide

    DMAPT, LC-1

    Dimethylamino Parthenolide  Chemical Structure
  60. GC74493 Dinutuximab

    Unituxin; APN-311

    Dinutuximab (Unituxin; APN-311) es un anticuerpo monoclonal anti-GD2 quimérico, human-murina. Dinutuximab  Chemical Structure
  61. GC49383 DL-Phenyl-d5-alanine

    (±)-Phenyl-d5-alanine

    An internal standard for the quantification of DL-phenylalanine DL-Phenyl-d5-alanine  Chemical Structure
  62. GC18254 DM1-SMe DM1-SMe es una forma no conjugada del maytansinoide en IMGN901. DM1-SMe es aproximadamente 3 a 10 veces mÁs potente que el fÁrmaco original Maytansine, con IC50 que van desde 0,003 a 0,01 nM para DM1-SMe en un panel de lÍneas de células tumorales humanas. DM1-SMe  Chemical Structure
  63. GC48968 Docetaxel (hydrate)

    DTX, NSC 628503, RP 56976, Taxotel

    An analog of taxol with antitumor properties

    Docetaxel (hydrate)  Chemical Structure
  64. GC47250 Docetaxel-d9

    DTX-d9, Taxotel-d9

    Docetaxel-d9 (RP-56976-d9) es el docetaxel etiquetado con deuterio. Docetaxel (RP-56976) es un inhibidor de la despolimerizaciÓn de microtÚbulos, con una IC50 de 0,2 μM. Docetaxel atenÚa los efectos de la expresiÓn de los genes bcl-2 y bcl-xL. Docetaxel detiene el ciclo celular en G2/M y conduce a la apoptosis celular. El docetaxel tiene actividad anticancerÍgena. Docetaxel-d9  Chemical Structure
  65. GC74603 Domvanalimab

    AB154

    Domvanalimab (AB154) es un anticuerpo monoclonal humanizado anti-TIGIT. Domvanalimab  Chemical Structure
  66. GC43565 Doxorubicinol (hydrochloride)

    13-Dihydroadriamycin hydrochloride

    Doxorubicinol is the major metabolite of doxorubicin, an anthracycline antitumor antibiotic that inhibits DNA topoisomerase II by inducing double-stranded DNA breaks. Doxorubicinol (hydrochloride)  Chemical Structure
  67. GC40082 Drimentine B Drimentine B is a terpenylated diketopiperazine antibiotic originally isolated from Actinomycete bacteria. Drimentine B  Chemical Structure
  68. GC43573 Drimentine C Drimentine C is a terpenylated diketopiperazine antibiotic originally isolated from Actinomycete bacteria. Drimentine C  Chemical Structure
  69. GC49001 DSPE-PEG(2000)-amine (sodium salt) A PEGylated derivative of DSPE DSPE-PEG(2000)-amine (sodium salt)  Chemical Structure
  70. GC91884 DSPE-PEG(2000)-Mannose

    1,2-Distearoyl-sn-glycero-3-PE-Polyethylene Glycol-2000-Mannose; 1,2-Distearoyl-sn-glycero-3-Phosphoethanolamine-Polyethylene Glycol-2000-Mannose; 1,2-DSPE-PEG(2000)-Mannose

    DSPE-PEG(2000)-Mannose se ha utilizado en la generación de liposomas y micelas mixtas para la administración de agentes anticancerosos a los macrófagos asociados a tumores TAMs in vitro e in vivo. DSPE-PEG(2000)-Mannose  Chemical Structure
  71. GC52333 DSPE-PEG(2000)-NHS

    DSPE-PEG(2000)-NHS is a PEGylated derivative of 1,2-distearoyl-sn-glycero-3-PE .

