GLPBio

(S,S)-CPI-1612

Catalog No.: GC73104Purity:>99.00%
(S,S)-CPI-1612 is the isomer of CPI-1612 , and can be used as an experimental control.

Products are for research use only. Not for human use. We do not sell to patients.


(S,S)-CPI-1612
Cas No.: 2374971-82-9
1 mgIn Stock
$281.00
1

Citations

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    Nature
    641, 529–536 (2025)
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    628, 630–638 (2024)
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    632, 686–694 (2024)
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    618, 1017–1023 (2023)
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    610, 366–372 (2022)
  • Cell cover
    Cell
    187(9):2288-2304 (2024)
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    Cell
    183(7):1867-1883 (2020)
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    Science
    388(6745) (2025)
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    387(6739) (2025)
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    387(6734) (2025)
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    Cell Research
    35, 97–116 (2025)
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    34, 683–706 (2024)
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    33, 273–287 (2023)
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    33, 546–561 (2023)
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    33, 904–922 (2023)
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    31, 1291–1307 (2021)

Description

(S,S)-CPI-1612 is the isomer of CPI-1612 , and can be used as an experimental control. CPI-1612 is a highly potent, orally active EP300/CBP histone acetyltransferase (HAT) inhibitor with an IC50 of 8.1 nM for EP300 HAT. CPI-1612 has an anticancer activity.

References:
[1]. Wang F, et al. Microstructure of poly(gamma-glutamic acid) produced by Bacillus subtilis consisting of clusters of D- and L-glutamic acid repeating units. J Agric Food Chem. 2008 Jun 11;56(11):4225-8.

Product Documents

Purity:>99.00%Appearance:A solid

Chemical Properties

CAS No.
2374971-82-9
Molecular Formula
C27H26N6O
Molecular Weight
450.53
Solubility
DMSO : 50 mg/mL (110.98 mM; Need ultrasonic)
Storage
-20°C
General tips
Select a suitable solvent according to the product solubility data. Once prepared, aliquot the stock solution to avoid repeated freeze-thaw cycles.
Use stock solutions within 6 months when stored at -80°C or within 1 month when stored at -20°C.
To improve solubility, warm the tube to 37°C and sonicate it for an appropriate period.
Shipping Condition
Evaluation samples are shipped with blue ice. Other available sizes are shipped at room temperature or with blue ice upon request.

CalculatorsMolarity / Dilution / Molecular Weight / Unit Conversion / In Vivo Formulation / Solubility

g/mol

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