GPCR/G protein
- Neuropeptide FF/AF Receptors(40)
- Neuropeptide S Receptor(1)
- GPBA Receptor(1)
- Trace Amine 1 Receptor(2)
- GPCR protein(1)
- FFAR3(1)
- Formyl Peptide Receptors(11)
- 5-HT Receptor(364)
- Acetylcholine(19)
- Adenosine Deaminase(10)
- Adenosine Receptor(121)
- Adenosine Kinase(4)
- Adiponectin Receptor(3)
- Adrenergic Receptor(376)
- Adrenergic Transporters(5)
- Apelin Receptor(9)
- Angiotensin Receptor(98)
- Bombesin Receptors(22)
- Bradykinin Receptors(26)
- Calcitonin and Related Receptors(10)
- Cannabinoid Receptor(97)
- Calcimimetic Agent(2)
- CaSR(19)
- CCK1 Receptors(7)
- CCK2 Receptors(7)
- CCR(66)
- Chemokine Receptors(25)
- CRF1 Receptors(9)
- CRF2 Receptors(3)
- CXCR(65)
- CysLT1 receptor(1)
- Endothelin Receptor(46)
- EP1 Receptor(2)
- EP4 Receptor(2)
- ERRγ(1)
- ETA Receptors(5)
- ETB Receptors(5)
- Free Fatty Acid Receptors(16)
- Galanin Receptors(11)
- Ghrelin Receptors(11)
- GHSR(18)
- GIP Receptor(5)
- Glucagon Receptor(58)
- Glucocorticoid Receptor(79)
- GLUT1(1)
- Gonadotropin-Releasing Hormone Receptors(3)
- GPCR19(12)
- GPR109A(3)
- GPR119(10)
- GPR120(9)
- GPR35(8)
- GPR44(1)
- GPR55(8)
- Hydroxycarboxylic Acid Receptors(5)
- Leukotriene Receptor(54)
- LPA Receptor(12)
- LPL Receptor(54)
- LTD4 Receptor(1)
- mGluR (102)
- Melanin-concentrating Hormone Receptors(7)
- Melanocortin (MC) Receptors(43)
- Melatonin Receptors(22)
- Motilin Receptor(6)
- MT Receptor(1)
- Non-selective CRF(7)
- Neurotensin Receptors(17)
- NK2 Receptors(7)
- NK3 Receptor(5)
- NOP Receptor(20)
- NPY Receptors(26)
- Orexin(3)
- Orphan 7-TM Receptors(6)
- OX Receptor(38)
- Oxytocin Receptors(20)
- P2Y Receptor(53)
- PACAP Receptors(3)
- PAF Receptors(7)
- Peptide Receptors(14)
- PGD2 Receptor(1)
- Prostaglandin Receptor(157)
- Prostanoid Receptors(25)
- Protease-Activated Receptors(10)
- RGS(2)
- S1P receptor(8)
- Secretin Receptors(1)
- Sensory Neuron-Specific Receptors(1)
- Somatostatin Receptor(32)
- Sigma Receptor(53)
- Vasopressin Receptor(29)
- 17,20-lyase(4)
- Ras(101)
- Urotensin-II Receptor(11)
- VIP Receptors(6)
- EBI2/GPR183(5)
- TSH Receptor(10)
- NK Receptor(1)
- GPR81(1)
- C3aR(1)
- CysLT2 receptor(1)
- S1P receptor inhibitor(22)
- CCKB(1)
- FFAR1 (GPR40)(20)
- GPR84(4)
- Neuromedin U Receptors(2)
- Kisspeptin Receptor(4)
- CRFR(21)
- RGS Protein(5)
- Urotensin Receptor(6)
- Cholecystokinin Receptor(23)
- GPR139(2)
- mAChR(168)
- MCHR1 (GPR24)(16)
- Neurokinin Receptor(67)
- cGMP(18)
- GRK(1)
- Cat.No. Product Name Information
-
GN10652
Norisoboldine
-
GN10542
Scopolamine butylbromide
-
GN10507
Baohuoside I
-
GN10489
Hyodeoxycholic acid
-
GN10419
Ligustroflavone
-
GN10285
Theobromine
-
GN10169
3-Hydroxy-4-methoxycinnamic acid
-
GN10112
Ginsenoside Rb2
-
GN10104
Gramine
-
GN10069
Ginsenoside Ro
-
GN10606
Yohimbine Hydrochloride
An α2-adrenoceptor antagonist
-
GC14860
Oncrasin 1
An anticancer agent
-
GC17421
Vicriviroc maleate
