ROCK
ROCK (Rho-associated protein kinase) is a kinase belonging to the AGC family of serine-threonine kinases and takes part in regulating the shape and movement of cells by acting on the cytoskeleton.
Products Related to ROCK(76)
| Catalog No. | Product Name | CAS No. | Purity | Structure |
|---|---|---|---|---|
| GC13423 | Y-39983 dihydrochloride | 173897-44-4 | >98.50% | |
ROCK family inhibitor | ||||
| GC15712 | Y-27632 | 146986-50-7 | >98.00% | |
Un inhibidor de ROCK, potente y selectivo. | ||||
| GC10722 | SR-3677 | 1072959-67-1 | >99.50% | |
SR-3677 es un inhibidor de ROCK-II potente y selectivo con una IC50 de ~3 nM. | ||||
| GC13869 | Fasudil | 103745-39-7 | >98.00% | |
Fasudil es un inhibidor no específico de RhoA/ROCK con un Ki de 0.33μM y un IC50 de 0.158μM para ROCK1, y un IC50 de 4.58μM, 12.30μM y 1.650μM para ROCK2, PKA, PKC y PKG, respectivamente. | ||||
