BET bromodomain inhibitor 4 (example 7) is an inhibitor of the BET bromodomain domain.
References:
[1]. Preparation of tricyclic compounds as bromodomain and BET inhibitors. World Intellectual Property Organization, WO2020001152 A1 2020-01-02.
BET bromodomain inhibitor 4
Catalog No.: GC73742Purity:>99.00%
BET bromodomain inhibitor 4 (example 7) is an inhibitor of the BET bromodomain domain.
Products are for research use only. Not for human use. We do not sell to patients.
Cas No.: 2407658-41-5
10mM (in 1mL DMSO)In Stock
$734.00
1
1 mgIn Stock
$257.00
1
| Pack Size | Price | Availability | Quantity | Action |
|---|---|---|---|---|
| 10mM (in 1mL DMSO) | $734.00 | In Stock | 1 | |
| 1 mg | $257.00 | In Stock | 1 |
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Citations
No citations are currently available for this product. Below are selected publications citing GlpBio products.
Nature641, 529–536 (2025)
Nature628, 630–638 (2024)
Nature632, 686–694 (2024)
Nature618, 1017–1023 (2023)
Nature610, 366–372 (2022)
Cell187(9):2288-2304 (2024)
Cell183(7):1867-1883 (2020)
Science388(6745) (2025)
Science387(6739) (2025)
Science387(6734) (2025)
Cell Research35, 97–116 (2025)
Cell Research34, 683–706 (2024)
Cell Research33, 273–287 (2023)
Cell Research33, 546–561 (2023)
Cell Research33, 904–922 (2023)
Cell Research31, 1291–1307 (2021)
Description
Product Documents
Purity:>99.00%Appearance:A solid
Chemical Properties
CAS No.
2407658-41-5
Molecular Formula
C27H31FN8O2
Molecular Weight
518.59
Solubility
DMSO : 100 mg/mL (192.83 mM; Need ultrasonic)
Storage
-20°C
General tips
Select a suitable solvent according to the product solubility data. Once prepared, aliquot the stock solution to avoid repeated freeze-thaw cycles.
Use stock solutions within 6 months when stored at -80°C or within 1 month when stored at -20°C.
To improve solubility, warm the tube to 37°C and sonicate it for an appropriate period.
Use stock solutions within 6 months when stored at -80°C or within 1 month when stored at -20°C.
To improve solubility, warm the tube to 37°C and sonicate it for an appropriate period.
Shipping Condition
Evaluation samples are shipped with blue ice. Other available sizes are shipped at room temperature or with blue ice upon request.
CalculatorsMolarity / Dilution / Molecular Weight / Unit Conversion / In Vivo Formulation / Solubility
g/mol
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