GLPBio

EZH2

EZH2 (enhancer of zeste homolog 2) is a polycomb group protein and histone methyltrasferase that associated with transcriptional repression. It catalyzes trimethylation of H3K27me3 (histone H3 lysine 27) as a catalytic subunit of PRC2 (polycomb repressive complex 2).

Products Related to EZH2(10)

  • GC11414 structure
    GC11414GSK503
    CAS: 1346572-63-1
    Purity: >99.50%

    GSK503 هو مثبط قوي ومحدد لـ EZH2 methyltransferase بقيم Kiapp من 3 إلى 27 نانومتر

  • GC13145 structure
    GC131453-Deazaneplanocin,DZNep
    CAS: 102052-95-9
    Purity: >98.00%

    An inhibitor of lysine methyltransferase EZH2

  • GC13878 structure
    GC13878EPZ005687
    CAS: 1396772-26-1
    Purity: >99.00%

    A potent, selective inhibitor of EZH2

  • GC15783 structure
    GC15783GSK126
    CAS: 1346574-57-9
    Purity: >98.00%

    مثبط انتقائي لـ EZH2

  • GC17534 structure
    GC17534GSK343
    CAS: 1346704-33-3
    Purity: >98.00%

    A selective, cell-permeable EZH2 inhibitor

  • GC17907 structure
    GC179073-Deazaneplanocin A (DZNep) hydrochloride
    CAS: 120964-45-6
    Purity: >99.50%

    مثبط لإنزيم الميثيل ترانسفيراز EZH2 الذي يعمل على إضافة مجموعات الميثيل على الأحماض الأمينية من نوع اللايسين.

  • GC14756 structure
    GC14756EI1
    CAS: 1418308-27-6
    Purity: >99.50%

    EI1 (KB-145943) هو مثبط EZH2 فعال وانتقائي مع IC50 من 15 نانومتر و 13 نانومتر لـ EZH2 (WT) و EZH2 (Y641F) ، على التوالي

  • GC11484 structure
    GC11484CPI-169 S-enantiomer
    Purity: >98%

    EZH2 inhibitor

  • GC12146 structure
    GC12146CPI-169 R-enantiomer
    CAS: 1802175-07-0
    Purity: >98%

    EZH2 inhibitor

  • GC16599 structure
    GC16599CPI-169
    CAS: 1450655-76-1
    Purity: >98.00%

    EZH2 inhibitor