San78-130 |
| Catalog No.GC37591 |
Products are for research use only. Not for human use. We do not sell to patients.
Cas No.: 66018-45-9
Sample solution is provided at 25 µL, 10mM.
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San78-130 is a selective and potent ALK1 inhibitor with an IC50 of 62 nM. San78-130 also inhibits FLT4/VEGFR3, KDR/VEGFR2, MEK2, and FLT3 with IC50s of 114, 162, 186.7, and 188 nM, respectively[1]. ALK1|62 nM (IC50)|FLT4/VEGFR3|114 nM (IC50)|KDR/VEGFR2|162 nM (IC50)|MEK2|186.7 nM (IC50)|FLT3|188 nM (IC50)
[1]. Cho H, et al. Identification of the First Selective Activin Receptor-Like Kinase 1 Inhibitor, a Reversible Version of L-783277. J Med Chem. 2017 Feb 23;60(4):1495-1508.
Average Rating: 5 (Based on Reviews and 24 reference(s) in Google Scholar.)
GLPBIO products are for RESEARCH USE ONLY. Please make sure your review or question is research based.
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