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GPCR/G protein

  1. Cat.No. Product Name Information
  2. GN10652 Norisoboldine Norisoboldine  Chemical Structure
  3. GN10542 Scopolamine butylbromide Scopolamine butylbromide  Chemical Structure
  4. GN10507 Baohuoside I Baohuoside I  Chemical Structure
  5. GN10489 Hyodeoxycholic acid Hyodeoxycholic acid  Chemical Structure
  6. GN10419 Ligustroflavone Ligustroflavone  Chemical Structure
  7. GN10285 Theobromine Theobromine  Chemical Structure
  8. GN10169 3-Hydroxy-4-methoxycinnamic acid 3-Hydroxy-4-methoxycinnamic acid  Chemical Structure
  9. GN10112 Ginsenoside Rb2 Ginsenoside Rb2  Chemical Structure
  10. GN10104 Gramine Gramine  Chemical Structure
  11. GN10069 Ginsenoside Ro Ginsenoside Ro  Chemical Structure
  12. GN10606 Yohimbine Hydrochloride

    An α2-adrenoceptor antagonist

    Yohimbine Hydrochloride  Chemical Structure
  13. GC14860 Oncrasin 1 An anticancer agent Oncrasin 1  Chemical Structure
  14. GC17421 Vicriviroc maleate A CCR5 antagonist Vicriviroc maleate  Chemical Structure
  15. GC11238 Verlukast Leukotriene D4 antagonist Verlukast  Chemical Structure
  16. GC11831 Umeclidinium bromide A muscarinic acetylcholine receptor antagonist Umeclidinium bromide  Chemical Structure
  17. GC16054 TUG-770 An agonist of FFA1/GPR40 TUG-770  Chemical Structure
  18. GC15973 Tozadenant An adenosine A2A receptor antagonist Tozadenant  Chemical Structure
  19. GC12554 Tiotropium Bromide A muscarinic receptor antagonist Tiotropium Bromide  Chemical Structure
  20. GC15574 Taranabant A CB1 receptor inverse agonist Taranabant  Chemical Structure
  21. GC16026 Talnetant A nonpeptide NK3 antagonist Talnetant  Chemical Structure
  22. GC18123 TAK-700 salt Androgen synthesis inhibitor TAK-700 salt  Chemical Structure
  23. GC16377 SRT3190 SRT3190  Chemical Structure
  24. GC16710 SRT3109 SRT3109  Chemical Structure
  25. GC13549 Setiptiline maleate Setiptiline maleate  Chemical Structure
  26. GC13990 Setiptiline Setiptiline  Chemical Structure
  27. GC15401 SCH 563705 SCH 563705  Chemical Structure
  28. GC16100 SCH 527123 An allosteric antagonist of CXCR1 and CXCR2 SCH 527123  Chemical Structure
  29. GC15534 SB-674042 A potent and selective orexin 1 receptor antagonist SB-674042  Chemical Structure
  30. GC16540 SB-408124 Hydrochloride A potent orexin 1 receptor antagonist SB-408124 Hydrochloride  Chemical Structure
  31. GC10107 SB-222200 An NK3 receptor antagonist SB-222200  Chemical Structure
  32. GC11531 Salmeterol xinafoate A long-acting β2-adrenergic receptor agonist Salmeterol xinafoate  Chemical Structure
  33. GC12188 Salmefamol β2-adrenergic receptor agonist Salmefamol  Chemical Structure
  34. GC10528 Salirasib A Ras inhibitor with anti-cancer and anti-atherogenic activity Salirasib  Chemical Structure
  35. GC15489 RS 504393 A CCR2 chemokine receptor antagonist RS 504393  Chemical Structure
  36. GC16017 Rotigotine hydrochloride A non-selective dopamine receptor agonist Rotigotine hydrochloride  Chemical Structure
  37. GC10614 Rotigotine A non-selective dopamine receptor agonist Rotigotine  Chemical Structure
  38. GC16466 Rimonabant hydrochloride A potent and selective CB1 receptor antagonist Rimonabant hydrochloride  Chemical Structure
  39. GC13813 Reparixin L-lysine salt Perifosine is an orally active alkyl phospholipid analogue that has shown antitumor activity in a variety of cancers by interfering . Reparixin L-lysine salt  Chemical Structure
  40. GC12849 Reparixin An allosteric inhibitor of CXCR1 and CXCR2 Reparixin  Chemical Structure
  41. GC11591 Preladenant An adenosine A2A receptor antagonist Preladenant  Chemical Structure
  42. GC17976 Phloretin A natural inhibitor of various transporters Phloretin  Chemical Structure
  43. GC11917 PF-543 A potent inhibitor of SPHK1 PF-543  Chemical Structure
  44. GC12200 Pentostatin A purine antimetabolite and an ADA inhibitor Pentostatin  Chemical Structure
  45. GC17384 PD 123319 ditrifluoroacetate A selective angiotensin II type 2 receptor antagonist PD 123319 ditrifluoroacetate  Chemical Structure
  46. GC14461 PB-22 Synthetic cannabinoid PB-22  Chemical Structure
  47. GC10843 Otenabant Otenabant  Chemical Structure
  48. GC16886 Orteronel A non-steroidal inhibitor of the 17,20-lyase activity of CYP17A1 Orteronel  Chemical Structure
  49. GC15662 ONO-AE3-208 An EP4 receptor antagonist ONO-AE3-208  Chemical Structure
  50. GC16936 Olmesartan An AT1 receptor antagonist and active metabolite of olmesartan medoxomil Olmesartan  Chemical Structure
  51. GC10899 Octreotide acetate A somatostatin receptor agonist Octreotide acetate  Chemical Structure
  52. GC12240 NPS-2143 hydrochloride An orally-active CaSR antagonist NPS-2143 hydrochloride  Chemical Structure
  53. GC11871 MTEP hydrochloride A selective mGlu5a receptor antagonist MTEP hydrochloride  Chemical Structure
  54. GC16172 MPEP Hydrochloride A potent, highly selective mGlu5a receptor antagonist MPEP Hydrochloride  Chemical Structure
  55. GC15006 MK-6892 MK-6892  Chemical Structure
  56. GC16477 MK-2894 MK-2894  Chemical Structure
  57. GC11636 MK-0812 A CCR2 antagonist MK-0812  Chemical Structure
  58. GC14793 MK 0893 MK 0893  Chemical Structure
  59. GC11954 mGlu2 agonist mGlu2 agonist  Chemical Structure
  60. GC13144 Medetomidine Medetomidine  Chemical Structure
  61. GC12514 MBX-2982 An agonist of GPR119 MBX-2982  Chemical Structure
  62. GC14555 LY341495 Selective antagonist of mGluR2 and mGluR3 LY341495  Chemical Structure
  63. GC15986 LUF6000 A positive allosteric modulator of adenosine A3 receptors LUF6000  Chemical Structure
  64. GC11833 Laropiprant A potent, selective DP1 receptor antagonist Laropiprant  Chemical Structure
  65. GC13808 Indacaterol A long-acting β2-adrenergic receptor agonist Indacaterol  Chemical Structure
  66. GC11994 INCB8761(PF-4136309) A CCR2 antagonist INCB8761(PF-4136309)  Chemical Structure
  67. GC10207 INCB3344 An antagonist of CCR2 INCB3344  Chemical Structure
  68. GC14821 INCB 3284 dimesylate An antagonist of the MCP-1 receptor CCR2 INCB 3284 dimesylate  Chemical Structure
  69. GC10287 Ibutamoren Mesylate

