GLPBio

TRPV1

TRPV1 (transient receptor potential vanilloid 1) is a calcium permeant cation channel that detects thermal stimuli and noxious chemical. It is a drug target for analgesics.

Products Related to TRPV1(10)

  • GC13003 structure
    GC13003AMG-517
    CAS: 659730-32-2
    Purity: >99.50%

    TRPV1 antagonist,potent and highly selective

  • GC14580 structure
    GC14580SB705498
    CAS: 501951-42-4
    Purity: >99.50%

    SB705498 is an orally bioavailable, competitive antagonist of the capsaicin-mediated of TRPV1 receptors (pKis = 7.6; 7.5; and 7.3 for human, rat, and guinea pig, respectively).SB705498 rapidly and reversibly inhibits capsaicin-, acid-, or heat-mediated activation of human TRPV1.

  • GC11147 structure
    GC11147Oleoyl Serotonin
    CAS: 1002100-44-8
    Purity: >98%

    TRPV1 channel inhibitor

  • GC12097 structure
    GC12097Palmitoyl Serotonin
    CAS: 212707-51-2
    Purity: >98.00%

    TRPV1 channel inhibitor

  • GC12636 structure
    GC12636Capsiconiate
    CAS: 946572-73-2
    Purity: >98%

    TRPV1 agonist

  • GC12772 structure
    GC12772Eicosapentaenoyl Serotonin
    CAS: 199875-71-3
    Purity: >98%

    TRPV1 channel inhibitor

  • GC14761 structure
    GC14761Mavatrep
    CAS: 956274-94-5
    Purity: >99.50%

    TRPV1 antagonist

  • GC15580 structure
    GC15580Stearoyl Serotonin
    CAS: 67964-87-8
    Purity: >98%

    TRPV1 channel inhibitor

  • GC16627 structure
    GC16627Docosahexaenoyl Serotonin
    CAS: 283601-58-1
    Purity: >98%

    TRPV1 channel inhibitor

  • GC17918 structure
    GC17918Capsazepine
    CAS: 138977-28-3
    Purity: >99.00%

    Capsazepine is a specific antagonist of the transient receptor potential vanilloid 1 (TRPV1) receptor with an IC 50 value of 562nM.