Lumekefamide TFA ([D-Arg2]Dermorphin-(1-4) amide TFA) is a N-terminal shorter peptide amide of [D-Arg2]dermorphin with the hypothermic effect. Lumekefamide shows analgesic activity and degradation in soluble mouse liver and brain extracts [1].
References:
[1]. Emel'ianova TG, et al. Termoreguliatornaia aktivnost' dermofinov [Thermoregulatory activity of dermorphin fragments]. Izv Akad Nauk Ser Biol. 2004 Sep-Oct;(5):570-6.
References:
[1]. Emel'ianova TG, et al. Termoreguliatornaia aktivnost' dermofinov [Thermoregulatory activity of dermorphin fragments]. Izv Akad Nauk Ser Biol. 2004 Sep-Oct;(5):570-6.
















