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NVP-2

Catalog No.GC34056

NVP-2 est une sonde puissante et sélective de la kinase 9 (CDK9) dépendante de la cycline compétitive pour l'ATP, inhibe l'activité CDK9/CycT avec une IC50 de 0,514 nM. NVP-2 affiche des effets inhibiteurs sur les kinases CDK1/CycB, CDK2/CycA et CDK16/CycY avec des valeurs IC50 de 0,584 μM, 0,706 μM et 0,605 μM, respectivement. NVP-2 induit l'apoptose cellulaire.

Products are for research use only. Not for human use. We do not sell to patients.

NVP-2 Chemical Structure

Cas No.: 1263373-43-8

Taille Prix Stock Qté
10mM (in 1mL DMSO)
152,00 $US
En stock
1mg
58,00 $US
En stock
5mg
135,00 $US
En stock
10mg
234,00 $US
En stock
50mg
864,00 $US
En stock
100mg
1 485,00 $US
En stock

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Sample solution is provided at 25 µL, 10mM.

Product has been cited by 1 publications

Description Chemical Properties Product Documents Related Products

NVP-2 is a CDK9 inhibitor with an IC50 of 0.5 nM.

[1]. Wang J, et al. SnapShot: Kinase Inhibitors I. Mol Cell. 2015 May 21;58(4):708.e1.

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