L2H2-6OTD intermediate-1 is an intermediate for the synthesis of L2H2-6OTD and can be used for ADC preparation. L2H2-6OTD, a telomestatin analog with telomerase inhibitory activity (IC50: 15 nM).
References:
[1]. Doi Takayuki, et al. Total Synthesis of (R)-Telomestatin. Organic Letters (2006), 8(18), 4165-4167. [2]. Kazuaki Shibata, et al. Synthesis of Heptaoxazole Macrocyclic Analogues of Telomestatin. Chem. Soc. Jpn. Vol. 86, No. 12, 14531465