GLPBio

BRD4 ligand-Linker Conjugate 1 TFA

Catalog No.: GC73033Purity:>98.00%
COASDSData Sheet
BRD4 ligand-Linker Conjugate 1 TFA (compound 106-1) is a target protein ligand-linker conjugate that can be used in the synthesis of PROTACs.

Products are for research use only. Not for human use. We do not sell to patients.

BRD4 ligand-Linker Conjugate 1 TFA
1 mgIn Stock
$225.00
1
Tel: (909) 407-4943 / (909) 689-7124Email: sales@glpbio.com

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Description

BRD4 ligand-Linker Conjugate 1 TFA (compound 106-1) is a target protein ligand-linker conjugate that can be used in the synthesis of PROTACs.

References:
[1]. Sun D, et al. Evaluation of the Small-molecule BRD4 Degrader CFT-2718 in Small-cell Lung Cancer and Pancreatic Cancer Models. Mol Cancer Ther. 2021 Aug;20(8):1367-1377.
[2]. Phillips AJ, et al. Preparation of bromodomain targeting degronimers for target protein degradation. World Intellectual Property Organization, WO2017197056 A1. 2017-11-16.

Product Documents

Purity:>98.00%Appearance:A liquid
COASDSData Sheet

Chemical Properties

Molecular Formula
C30H31ClF3N7O2
Molecular Weight
614.06
Solubility
H2O : 100 mg/mL (162.85 mM; Need ultrasonic)
Storage
4°C, stored under nitrogen, away from moisture
General tips
Select a suitable solvent according to the product solubility data. Once prepared, aliquot the stock solution to avoid repeated freeze-thaw cycles.
Use stock solutions within 6 months when stored at -80°C or within 1 month when stored at -20°C.
To improve solubility, warm the tube to 37°C and sonicate it for an appropriate period.
Shipping Condition
Evaluation samples are shipped with blue ice. Other available sizes are shipped at room temperature or with blue ice upon request.

CalculatorsMolarity / Dilution / Molecular Weight / Unit Conversion / In Vivo Formulation / Solubility

g/mol

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