    A growth hormone secretagogue and ghrelin receptor agonist

    Ibutamoren Mesylate  Chemical Structure
  70. GC12243 HOKU-81 HOKU-81  Chemical Structure
  71. GC14027 GW-1100 A selective GPR40 antagonist GW-1100  Chemical Structure
  72. GC12132 Guanfacine hydrochloride An α2-adrenergic receptor agonist Guanfacine hydrochloride  Chemical Structure
  73. GC16016 GPR120 modulator 2 GPR120 modulator 2  Chemical Structure
  74. GC14836 GPR120 modulator 1 GPR120 modulator 1  Chemical Structure
  75. GC11399 Glucocorticoid receptor agonist Glucocorticoid receptor agonist  Chemical Structure
  76. GC13512 glucagon receptor antagonists 3 glucagon receptor antagonists 3  Chemical Structure
  77. GC12569 glucagon receptor antagonists 2 glucagon receptor antagonists 2  Chemical Structure
  78. GC15486 glucagon receptor antagonists 1 glucagon receptor antagonists 1  Chemical Structure
  79. GC13391 Exendin-4 Exendin-4  Chemical Structure
  80. GC10394 DY131 An ERRβ/γ agonist DY131  Chemical Structure
  81. GC16073 Dronedarone An antiarrhythmic agent Dronedarone  Chemical Structure
  82. GC16523 Dipraglurant Dipraglurant  Chemical Structure
  83. GC11265 Desmopressin Acetate Desmopressin Acetate  Chemical Structure
  84. GC12303 Desmopressin A vasopressin receptor agonist Desmopressin  Chemical Structure
  85. GC13076 Deltarasin A KRAS inhibitor Deltarasin  Chemical Structure
  86. GC13426 CPPHA A positive allosteric modulator of the mGluR5 CPPHA  Chemical Structure
  87. GC10822 Clozapine N-oxide (CNO) A metabolite of clozapine and muscarinic DREADD agonist Clozapine N-oxide (CNO)  Chemical Structure
  88. GC13518 Cinacalcet Cinacalcet  Chemical Structure
  89. GC10172 CGS 21680 A selective agonist of the adenosine A2A receptor CGS 21680  Chemical Structure
  90. GC17157 Cevimeline hydrochloride hemihydrate Cevimeline hydrochloride hemihydrate  Chemical Structure
  91. GC14215 Cevimeline A muscarinic receptor agonist Cevimeline  Chemical Structure
  92. GC14412 CCG-63808 CCG-63808  Chemical Structure
  93. GC10658 CCG-63802 CCG-63802  Chemical Structure
  94. GC14935 Capadenoson A partial adenosine receptor agonist Capadenoson  Chemical Structure
  95. GC17244 Calcium-Sensing Receptor Antagonists I Calcium-Sensing Receptor Antagonists I  Chemical Structure
  96. GC14491 B-HT 920 A potent agonist of D2 receptors B-HT 920  Chemical Structure
  97. GC15926 BAN ORL 24 A nociceptin receptor antagonist BAN ORL 24  Chemical Structure
  98. GC11405 Avosentan Avosentan  Chemical Structure
  99. GC11783 Atrasentan hydrochloride Atrasentan hydrochloride  Chemical Structure
  100. GC13253 Anamorelin A small molecule agonist of GHS-R1a Anamorelin  Chemical Structure
  101. GC17018 AMD-070 hydrochloride CXCR4 antagonist,potent and selective AMD-070 hydrochloride  Chemical Structure

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