GHSR
GHSR (growth hormone secretagogue receptor) is a G protein-coupled receptor that binds ghrelin and plays a role in energy homeostasis and regulation of body weight.
Products for GHSR
- Cat.No. Product Name Information
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GC67681
(αR,8aS)-GSK1614343
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GC35282
Alexamorelin Met 1
-
GC13253
Anamorelin
RC-1291
A small molecule agonist of GHS-R1a -
GC35337
Anamorelin Fumarate
Anamorelin Fumarate is a novel ghrelin receptor agonist with EC50 value of 0.74 nM in the FLIPR assay.
-
GC35338
Anamorelin hydrochloride
Anamorelin (RC-1291) hydrochloride is a potent ghrelin receptor agonist with EC50 value of 0.74 nM in the FLIPR assay.
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GC31430
AZP-531
AZP-531 is an analogue of unacylated ghrelin designed to improve glycaemic control and reduce weight.
-
GC19087
Capromorelin Tartrate
CP 424,391-18, RQ-00000005
Capromorelin Tartrate is an orally active, potent growth hormone secretagogue receptor (GHSR) agonist, with Ki of 7 nM for hGHS-R1a. -
GC30388
Human growth hormone-releasing factor (Growth Hormone Releasing Factor human)
Human growth hormone-releasing factor (Growth Hormone Releasing Factor human) (Growth Hormone Releasing Factor human) is a hypothalamic polypeptide and stimulates GH production and release by binding to the GHRH Receptor (GHRHR) on cells in the anterior pituitary.
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GC61519
Human growth hormone-releasing factor TFA
Growth Hormone Releasing Factor human TFA
Human growth hormone-releasing factor TFA (Growth Hormone Releasing Factor human TFA) is a hypothalamic polypeptide and stimulates GH production and release by binding to the GHRH Receptor (GHRHR) on cells in the anterior pituitary. -
GC10287
Ibutamoren Mesylate
L-163,191, MK-0677
A growth hormone secretagogue and ghrelin receptor agonist
-
GC31274
JMV 2959
JMV 2959 is a growth hormone secretagogue receptor type 1a (GHS-R1a) antagonist with an IC50 of 32 nM.
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GC34207
JMV 2959 hydrochloride
JMV 2959 hydrochloride is a growth hormone secretagogue receptor type 1a (GHS-R1a) antagonist with an IC50 of 32±3 nM in LLC-PK1 cells.
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GC60971
L-692429
MK-0751
L-692429 (MK-0751) is a benzolactam derivative and a nonpeptidyl growth hormone secretagogue (GHS) agonist. -
GC71024
Macimorelin acetate
Macimorelin (EP-1572) acetate, a GH secretagogue, is an orally active GHSR agonist.
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GC34095
ONC212
A GPR132 agonist
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GC31478
PF-5190457
PF-05190457
PF-5190457 (PF-05190457) is a potent and selective ghrelin receptor inverse agonist with a pKi of 8.36. -
GC63727
Relamorelin TFA
RM-131 TFA; BIM-28131 TFA
Relamorelin (RM-131) TFA, a pentapeptide ghrelin analog, is a selective ghrelin/growth hormone secretagogue receptor (GHSR) agonist with a Ki of 0.42 nM for GHS-1a receptor. -
GC19349
TC-G-1008
GPR39-C3
TC-G-1008 (GPR39-C3) is a potent and orally available GPR39 agonist with EC50 values of 0.4 and 0.8 nM for rat and human receptors respectively. -
GC31074
TM-N1324
Compound 1324, Cpd1324
TM-N1324 is an agonist of G-Protein-Coupled Receptor 39 (GPR39) with EC50s of 9 nM/5 nM in the presence of Zn2+, and 280 nM/180 nM in the absence of Zn2+ for human/murine GPR39.