TC AC 28 |
| Catalog No.GC50340 |
High affinity BET bromodomain ligand
Products are for research use only. Not for human use. We do not sell to patients.
Cas No.: 1809296-92-1
Sample solution is provided at 25 µL, 10mM.
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High affinity BET bromodomain ligand (Kd values are 40 and 800 nM for Brd2(2) and Brd2(1), respectively). Exhibits 20-fold selectively for the second over the first bromodomain.
Baud et al (2016) New synthetic routes to triazolo-benzodiazepine analogues: expanding the scope of the bump-and-hole approach for selective bromo and extra-terminal (BET) bromodomain inhibition. J.Med.Chem. 59 1492 PMID:26367539
Average Rating: 5 (Based on Reviews and 7 reference(s) in Google Scholar.)
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