3-Amino-5-(2-furyl)pyrazole (Compound 14) is aPDK1binder with anIC50of 313 μM. 3-Amino-5-(2-furyl)pyrazole can be used incancerresearch[1].
References:
[1].Medina JR, et al. Aminoindazole PDK1 Inhibitors: A Case Study in Fragment-Based Drug Discovery. ACS Med Chem Lett. 2010 Jul 22;1(8):439-42.
















