Drug Metabolite
Drug metabolite results when a drug is metabolized into a modified form which continues to produce effects. Drug metabolism redox reactions such as heteroatom dealkylations, hydroxylations, heteroatom oxygenations, reductions, and dehydrogenations can yield active metabolites, and in rare cases even conjugation reactions can yield an active metabolite.
Products Related to Drug Metabolite(546)
- GC49399N-Desbutyl Dronedarone (hydrochloride)CAS: 197431-02-0Purity: >95.00%
El clorhidrato de debutildronedarona (SR35021), el principal metabolito de Dronedarona, es un inhibidor selectivo del receptor de la hormona tiroidea α1 (TRα1).
- GC49406ACT-373898CAS: 1433875-14-9Purity: >90.00%
ACT-373898 es un metabolito de Ácido carboxÍlico inactivo de Macitentan.
- GC49421Atorvastatin lactone-d5CAS: 125995-03-1Purity: >99.00%
An internal standard for the quantification of atorvastatin lactone
- GC49428O-Des[2-aminoethyl]-O-carboxymethyl dehydroamlodipineCAS: 113994-45-9Purity: >95.00%
A major metabolite of amlodipine
- GC49480Salicylic Acid-d4CAS: 78646-17-0Purity: >98.00%
El Ácido salicÍlico-d4 es el 2-carboxifenol marcado con deuterio.
- GC494886-Methylmercaptopurine-d3CAS: 33312-93-5Purity: >99.00%
An internal standard for the quantification of 6-MMP
- GC49559Hydroxymethyl Tolperisone (hydrochloride)CAS: 352233-14-8Purity: >95.00%
A metabolite of tolperisone
- GC49565RoxatidineCAS: 78273-80-0Purity: >95.00%
La roxatidina es un metabolito activo del clorhidrato de acetato de roxatidina, es un antagonista del receptor H2 de la histamina.
- GC49583N-desmethyl Sertraline (hydrochloride)CAS: 675126-09-7Purity: >95.00%
A metabolite of sertraline
- GC49637O-desethyl DapagliflozinCAS: 864070-37-1Purity: >98.00%
An SGLT2 inhibitor and active metabolite of dapagliflozin
- GC49677Olmesartan-d6CAS: 1185144-74-4Purity: >99.00%
An internal standard for the quantification of olmesartan
- GC49686N-desmethyl Regorafenib N-oxideCAS: 835621-12-0Purity: >90.00%
An active metabolite of regorafenib
| Catalog No. | Product Name | CAS No. | Purity | Structure |
|---|---|---|---|---|
| GC49399 | N-Desbutyl Dronedarone (hydrochloride) | 197431-02-0 | >95.00% | |
El clorhidrato de debutildronedarona (SR35021), el principal metabolito de Dronedarona, es un inhibidor selectivo del receptor de la hormona tiroidea α1 (TRα1). | ||||
| GC49403 | Benzarone | 1477-19-6 | >98.00% | |
La benzarona (Fragivix) es un potente inhibidor del transportador de Ácido Úrico humano 1 (hURAT1), con una IC50 de 2,8 μM en el ovocito. | ||||
| GC49406 | ACT-373898 | 1433875-14-9 | >90.00% | |
ACT-373898 es un metabolito de Ácido carboxÍlico inactivo de Macitentan. | ||||
| GC49409 | Desmethyl Ranolazine | 172430-45-4 | >95.00% | |
A metabolite of ranolazine | ||||
| GC49410 | CVT-2738 | 5294-61-1 | >98.00% | |
An active metabolite of ranolazine | ||||
| GC49421 | Atorvastatin lactone-d5 | 125995-03-1 | >99.00% | |
An internal standard for the quantification of atorvastatin lactone | ||||
| GC49428 | O-Des[2-aminoethyl]-O-carboxymethyl dehydroamlodipine | 113994-45-9 | >95.00% | |
A major metabolite of amlodipine | ||||
| GC49480 | Salicylic Acid-d4 | 78646-17-0 | >98.00% | |
El Ácido salicÍlico-d4 es el 2-carboxifenol marcado con deuterio. | ||||
| GC49488 | 6-Methylmercaptopurine-d3 | 33312-93-5 | >99.00% | |
An internal standard for the quantification of 6-MMP | ||||
| GC49501 | Nirvanol | 631-07-2 | >98.00% | |
An active metabolite of mephenytoin | ||||
| GC49511 | Nicorandil N-oxide | 107833-98-7 | >98.00% | |
A metabolite of nicorandil | ||||
| GC49538 | Lamotrigine N2-oxide | 136565-76-9 | >95.00% | |
A metabolite of lamotrigine | ||||
| GC49544 | 8-hydroxy Mirtazapine | 102335-57-9 | >95.00% | |
A metabolite of mirtazapine | ||||
| GC49559 | Hydroxymethyl Tolperisone (hydrochloride) | 352233-14-8 | >95.00% | |
A metabolite of tolperisone | ||||
| GC49565 | Roxatidine | 78273-80-0 | >95.00% | |
La roxatidina es un metabolito activo del clorhidrato de acetato de roxatidina, es un antagonista del receptor H2 de la histamina. | ||||
| GC49575 | 4-hydroxy Omeprazole sulfide | 103876-98-8 | >98.00% | |
A metabolite of omeprazole | ||||
| GC49583 | N-desmethyl Sertraline (hydrochloride) | 675126-09-7 | >95.00% | |
A metabolite of sertraline | ||||
| GC49627 | Rabeprazole sulfone | 117976-47-3 | >95.00% | |
A metabolite of rabeprazole | ||||
| GC49629 | 6β-hydroxy Prednisolone | 16355-29-6 | >95.00% | |
A metabolite of prednisolone | ||||
| GC49637 | O-desethyl Dapagliflozin | 864070-37-1 | >98.00% | |
An SGLT2 inhibitor and active metabolite of dapagliflozin | ||||
| GC49655 | 5-hydroxy Buspirone | 105496-33-1 | >95.00% | |
A metabolite of buspirone | ||||
| GC49676 | 6β-hydroxy Budesonide | - | >95.00% | |
A metabolite of budesonide | ||||
| GC49677 | Olmesartan-d6 | 1185144-74-4 | >99.00% | |
An internal standard for the quantification of olmesartan | ||||
| GC49686 | N-desmethyl Regorafenib N-oxide | 835621-12-0 | >90.00% | |
An active metabolite of regorafenib | ||||