Drug Metabolite
Drug metabolite results when a drug is metabolized into a modified form which continues to produce effects. Drug metabolism redox reactions such as heteroatom dealkylations, hydroxylations, heteroatom oxygenations, reductions, and dehydrogenations can yield active metabolites, and in rare cases even conjugation reactions can yield an active metabolite.
Products Related to Drug Metabolite(546)
- GC49399N-Desbutyl Dronedarone (hydrochloride)CAS: 197431-02-0Purity: >95.00%
ديبوتيلدرونيدارون (SR35021) هيدروكلوريد ، المستقلب الرئيسي للدرونيدارون ، هو مستقبل هرمون الغدة الدرقية الانتقائي α ؛ 1 (TRα ؛ 1) مثبط.
- GC49406ACT-373898CAS: 1433875-14-9Purity: >90.00%
ACT-373898 هو مستقلب حمض الكربوكسيل غير النشط لماسيتينتان
- GC49421Atorvastatin lactone-d5CAS: 125995-03-1Purity: >99.00%
An internal standard for the quantification of atorvastatin lactone
- GC49428O-Des[2-aminoethyl]-O-carboxymethyl dehydroamlodipineCAS: 113994-45-9Purity: >95.00%
A major metabolite of amlodipine
- GC49480Salicylic Acid-d4CAS: 78646-17-0Purity: >98.00%
حمض الساليسيليك- d4 هو الديوتيريوم المسمى 2-كاربوكسيفينول.
- GC494886-Methylmercaptopurine-d3CAS: 33312-93-5Purity: >99.00%
An internal standard for the quantification of 6-MMP
- GC49559Hydroxymethyl Tolperisone (hydrochloride)CAS: 352233-14-8Purity: >95.00%
A metabolite of tolperisone
- GC49565RoxatidineCAS: 78273-80-0Purity: >95.00%
Roxatidine هو مستقلب نشط من Roxatidine acetate hydrochloride ، وهو مضاد مستقبلات الهيستامين H2
- GC49583N-desmethyl Sertraline (hydrochloride)CAS: 675126-09-7Purity: >95.00%
A metabolite of sertraline
- GC49637O-desethyl DapagliflozinCAS: 864070-37-1Purity: >98.00%
An SGLT2 inhibitor and active metabolite of dapagliflozin
- GC49677Olmesartan-d6CAS: 1185144-74-4Purity: >99.00%
An internal standard for the quantification of olmesartan
- GC49686N-desmethyl Regorafenib N-oxideCAS: 835621-12-0Purity: >90.00%
An active metabolite of regorafenib
| Catalog No. | Product Name | CAS No. | Purity | Structure |
|---|---|---|---|---|
| GC49399 | N-Desbutyl Dronedarone (hydrochloride) | 197431-02-0 | >95.00% | |
ديبوتيلدرونيدارون (SR35021) هيدروكلوريد ، المستقلب الرئيسي للدرونيدارون ، هو مستقبل هرمون الغدة الدرقية الانتقائي α ؛ 1 (TRα ؛ 1) مثبط. | ||||
| GC49403 | Benzarone | 1477-19-6 | >98.00% | |
Benzarone (Fragivix) هو مثبط فعال لنقل حمض اليوريك البشري 1 (hURAT1) ، مع IC 50 من 2.8 ميكرومتر في البويضة | ||||
| GC49406 | ACT-373898 | 1433875-14-9 | >90.00% | |
ACT-373898 هو مستقلب حمض الكربوكسيل غير النشط لماسيتينتان | ||||
| GC49409 | Desmethyl Ranolazine | 172430-45-4 | >95.00% | |
A metabolite of ranolazine | ||||
| GC49410 | CVT-2738 | 5294-61-1 | >98.00% | |
An active metabolite of ranolazine | ||||
| GC49421 | Atorvastatin lactone-d5 | 125995-03-1 | >99.00% | |
An internal standard for the quantification of atorvastatin lactone | ||||
| GC49428 | O-Des[2-aminoethyl]-O-carboxymethyl dehydroamlodipine | 113994-45-9 | >95.00% | |
A major metabolite of amlodipine | ||||
| GC49480 | Salicylic Acid-d4 | 78646-17-0 | >98.00% | |
حمض الساليسيليك- d4 هو الديوتيريوم المسمى 2-كاربوكسيفينول. | ||||
| GC49488 | 6-Methylmercaptopurine-d3 | 33312-93-5 | >99.00% | |
An internal standard for the quantification of 6-MMP | ||||
| GC49501 | Nirvanol | 631-07-2 | >98.00% | |
An active metabolite of mephenytoin | ||||
| GC49511 | Nicorandil N-oxide | 107833-98-7 | >98.00% | |
A metabolite of nicorandil | ||||
| GC49538 | Lamotrigine N2-oxide | 136565-76-9 | >95.00% | |
A metabolite of lamotrigine | ||||
| GC49544 | 8-hydroxy Mirtazapine | 102335-57-9 | >95.00% | |
A metabolite of mirtazapine | ||||
| GC49559 | Hydroxymethyl Tolperisone (hydrochloride) | 352233-14-8 | >95.00% | |
A metabolite of tolperisone | ||||
| GC49565 | Roxatidine | 78273-80-0 | >95.00% | |
Roxatidine هو مستقلب نشط من Roxatidine acetate hydrochloride ، وهو مضاد مستقبلات الهيستامين H2 | ||||
| GC49575 | 4-hydroxy Omeprazole sulfide | 103876-98-8 | >98.00% | |
A metabolite of omeprazole | ||||
| GC49583 | N-desmethyl Sertraline (hydrochloride) | 675126-09-7 | >95.00% | |
A metabolite of sertraline | ||||
| GC49627 | Rabeprazole sulfone | 117976-47-3 | >95.00% | |
A metabolite of rabeprazole | ||||
| GC49629 | 6β-hydroxy Prednisolone | 16355-29-6 | >95.00% | |
A metabolite of prednisolone | ||||
| GC49637 | O-desethyl Dapagliflozin | 864070-37-1 | >98.00% | |
An SGLT2 inhibitor and active metabolite of dapagliflozin | ||||
| GC49655 | 5-hydroxy Buspirone | 105496-33-1 | >95.00% | |
A metabolite of buspirone | ||||
| GC49676 | 6β-hydroxy Budesonide | - | >95.00% | |
A metabolite of budesonide | ||||
| GC49677 | Olmesartan-d6 | 1185144-74-4 | >99.00% | |
An internal standard for the quantification of olmesartan | ||||
| GC49686 | N-desmethyl Regorafenib N-oxide | 835621-12-0 | >90.00% | |
An active metabolite of regorafenib | ||||