GLPBio

KRAS-PDEδ

PDEδ is a GDI-like solubilizing factor, which regulates the farnesylated KRAS signaling. KRAS-PDEδ interaction is a drug target for cancer treatment.

Products Related to KRAS-PDEδ(3)

  • GC13076 structure
    GC13076Deltarasin
    CAS: 1440898-61-2
    Purity: >98%

    A KRAS inhibitor

  • GC17669 structure
    GC17669AMG-47A
    CAS: 882663-88-9
    Purity: >98.50%

    AMG-47a는 IC50이 0.2nM인 강력하고 경구 활성인 림프구 특이적 단백질 티로신 키나제(Lck) 억제제입니다.

  • GC12060 structure
    GC12060Deltarasin hydrochloride
    CAS: 1440898-82-7
    Purity: >99.50%

    Deltarasin 염산염은 정제된 PDEδ에 결합하기 위해 38nM의 Kd와 KRAS-PDEδ상호작용의 억제제입니다.