Proteolysis
Products Related to Proteolysis(179)
- GC40124Ac-WEAD-AMC (trifluoroacetate salt)Purity: >95.00%
Ac-WEAD-AMC is a fluorogenic substrate for caspase-1 and caspase-4.
- GC40125Z-VA-DL-D(OMe)-FMK (trifluoroacetate salt)Purity: >95.00%
Z-VA-DL-D(OMe)-FMK (Z-VAD-FMK) is a pan-caspase inhibitor.
- GC40145(S)-LaudanosineCAS: 2688-77-9Purity: >98.00%
(S)-Laudanosine is the (S) enantiomer of laudanosine, a metabolite of the neuromuscular blocking agents atracurium and cisatracurium.
- GC40149Boc-AEVD-CHO (trifluoroacetate salt)Purity: >95.00%
Boc-AEVD-CHO is an inhibitor of caspase-8 (Ki = 1.6 nM) that also inhibits caspase-1, -3, -6, and -9 (Kis = 10,000, 375, 438, 425, and 320 nM, respectively).
- GC40150Z-VEID-AFC (trifluoroacetate salt)Purity: >95.00%
Z-VEID-AFC is a fluorogenic substrate for caspase-6.
- GC40152Ac-IEPD-pNA (trifluoroacetate salt)Purity: >95.00%
Ac-IEPD-pNA is a colorimetric substrate for granzyme B and caspase-8.
- GC40153Z-YVAD-AFC (trifluoroacetate salt)Purity: >95.00%
Z-YVAD-AFC is a fluorogenic substrate for caspase-1.
- GC40154Ac-ESMD-CHO (trifluoroacetate salt)Purity: >95.00%
Ac-ESMD-CHO is an inhibitor of caspase-3 maturation.
- GC40155Biotin-DEVD-CHO (trifluoroacetate salt)Purity: >95.00%
Biotin-DEVD-CHO is a biotin-conjugated form of the caspase-3 and -7 inhibitor Ac-DEVD-CHO.
- GC40164Ac-IETD-CHO (trifluoroacetate salt)Purity: >95.00%
Ac-IETD-CHO (trifluoroacetate salt) is a caspase 8 inhibitor that can prevent the focal adhesion kinase (Fak) from being cleaved by caspase, with an IC 50 value of 200nM.
- GC402027α-hydroxy Cholesterol-d7CAS: 349553-94-2Purity: >99.00%
7α-hydroxy Cholesterol-d7 is intended for use as an internal standard for the quantification of 7α-hydroxy cholesterol by GC- or LC-MS.
- GC40256p-APMSF (hydrochloride)CAS: 74938-88-8Purity: >95.00%
p-APMSF is an irreversible inhibitor of serine proteases with Ki values of 1.02, 1.18, 1.5, and 1.54 μM for bovine trypsin, human thrombin, bovine plasmin, and bovine Factor Xa, respectively.
- GC40622PenicillideCAS: 55303-92-9Purity: >95.00%
يُظهر البنسليد (Vermixocin A) ، المعزول من Talaromyces derxii المزروع على الأرز ، نشاطًا مثبطًا ضد acyl-CoA: الكوليسترول acyltransferase (ACAT)
- GC40624MMP-3 Inhibitor VIIICAS: 208663-26-7Purity: >95.00%
Matrix metalloproteinases (MMPs) belong to a family of proteases that play a crucial role in tissue remodeling and repair by degrading extracellular matrix proteins to enable cell migration.
- GC40758Gly-Phe-β-naphthylamideCAS: 21438-66-4Purity: >98.00%
Gly-Phe-β ؛ -naphthylamide هو الركيزة لـ Cathepsin C.
- GC414235-trans Prostaglandin E2CAS: 36150-00-2Purity: >98.00%
5-trans PGE2 occurs naturally in some gorgonian corals and is a common impurity in commercial lots of PGE1.
- GC41656(±)2-(14,15-Epoxyeicosatrienoyl) GlycerolCAS: 848667-56-1Purity: >95.00%
2-Arachidonoyl glycerol (2-AG) is an endogenous central cannabinoid (CB1) receptor agonist that is present at relatively high levels in the central nervous system.
- GC41698(D)2-Rh 110 (trifluoroacetate salt)Purity: >95.00%
(D)2-Rh 110 is a fluorogenic caspase substrate.
- GC41742(Z-IETD)2-Rh 110 (trifluoroacetate salt)Purity: >95.00%
(Z-IETD)2-Rh 110 is a fluorogenic substrate for caspase-8.
