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GPR52 agonist-4

Catalog No.GC81693 Copy One-Click Copy Product Info

GPR52 agonist-4 (Compound 65) is a highly selective G-protein-coupled receptor GPR52 modulator.

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GPR52 agonist-4 Chemical Structure

Cas No.: 1313195-88-8

Size Price Stock Qty
5mg
$149.00
In stock
10mg
$237.00
In stock

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Sample solution is provided at 25 µL, 10mM.



Description of GPR52 agonist-4

GPR52 agonist-4 (Compound 65) is a highly selective G-protein-coupled receptor GPR52 modulator. GPR52 agonist-4 is promising for research of neuropsychiatric diseases [1].

References:
[1]. 正記 瀬藤, et al. Amide compounds. JPWO2011078360A1. 2013-05-09.

Chemical Properties of GPR52 agonist-4

Cas No. 1313195-88-8 SDF
Formula C24H22F3N3O3S M.Wt 489.51
Solubility DMSO: 100 mg/mL (204.29 mM; Need ultrasonic) Storage Store at -20°C
Shipping Condition Evaluation sample solution: shipped with blue ice. All other sizes available: with RT, or with Blue Ice upon request.

Complete Stock Solution Preparation Table of GPR52 agonist-4

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1 mg 5 mg 10 mg
1 mM 2.0429 mL 10.2143 mL 20.4286 mL
5 mM 408.6 μL 2.0429 mL 4.0857 mL
10 mM 204.3 μL 1.0214 mL 2.0429 mL
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In vivo Formulation Calculator (Clear solution) of GPR52 agonist-4

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Method for preparing DMSO master liquid: mg drug pre-dissolved in μL DMSO ( Master liquid concentration mg/mL, Please contact us first if the concentration exceeds the DMSO solubility of the batch of drug. )

Method for preparing in vivo formulation: Take μL DMSO master liquid, next addμL PEG300, mix and clarify, next addμL Tween 80, mix and clarify, next add μL saline, mix and clarify.

Method for preparing in vivo formulation: Take μL DMSO master liquid, next add μL Corn oil, mix and clarify.

Note: 1. Please make sure the liquid is clear before adding the next solvent.
2. Be sure to add the solvent(s) in order. You must ensure that the solution obtained, in the previous addition, is a clear solution before proceeding to add the next solvent. Physical methods such as vortex, ultrasound or hot water bath can be used to aid dissolving.
3. All of the above co-solvents are available for purchase on the GlpBio website.

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Average Rating: 5 ★★★★★ (Based on Reviews and 30 reference(s) in Google Scholar.)

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