    DSPE-PEG(2000)-NHS  Chemical Structure
  72. GC26427 DSPE-PEG2000-Mal ammonium

    Poly(oxy-1,2-ethanediyl), α-[(9R)-6-hydroxy-6-oxido-1,12-dioxo-9-[(1-oxooctadecyl)oxy]-5,7,11-trioxa-2-aza-6-phosphanonacos-1-yl]-ω-[2-[[3-(2,5-dihydro-2,5-dioxo-1H-pyrrol-1-yl)-1-oxopropyl]amino]ethoxy]-, ammonium salt (1:1)

    DSPE-PEG2000-Mal ammonium  Chemical Structure
  73. GC49058 DTPA

    Diethylenetriaminepentaacetic Acid, NSC 7340, Pentetic Acid

    El DTPA es un compuesto que se utiliza para construir un adsorbente magnético que puede eliminar simultÁneamente metales pesados y colorantes de aguas residuales complejas. DTPA  Chemical Structure
  74. GC18992 Duclauxin

    NSC 258308

    Duclauxin decreases proliferation of tumor cells in vitro and increases the lifespan of mice innoculated with Ehrlich ascitic tumor cells. Duclauxin  Chemical Structure
  75. GP10022 Dynamin inhibitory peptide

    Gln-Val-Pro-Ser-Arg-Pro-Asn-Arg-Ala-Pro

    Dynamin inhibitory peptide  Chemical Structure
  76. GC65123 Eclalbasaponin I Eclalbasaponin I se aÍsla de Eclipta prostrata L con actividad antitumoral. La eclalbasaponina I inhibe la proliferaciÓn de células de hepatoma smmc-7721 con un valor IC50 de 111,1703 μg/ml. Eclalbasaponin I  Chemical Structure
  77. GP10030 EGF receptor substrate eps15 acetyl - [Mus musculus]/[Homo sapiens]

    Ac-Gln-Glu-Gln-Glu-Asp-Leu-Glu-Leu-Ala-Ile-Ala-Leu-Ser-Lys-Ser-Glu-Ile-Ser-Glu-Ala-OH

    EGF receptor substrate eps15 (Eps15) has been identified as a 142-kDa substrate of the EGF receptor1. EGF receptor substrate eps15 acetyl - [Mus musculus]/[Homo sapiens]  Chemical Structure
  78. GP10108 EGF-R (661-681) T669 Peptide

    H2N-Lys-Arg-Glu-Leu-Val-Glu-Pro-Leu-Thr-Pro-Ser-Gly-Glu-Ala-Pro-Asn-Gln-Ala-Leu-Leu-Arg-OH

    EGF-R (661-681) T669 Peptide  Chemical Structure
  79. GC43591 Eicosapentaenoyl 1-propanol-2-amide Monoacylglycerols (MAGs) of ω-3 polyunsaturated fatty acids have diverse physiological and health effects. Eicosapentaenoyl 1-propanol-2-amide  Chemical Structure
  80. GC49522 EM-12

    EM-12

    EM-12 (EM-12), un anÁlogo de talidomida teratogénico, es mÁs activo que la talidomida y es mucho mÁs estable para la hidrÓlisis. EM-12 mejora la inducciÓn de 1,2-dimetilhidrazina de adenocarcinomas de colon de rata. EM-12  Chemical Structure
  81. GC46137 Emestrin A mycotoxin Emestrin  Chemical Structure
  82. GC49124 EN219 EN219 es un ligando covalente sintético moderadamente selectivo frente a una cisteÍna N-terminal (C8) de RNF114 con una IC50 de 470 nM. EN219 inhibe la autoubiquitinaciÓn mediada por RNF114 y la ubiquitinaciÓn de p21. EN219  Chemical Structure
  83. GP10117 Endostatin (84-114)-NH2 (JKC367)

    H2N-Pro-Gly-Ala-Arg-Ile-Phe-Ser-Phe-Asp-Gly-Lys-Asp-Val-Leu-Arg-His-Pro-Thr-Trp-Pro-Gln-Lys-Ser-Val-Trp-His-Gly-Ser-Asp-Pro-Asn-NH2

    Endostatin (84-114)-NH2 (JKC367)  Chemical Structure
  84. GC43606 Endothelin-1 (human, porcine) (trifluoroacetate salt)

