GLPBio

BTR2000 TFA

Catalog No.: GC81019Purity:>98.50%
COASDSData Sheet
BTR2000 TFA, a specifically KLHL20 ligand, is capable of binding to the KLHL20 Kelch domain with high affinity.

제품은 연구용으로만 사용됩니다. 인체에 사용할 수 없으며 환자에게 판매하지 않습니다.

BTR2000 TFA
5mgIn Stock
$153.00
1
10mgIn Stock
$245.00
1
Tel: (909) 407-4943 / (909) 689-7124Email: sales@glpbio.com

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제품 설명 (Description)

BTR2000 TFA, a specifically KLHL20 ligand, is capable of binding to the KLHL20 Kelch domain with high affinity. BTR2000 TFA can be used as a ligand for E3 ligase for the synthesis of BTR2004 [1] [2].

References:
[1]. Farrell BM, et, al. A synthetic KLHL20 ligand to validate CUL3KLHL20 as a potent E3 ligase for targeted protein degradation. Genes Dev. 2022 Sep 1;36(17-18):1031-1042.
[2]. Fechtmeyer PH, et, al. Temporal and Spatial Characterization of CUL3KLHL20-driven Targeted Degradation of BET family, BRD Proteins by the Macrocycle-based Degrader BTR2004. bioRxiv. 2024 Dec 7:2024.12.07.627262.

제품 문서 (Product Documents)

Purity:>98.50%Appearance:A solid
COASDSData Sheet

화학적 특성 (Chemical Properties)

분자식
C31H43F3N6O9S2
분자량
764.83
용해도
DMSO: 62.5 mg/mL (81.72 mM; Need ultrasonic)
보관
Store at -20°C
배송 조건
평가용 샘플은 아이스팩과 함께 배송됩니다. 그 외 용량은 실온 배송되며, 요청 시 아이스팩과 함께 배송할 수 있습니다.

계산 도구 (Calculators)몰 농도 / 희석 / 분자량 / 단위 변환 / 생체 내 제형 / 용해도

g/mol

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