GHSR
GHSR (growth hormone secretagogue receptor) is a G protein-coupled receptor that binds ghrelin and plays a role in energy homeostasis and regulation of body weight.
Products for GHSR
- Cat.No. Product Name Information
- GC67681 (αR,8aS)-GSK1614343
- GC35282 Alexamorelin Met 1
- GC13253 Anamorelin A small molecule agonist of GHS-R1a
- GC35337 Anamorelin Fumarate Anamorelin Fumarate is a novel ghrelin receptor agonist with EC50 value of 0.74 nM in the FLIPR assay.
- GC35338 Anamorelin hydrochloride Anamorelin (RC-1291) hydrochloride is a potent ghrelin receptor agonist with EC50 value of 0.74 nM in the FLIPR assay.
- GC31430 AZP-531 AZP-531 is an analogue of unacylated ghrelin designed to improve glycaemic control and reduce weight.
- GC19087 Capromorelin Tartrate Capromorelin Tartrate is an orally active, potent growth hormone secretagogue receptor (GHSR) agonist, with Ki of 7 nM for hGHS-R1a.
- GC30388 Human growth hormone-releasing factor (Growth Hormone Releasing Factor human) Human growth hormone-releasing factor (Growth Hormone Releasing Factor human) (Growth Hormone Releasing Factor human) is a hypothalamic polypeptide and stimulates GH production and release by binding to the GHRH Receptor (GHRHR) on cells in the anterior pituitary.
- GC61519 Human growth hormone-releasing factor TFA Human growth hormone-releasing factor TFA (Growth Hormone Releasing Factor human TFA) is a hypothalamic polypeptide and stimulates GH production and release by binding to the GHRH Receptor (GHRHR) on cells in the anterior pituitary.
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GC10287
Ibutamoren Mesylate
A growth hormone secretagogue and ghrelin receptor agonist
- GC31274 JMV 2959 JMV 2959 is a growth hormone secretagogue receptor type 1a (GHS-R1a) antagonist with an IC50 of 32 nM.
- GC34207 JMV 2959 hydrochloride JMV 2959 hydrochloride is a growth hormone secretagogue receptor type 1a (GHS-R1a) antagonist with an IC50 of 32±3 nM in LLC-PK1 cells.
- GC60971 L-692429 L-692429 (MK-0751) is a benzolactam derivative and a nonpeptidyl growth hormone secretagogue (GHS) agonist.
- GC34095 ONC212 A GPR132 agonist
- GC31478 PF-5190457 PF-5190457 (PF-05190457) is a potent and selective ghrelin receptor inverse agonist with a pKi of 8.36.
- GC63727 Relamorelin TFA Relamorelin (RM-131) TFA, a pentapeptide ghrelin analog, is a selective ghrelin/growth hormone secretagogue receptor (GHSR) agonist with a Ki of 0.42 nM for GHS-1a receptor.
- GC19349 TC-G-1008 TC-G-1008 (GPR39-C3) is a potent and orally available GPR39 agonist with EC50 values of 0.4 and 0.8 nM for rat and human receptors respectively.
- GC31074 TM-N1324 TM-N1324 is an agonist of G-Protein-Coupled Receptor 39 (GPR39) with EC50s of 9 nM/5 nM in the presence of Zn2+, and 280 nM/180 nM in the absence of Zn2+ for human/murine GPR39.