    ET-1

    Endothelin-1 is a peptide vasoconstrictor and agonist of endothelin (ET) receptors ETA and ETB (IC50s = 0.15 and 0.12 nM, respectively). Endothelin-1 (human, porcine) (trifluoroacetate salt)  Chemical Structure
  85. GC49648 Enobosarm-d4

    (S)-Enobosarm-d4

    An internal standard for the quantification of enobosarm Enobosarm-d4  Chemical Structure
  86. GC48664 Enoxacin-d8 (hydrochloride) Enoxacin-d8 (hydrochloride)  Chemical Structure
  87. GC47297 EP4 Receptor Antagonist 1 El antagonista del receptor EP4 1 es un antagonista competitivo del receptor prostanoide EP4 muy potente y selectivo para la inmunoterapia contra el cÁncer. EP4 Receptor Antagonist 1  Chemical Structure
  88. GP10005 Epidermal growth factor receptor (994-1002) acetyl/amide

    Ac-Asp-Ser-Asn-Phe-Tyr-Arg-Ala-Leu-Met-amide

    EGF-family receptor

    Epidermal growth factor receptor (994-1002) acetyl/amide  Chemical Structure
  89. GP10095 Epidermal Growth Factor Receptor Peptide (985-996)

    H2N-Asp-Val-Val-Asp-Ala-Asp-Glu-Tyr-Leu-Ile-Pro-Gln-OH

    Epidermal Growth Factor Receptor Peptide (985-996)  Chemical Structure
  90. GC72845 Epoetin beta

    rhEPO; EPOCH; Genetical recombination

    Epoetin β (rhEPO) es una forma recombinante de eritropoyetina. Epoetin beta  Chemical Structure
  91. GP10132 erbB-2

    H2N-Lys-Ile-Phe-Gly-Ser-Leu-Ala-Phe-Leu-OH

    erbB-2  Chemical Structure
  92. GC90653 ERX-41

    Un inductor de estrés del ER (retículo endoplásmico).

    ERX-41  Chemical Structure
  93. GC52303 Ethyl Mycophenolate A potential impurity found in commercial preparations of mycophenolate mofetil Ethyl Mycophenolate  Chemical Structure
  94. GC74618 Etigilimab

    OMP-313M32

    Etigilimab (OMP-313M32), un anticuerpo monoclonal IgG1 humanizado, bloquea la interacción del TIGIT con PVR (CD155; Poliovirus) e inhila la señalización posterior con la destrucción de la célula diana. Etigilimab  Chemical Structure
  95. GC15555 Farnesyl Thiosalicylic Acid Amide

    FTS Amide,Salirasib Amide

    inhibits tumor growth

    Farnesyl Thiosalicylic Acid Amide  Chemical Structure
  96. GP10123 Fas C- Terminal Tripeptide

    Ac-Ser-Leu-Val-OH

    Fas C- Terminal Tripeptide  Chemical Structure
  97. GC60833 FB23 FB23 es un inhibidor potente y selectivo de la FTO desmetilasa con una IC50 de 60 nM. FB23 se une directamente a FTO e inhibe selectivamente la actividad desmetilasa del ARNm N6-metiladenosina (m6A) de FTO. FB23  Chemical Structure
  98. GC46146 FD-211

    (-)-Waol A

    A δ lactone with anticancer activity FD-211  Chemical Structure
  99. GC49563 Fenhexamid

    KBR 2738

    Fenhexamid, un botryticida, es un inhibidor de la biosÍntesis de esteroles. Fenhexamid  Chemical Structure
  100. GP10146 ferritin heavy chain fragment [Multiple species]

    H2N-Tyr-Leu-Asn-Glu-Gln-Val-Lys-Ala-Ile-OH

    ferritin heavy chain fragment [Multiple species]  Chemical Structure
  101. GC39811 FIT-039 FIT-039 es un inhibidor de CDK9 selectivo, competitivo con ATP y activo por vÍa oral con una IC50 de 5,8 μM para CKD9/ciclina T1. FIT-039  Chemical Structure

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