GLPBio

(S)-PF-5190457

Catalog No.: GC79204Purity:>99.00%Synonyms: (S)-PF-05190457
COASDSData Sheet
(S)-PF-5190457 ((S)-PF-05190457) is the S-enantiomer of PF-5190457.

Products are for research use only. Not for human use. We do not sell to patients.

(S)-PF-5190457
5mgIn Stock
$104.00
1
10mgIn Stock
$182.00
1
25mgIn Stock
$364.00
1
50mgIn Stock
$527.00
1
Tel: (909) 407-4943 / (909) 689-7124Email: sales@glpbio.com

Citations

No citations are currently available for this product. Below are selected publications citing GlpBio products.
  • Nature cover
    Nature
    641, 529–536 (2025)
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    Nature
    628, 630–638 (2024)
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    Nature
    632, 686–694 (2024)
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    618, 1017–1023 (2023)
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    Nature
    610, 366–372 (2022)
  • Cell cover
    Cell
    187(9):2288-2304 (2024)
  • Cell cover
    Cell
    183(7):1867-1883 (2020)
  • Science cover
    Science
    388(6745) (2025)
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    387(6739) (2025)
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    Science
    387(6734) (2025)
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    Cell Research
    35, 97–116 (2025)
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    Cell Research
    34, 683–706 (2024)
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    33, 273–287 (2023)
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    33, 546–561 (2023)
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    33, 904–922 (2023)
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    Cell Research
    31, 1291–1307 (2021)

Description

(S)-PF-5190457 ((S)-PF-05190457) is the S-enantiomer of PF-5190457. PF-5190457 (PF-05190457) is a potent and selective ghrelin receptor inverse agonist with a pK i of 8.36 [1].

References:
[1]. Bhattacharya SK, et al. Discovery of PF-5190457, a Potent, Selective, and Orally Bioavailable Ghrelin Receptor Inverse Agonist Clinical Candidate. ACS Med Chem Lett. 2014 Feb 24;5(5):474-9.

Product Documents

Purity:>99.00%Appearance:A solid
COASDSData Sheet

Chemical Properties

Synonyms
(S)-PF-05190457
Molecular Formula
C29H32N6OS
Molecular Weight
512.67
Storage
Store at -20°C
Shipping Condition
Evaluation samples are shipped with blue ice. Other available sizes are shipped at room temperature or with blue ice upon request.

CalculatorsMolarity / Dilution / Molecular Weight / Unit Conversion / In Vivo Formulation / Solubility

g/mol

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