GLPBio

PROTAC BRD4 ligand-2 hydrochloride

Catalog No.: GC73032Purity:>99.00%
COASDSData Sheet
PROTAC BRD4 ligand-2 drochloride is a ligand for target BRD4 protein for PROTAC CFT-2718.

Products are for research use only. Not for human use. We do not sell to patients.

PROTAC BRD4 ligand-2 hydrochloride
1 mgIn Stock
$382.00
1
Tel: (909) 407-4943 / (909) 689-7124Email: sales@glpbio.com

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    187(9):2288-2304 (2024)
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    183(7):1867-1883 (2020)
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    31, 1291–1307 (2021)

Description

PROTAC BRD4 ligand-2 drochloride is a ligand for target BRD4 protein for PROTAC CFT-2718.

References:
[1]. Sun D, et al. Evaluation of the Small-molecule BRD4 Degrader CFT-2718 in Small-cell Lung Cancer and Pancreatic Cancer Models. Mol Cancer Ther. 2021 Aug;20(8):1367-1377.

Product Documents

Purity:>99.00%Appearance:A solid
COASDSData Sheet

Chemical Properties

Molecular Formula
C22H18Cl2N6
Molecular Weight
437.32
Solubility
DMSO : 100 mg/mL (228.67 mM; Need ultrasonic)
Storage
4°C, sealed storage, away from moisture and light
General tips
Select a suitable solvent according to the product solubility data. Once prepared, aliquot the stock solution to avoid repeated freeze-thaw cycles.
Use stock solutions within 6 months when stored at -80°C or within 1 month when stored at -20°C.
To improve solubility, warm the tube to 37°C and sonicate it for an appropriate period.
Shipping Condition
Evaluation samples are shipped with blue ice. Other available sizes are shipped at room temperature or with blue ice upon request.

CalculatorsMolarity / Dilution / Molecular Weight / Unit Conversion / In Vivo Formulation / Solubility

g/mol

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