SMARCA2/4-IN-2

Name: SMARCA2/4-IN-2
Brand: GlpBio
SKU: GC75800
Availability: InStock

Catalog No.: GC75800Purity:>99.00%

COASDSData Sheet

SMARCA2/4-IN-2 is a PROTAC target protein ligand (Ligands for Target Protein for PROTACs).

Products are for research use only. Not for human use. We do not sell to patients.

Cas No.: 1339378-93-6

5 mgIn Stock

$95.00

10 mgIn Stock

$153.00

25 mgIn Stock

$321.00

50 mgIn Stock

$498.00

Pack Size	Price	Availability	Quantity
5 mg	$95.00	In Stock	1
10 mg	$153.00	In Stock	1
25 mg	$321.00	In Stock	1
50 mg	$498.00	In Stock	1

Tel: (909) 407-4943 / (909) 689-7124Email: sales@glpbio.com

Citations

No citations are currently available for this product. Below are selected publications citing GlpBio products.

Nature
641, 529–536 (2025)
Nature
628, 630–638 (2024)
Nature
632, 686–694 (2024)
Nature
618, 1017–1023 (2023)
Nature
610, 366–372 (2022)
Cell
187(9):2288-2304 (2024)
Cell
183(7):1867-1883 (2020)
Science
388(6745) (2025)
Science
387(6739) (2025)
Science
387(6734) (2025)
Cell Research
35, 97–116 (2025)
Cell Research
34, 683–706 (2024)
Cell Research
33, 273–287 (2023)
Cell Research
33, 546–561 (2023)
Cell Research
33, 904–922 (2023)
Cell Research
31, 1291–1307 (2021)

Description

SMARCA2/4-IN-2 is a PROTAC target protein ligand (Ligands for Target Protein for PROTACs). SMARCA2/4-IN-2 can be used for synthesis PROTAC SMARCA2/4-degrader-5 ^[1].

References:
[1]. Preparation of heterocyclic compounds as SMARCA degraders and uses thereof. USA, US20230072658A1 2020-12-17

Product Documents

Batch:Purity:>99.00%Appearance:A solid

COA SDS Data Sheet

Chemical Properties

CAS No.

1339378-93-6

Molecular Formula

C₁₀H₉N₃O

Molecular Weight

187.2

Solubility

DMSO: 100 mg/mL (534.19 mM; Need ultrasonic)

Storage

-20°C

General tips

Select a suitable solvent according to the product solubility data. Once prepared, aliquot the stock solution to avoid repeated freeze-thaw cycles.
Use stock solutions within 6 months when stored at -80°C or within 1 month when stored at -20°C.
To improve solubility, warm the tube to 37°C and sonicate it for an appropriate period.

Shipping Condition

Evaluation samples are shipped with blue ice. Other available sizes are shipped at room temperature or with blue ice upon request.

CalculatorsMolarity / Dilution / Molecular Weight / Unit Conversion / In Vivo Formulation / Solubility

Mass

Volume

Concentration

Molecular Weight

g/mol

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