DAPK

DAPK (death-associated protein kinase) is a positive mediator of gamma-interferon induced programmed cell death.

Products Related to DAPK(10)

GC13950 TC-DAPK 6
CAS: 315694-89-4
Purity: >98%
GC34557 DIM-C-pPhCO2Me
CAS: 151358-48-4
Purity: >99.50%
DIM-C-pPhCO2Me is a nuclear receptor 4A1 (NR4A1) antagonist, with a K i value of 0.25μM.
GC50260 HS 38
CAS: 1030203-81-6
Purity: >99.00%
ATP-competitive inhibitor of DAPK and ZIPK
GC61593 DAPK Substrate Peptide TFA
Purity: >99.00%
DAPK Substrate Peptide TFA is a synthetic peptide substrate for death associated protein kinase (DAPK), with a Km of 9 μM.
GC65140 DRAK2-IN-1
CAS: 871837-60-4
Purity: >99.50%
DRAK2-IN-1, compound 16, is a potent, selective and ATP-competitive DRAK2 inhibitor with IC50and Kivalues of 3 nM and 0.26 nM, respectively.
GC65328 TNIK-IN-3
CAS: 2754265-25-1
Purity: >99.00%
TNIK-IN-3 is a potent, selective and orally active inhibitor of Traf2- and Nck-interacting protein kinase (TNIK), with an IC50 of 0.026 μM. TNIK-IN-3 could also inhibit Flt4 (IC50=0.030 μM), Flt1 (IC50=0.191 μM) and DRAK1 (IC50=0.411 μM). TNIK-IN-3 can be used for the research of colorectal cancer.
GC72879 HS148
CAS: 1892595-16-2
Purity: >95.00%
HS148 (compound 22) is a selective DAPK3 inhibitor with an Ki value of 119 nM.
GC73211 CK156
CAS: 2910938-59-7
Purity: >99.50%
CK156 is a highly selective death-associated protein kinase (DAPK) inhibitor with IC50s of 182 nM,34 μM, and 39 μM in the DRAK1 NanoBRET assay for DRAK1, CK2a1, and CK2a2, respectively.
GC80881 PROTAC DAPK1 Degrader-1
CAS: 3063030-38-3
Purity: >96.50%
PROTAC DAPK1 Degrader-1 is a death-associated protein kinase 1 (DAPK1) degrader with a DC 50 of 119.6 nM.
GC81304 GW296115
CAS: 118458-58-5
Purity: >98.50%
GW296115 is a multi-target inhibitor with the following IC 50 values against its targets: 8.4 nM for BRSK2, 21 nM for BRSK1, 1.8 μM for PDGFRβ, 5.5 nM for STK17B/DRAK2, 28 nM for DRAK1, 20 nM for PHKG1, and 89 nM for DCAMKL3.

Category Product List
Catalog No.	Product Name	CAS No.	Purity
GC13950	TC-DAPK 6	315694-89-4	>98%
GC34557	DIM-C-pPhCO2Me	151358-48-4	>99.50%
GC34557	DIM-C-pPhCO2Me is a nuclear receptor 4A1 (NR4A1) antagonist, with a K i value of 0.25μM.
GC50260	HS 38	1030203-81-6	>99.00%
GC50260	ATP-competitive inhibitor of DAPK and ZIPK
GC61593	DAPK Substrate Peptide TFA	-	>99.00%
GC61593	DAPK Substrate Peptide TFA is a synthetic peptide substrate for death associated protein kinase (DAPK), with a Km of 9 μM.
GC65140	DRAK2-IN-1	871837-60-4	>99.50%
GC65140	DRAK2-IN-1, compound 16, is a potent, selective and ATP-competitive DRAK2 inhibitor with IC50and Kivalues of 3 nM and 0.26 nM, respectively.
GC65328	TNIK-IN-3	2754265-25-1	>99.00%
GC65328	TNIK-IN-3 is a potent, selective and orally active inhibitor of Traf2- and Nck-interacting protein kinase (TNIK), with an IC50 of 0.026 μM. TNIK-IN-3 could also inhibit Flt4 (IC50=0.030 μM), Flt1 (IC50=0.191 μM) and DRAK1 (IC50=0.411 μM). TNIK-IN-3 can be used for the research of colorectal cancer.
GC72879	HS148	1892595-16-2	>95.00%
GC72879	HS148 (compound 22) is a selective DAPK3 inhibitor with an Ki value of 119 nM.
GC73211	CK156	2910938-59-7	>99.50%
GC73211	CK156 is a highly selective death-associated protein kinase (DAPK) inhibitor with IC50s of 182 nM,34 μM, and 39 μM in the DRAK1 NanoBRET assay for DRAK1, CK2a1, and CK2a2, respectively.
GC80881	PROTAC DAPK1 Degrader-1	3063030-38-3	>96.50%
GC80881	PROTAC DAPK1 Degrader-1 is a death-associated protein kinase 1 (DAPK1) degrader with a DC 50 of 119.6 nM.
GC81304	GW296115	118458-58-5	>98.50%
GC81304	GW296115 is a multi-target inhibitor with the following IC 50 values against its targets: 8.4 nM for BRSK2, 21 nM for BRSK1, 1.8 μM for PDGFRβ, 5.5 nM for STK17B/DRAK2, 28 nM for DRAK1, 20 nM for PHKG1, and 89 nM for DCAMKL3.