GLPBio

TBK1 ligand 3

Catalog No.: GC79809Purity:>99.00%
COASDSData Sheet
TBK1 ligand 3 is a TBK1 ligand, which can be used as a target protein ligand for the synthesis of PROTAC UNC8209 and UNC8461 [1].

Products are for research use only. Not for human use. We do not sell to patients.

TBK1 ligand 3
Cas No.: 2115897-10-2
10mM (in 1mL DMSO)In Stock
$488.00
1
1mgIn Stock
$178.00
1
5mgIn Stock
$444.00
1
Tel: (909) 407-4943 / (909) 689-7124Email: sales@glpbio.com

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    641, 529–536 (2025)
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    610, 366–372 (2022)
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    Cell
    187(9):2288-2304 (2024)
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    Cell
    183(7):1867-1883 (2020)
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    388(6745) (2025)
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    Cell Research
    35, 97–116 (2025)
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    34, 683–706 (2024)
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    33, 546–561 (2023)
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    33, 904–922 (2023)
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    31, 1291–1307 (2021)

Description

TBK1 ligand 3 is a TBK1 ligand, which can be used as a target protein ligand for the synthesis of PROTAC UNC8209 and UNC8461 [1].

References:
[1]. Liao C, et al. Selective degradation of TBK1 uncovers mechanistic insights into blocking ccRCC progression. Cell Chem Biol. 2026 Apr 16;33(4):461-473.e7.

Product Documents

Purity:>99.00%Appearance:A solid
COASDSData Sheet

Chemical Properties

CAS No.
2115897-10-2
Molecular Formula
C19H24BrN5O2
Molecular Weight
434.33
Solubility
DMSO: ≥ 100 mg/mL (230.24 mM)
Storage
Store at 4°C, stored under nitrogen
Shipping Condition
Evaluation samples are shipped with blue ice. Other available sizes are shipped at room temperature or with blue ice upon request.

CalculatorsMolarity / Dilution / Molecular Weight / Unit Conversion / In Vivo Formulation / Solubility

g/mol

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