GLPBio

JZY3221

Catalog No.: GC81355Purity:>98.00%
COASDSData Sheet
JZY3221 is an androgen receptor ( AR ) inhibitor.

제품은 연구용으로만 사용됩니다. 인체에 사용할 수 없으며 환자에게 판매하지 않습니다.

JZY3221
10mM (in 1mL DMSO)In Stock
$285.00
1
5mgIn Stock
$259.00
1
10mgIn Stock
$418.00
1
Tel: (909) 407-4943 / (909) 689-7124Email: sales@glpbio.com

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제품 설명 (Description)

JZY3221 is an androgen receptor ( AR ) inhibitor. JZY3221 binds to the AR ligand-binding domain to inhibit AR function. JZY3221 constitutes the AR inhibitory moiety of DALTAC JZY3032. JZY3221 is applicable to research related to prostate cancer [1].

In Vitro, JZY3221 exhibits only limited cell growth inhibitory activity in AR-positive 22Rv1 prostate cancer cells[1]. JZY3221 directly binds to purified AR protein[1].

References:
[1]. Luo J, et al. Rewiring Oncogenic Transcriptional Complexes with Domain-ALTeration Chimeras (DALTACs) in Prostate Cancer. bioRxiv [Preprint]. 2026 Apr 28:2026.04.24.720638.

제품 문서 (Product Documents)

Purity:>98.00%Appearance:A solid
COASDSData Sheet

화학적 특성 (Chemical Properties)

분자식
C19H20ClN5O
분자량
369.85
용해도
DMSO: 100 mg/mL (270.38 mM; Need ultrasonic)
보관
Store at -20°C
배송 조건
평가용 샘플은 아이스팩과 함께 배송됩니다. 그 외 용량은 실온 배송되며, 요청 시 아이스팩과 함께 배송할 수 있습니다.

계산 도구 (Calculators)몰 농도 / 희석 / 분자량 / 단위 변환 / 생체 내 제형 / 용해도

g/mol

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