Urotensin Receptor
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Urotensin receptor (UT) is a G-protein coupled receptor which binds the peptide hormoneurotensin. The urotensin-II (UT) receptor is a Gq/11-protein-coupled receptor that mediates complex hemodynamic effects and influences neuromuscular physiology. The UT receptor displays greatest expression levels in the peripheral vasculature, heart and kidney, although they are found elsewhere, notably the central nervous system, at lower levels. The UT receptor produces potent but variable vasoconstrictor effects in some vascular beds, yet mediates vasodilation in others; it has also been implicated in osmoregulation.
Products Related to Urotensin Receptor(7)
- GC34236Urotensin II, mouseCAS: 405137-01-1Purity: >98%
Urotensin II, mouse is an endogenous ligand for the orphan G-protein-coupled receptor GPR14 or SENR.
- GC37871Urotensin II (114-124), human TFACAS: 251293-28-4Purity: >98.00%
Urotensin II (114-124), human TFA is an 11-amino-acid peptide that stimulates its obligatory G protein-coupled urotensin II receptors (UT), by binding to the orphan G-protein-coupled receptor 14 (GPR14) to modulate cardiovascular function in humans.
- GC39578Urotensin II, mouse TFAPurity: >99.50%
Urotensin II, mouse TFA is an endogenous ligand for the orphan G-protein-coupled receptor GPR14 or SENR.
- GC61546Palosuran hydrochlorideCAS: 2469274-58-4Purity: >98.50%
Palosuran hydrochloride (ACT-058362 hydrochloride) is a potent, selective, and orally active antagonist of urotensin II receptor, with an IC50 of 3.6 nM for CHO cell membranes expressing human recombinant receptors.
- GC62225Urotensin II, mouse acetatePurity: >99.50%
Urotensin II, mouse acetate is an endogenous ligand for the orphan G-protein-coupled receptor GPR14 or SENR.
| Catalog No. | Product Name | CAS No. | Purity | Structure |
|---|---|---|---|---|
| GC17414 | Palosuran | 540769-28-6 | >99.00% | |
Urotensin-II receptor antagonist | ||||
| GC34236 | Urotensin II, mouse | 405137-01-1 | >98% | |
Urotensin II, mouse is an endogenous ligand for the orphan G-protein-coupled receptor GPR14 or SENR. | ||||
| GC37871 | Urotensin II (114-124), human TFA | 251293-28-4 | >98.00% | |
Urotensin II (114-124), human TFA is an 11-amino-acid peptide that stimulates its obligatory G protein-coupled urotensin II receptors (UT), by binding to the orphan G-protein-coupled receptor 14 (GPR14) to modulate cardiovascular function in humans. | ||||
| GC39578 | Urotensin II, mouse TFA | - | >99.50% | |
Urotensin II, mouse TFA is an endogenous ligand for the orphan G-protein-coupled receptor GPR14 or SENR. | ||||
| GC50138 | Urantide | 669089-53-6 | >98% | |
Urantide is a selective and competitive urotensin-II (UT) receptor antagonist, with the pK B value of 8.32. | ||||
| GC61546 | Palosuran hydrochloride | 2469274-58-4 | >98.50% | |
Palosuran hydrochloride (ACT-058362 hydrochloride) is a potent, selective, and orally active antagonist of urotensin II receptor, with an IC50 of 3.6 nM for CHO cell membranes expressing human recombinant receptors. | ||||
| GC62225 | Urotensin II, mouse acetate | - | >99.50% | |
Urotensin II, mouse acetate is an endogenous ligand for the orphan G-protein-coupled receptor GPR14 or SENR. | ||||