- GC425485-hydroxy Saxagliptin (hydrochloride)Purity: >95.00%
5-hydroxy Saxagliptin is a major active metabolite of saxagliptin.
| Catalog No. | Product Name | CAS No. | Purity | Structure |
|---|---|---|---|---|
| GC40124 | Ac-WEAD-AMC (trifluoroacetate salt) | - | >95.00% | |
Ac-WEAD-AMC is a fluorogenic substrate for caspase-1 and caspase-4. | ||||
| GC40125 | Z-VA-DL-D(OMe)-FMK (trifluoroacetate salt) | - | >95.00% | |
Z-VA-DL-D(OMe)-FMK (Z-VAD-FMK) is a pan-caspase inhibitor. | ||||
| GC40145 | (S)-Laudanosine | 2688-77-9 | >98.00% | |
(S)-Laudanosine is the (S) enantiomer of laudanosine, a metabolite of the neuromuscular blocking agents atracurium and cisatracurium. | ||||
| GC40149 | Boc-AEVD-CHO (trifluoroacetate salt) | - | >95.00% | |
Boc-AEVD-CHO is an inhibitor of caspase-8 (Ki = 1.6 nM) that also inhibits caspase-1, -3, -6, and -9 (Kis = 10,000, 375, 438, 425, and 320 nM, respectively). | ||||
| GC40150 | Z-VEID-AFC (trifluoroacetate salt) | - | >95.00% | |
Z-VEID-AFC is a fluorogenic substrate for caspase-6. | ||||
| GC40151 | Z-VAD-AMC (acetate) | - | >95.00% | |
Z-VAD-AMC is a fluorogenic substrate for caspase-1. | ||||
| GC40152 | Ac-IEPD-pNA (trifluoroacetate salt) | - | >95.00% | |
Ac-IEPD-pNA is a colorimetric substrate for granzyme B and caspase-8. | ||||
| GC40153 | Z-YVAD-AFC (trifluoroacetate salt) | - | >95.00% | |
Z-YVAD-AFC is a fluorogenic substrate for caspase-1. | ||||
| GC40154 | Ac-ESMD-CHO (trifluoroacetate salt) | - | >95.00% | |
Ac-ESMD-CHO is an inhibitor of caspase-3 maturation. | ||||
| GC40155 | Biotin-DEVD-CHO (trifluoroacetate salt) | - | >95.00% | |
Biotin-DEVD-CHO is a biotin-conjugated form of the caspase-3 and -7 inhibitor Ac-DEVD-CHO. | ||||
| GC40162 | Ac-VEID-pNA (trifluoroacetate salt) | - | >95.00% | |
Ac-VEID-pNA is a substrate for caspase-6. | ||||
| GC40164 | Ac-IETD-CHO (trifluoroacetate salt) | - | >95.00% | |
Ac-IETD-CHO (trifluoroacetate salt) is a caspase 8 inhibitor that can prevent the focal adhesion kinase (Fak) from being cleaved by caspase, with an IC 50 value of 200nM. | ||||
| GC40202 | 7α-hydroxy Cholesterol-d7 | 349553-94-2 | >99.00% | |
7α-hydroxy Cholesterol-d7 is intended for use as an internal standard for the quantification of 7α-hydroxy cholesterol by GC- or LC-MS. | ||||
| GC40256 | p-APMSF (hydrochloride) | 74938-88-8 | >95.00% | |
p-APMSF is an irreversible inhibitor of serine proteases with Ki values of 1.02, 1.18, 1.5, and 1.54 μM for bovine trypsin, human thrombin, bovine plasmin, and bovine Factor Xa, respectively. | ||||
| GC40265 | Pheleuin | 169195-23-7 | >98.00% | |
Pheleuin is a pyrazinone derivative synthesized from a dipeptide aldehyde. | ||||
| GC40556 | Ac-LETD-AFC | 210345-02-1 | >95.00% | |
Ac-LETD-AFC عبارة عن ركيزة فلورية من كاسباس 8. | ||||
| GC40622 | Penicillide | 55303-92-9 | >95.00% | |
يُظهر البنسليد (Vermixocin A) ، المعزول من Talaromyces derxii المزروع على الأرز ، نشاطًا مثبطًا ضد acyl-CoA: الكوليسترول acyltransferase (ACAT) | ||||
| GC40624 | MMP-3 Inhibitor VIII | 208663-26-7 | >95.00% | |
Matrix metalloproteinases (MMPs) belong to a family of proteases that play a crucial role in tissue remodeling and repair by degrading extracellular matrix proteins to enable cell migration. | ||||
| GC40758 | Gly-Phe-β-naphthylamide | 21438-66-4 | >98.00% | |
Gly-Phe-β ؛ -naphthylamide هو الركيزة لـ Cathepsin C. | ||||
| GC41423 | 5-trans Prostaglandin E2 | 36150-00-2 | >98.00% | |
5-trans PGE2 occurs naturally in some gorgonian corals and is a common impurity in commercial lots of PGE1. | ||||
| GC41656 | (±)2-(14,15-Epoxyeicosatrienoyl) Glycerol | 848667-56-1 | >95.00% | |
2-Arachidonoyl glycerol (2-AG) is an endogenous central cannabinoid (CB1) receptor agonist that is present at relatively high levels in the central nervous system. | ||||
| GC41698 | (D)2-Rh 110 (trifluoroacetate salt) | - | >95.00% | |
(D)2-Rh 110 is a fluorogenic caspase substrate. | ||||
| GC41742 | (Z-IETD)2-Rh 110 (trifluoroacetate salt) | - | >95.00% | |
(Z-IETD)2-Rh 110 is a fluorogenic substrate for caspase-8. | ||||
| GC42548 | 5-hydroxy Saxagliptin (hydrochloride) | - | >95.00% | |
5-hydroxy Saxagliptin is a major active metabolite of saxagliptin. | ||||