A CCR5 antagonist
-
GC11238
Verlukast
Leukotriene D4 antagonist
-
GC11831
Umeclidinium bromide
A muscarinic acetylcholine receptor antagonist
-
GC16054
TUG-770
An agonist of FFA1/GPR40
-
GC15973
Tozadenant
An adenosine A2A receptor antagonist
-
GC12554
Tiotropium Bromide
A muscarinic receptor antagonist
-
GC15574
Taranabant
A CB1 receptor inverse agonist
-
GC16026
Talnetant
A nonpeptide NK3 antagonist
-
GC18123
TAK-700 salt
Androgen synthesis inhibitor
-
GC16377
SRT3190
-
GC16710
SRT3109
-
GC13549
Setiptiline maleate
-
GC13990
Setiptiline
-
GC15401
SCH 563705
-
GC16100
SCH 527123
An allosteric antagonist of CXCR1 and CXCR2
-
GC15534
SB-674042
A potent and selective orexin 1 receptor antagonist
-
GC16540
SB-408124 Hydrochloride
A potent orexin 1 receptor antagonist
-
GC10107
SB-222200
An NK3 receptor antagonist
-
GC11531
Salmeterol xinafoate
A long-acting β2-adrenergic receptor agonist
-
GC12188
Salmefamol
β2-adrenergic receptor agonist
-
GC10528
Salirasib
A Ras inhibitor with anti-cancer and anti-atherogenic activity
-
GC15489
RS 504393
A CCR2 chemokine receptor antagonist
-
GC16017
Rotigotine hydrochloride
A non-selective dopamine receptor agonist
-
GC10614
Rotigotine
A non-selective dopamine receptor agonist
-
GC16466
Rimonabant hydrochloride
A potent and selective CB1 receptor antagonist
-
GC13813
Reparixin L-lysine salt
Perifosine is an orally active alkyl phospholipid analogue that has shown antitumor activity in a variety of cancers by interfering .
-
GC12849
Reparixin
An allosteric inhibitor of CXCR1 and CXCR2
-
GC11591
Preladenant
An adenosine A2A receptor antagonist
-
GC17976
Phloretin
A natural inhibitor of various transporters
-
GC11917
PF-543
A potent inhibitor of SPHK1
-
GC12200
Pentostatin
A purine antimetabolite and an ADA inhibitor
-
GC17384
PD 123319 ditrifluoroacetate
A selective angiotensin II type 2 receptor antagonist
-
GC14461
PB-22
Synthetic cannabinoid
-
GC10843
Otenabant
-
GC16886
Orteronel
A non-steroidal inhibitor of the 17,20-lyase activity of CYP17A1
-
GC15662
ONO-AE3-208
An EP4 receptor antagonist
-
GC16936
Olmesartan
An AT1 receptor antagonist and active metabolite of olmesartan medoxomil
-
GC10899
Octreotide acetate
A somatostatin receptor agonist
-
GC12240
NPS-2143 hydrochloride
An orally-active CaSR antagonist
-
GC11871
MTEP hydrochloride
A selective mGlu5a receptor antagonist
-
GC16172
MPEP Hydrochloride
A potent, highly selective mGlu5a receptor antagonist
-
GC15006
MK-6892
-
GC16477
MK-2894
-
GC11636
MK-0812
A CCR2 antagonist
-
GC14793
MK 0893
-
GC11954
mGlu2 agonist
-
GC13144
Medetomidine
-
GC12514
MBX-2982
An agonist of GPR119
-
GC14555
LY341495
Selective antagonist of mGluR2 and mGluR3
-
GC15986
LUF6000
A positive allosteric modulator of adenosine A3 receptors
-
GC11833
Laropiprant
A potent, selective DP1 receptor antagonist
-
GC13808
Indacaterol
A long-acting β2-adrenergic receptor agonist
-
GC11994
INCB8761(PF-4136309)
A CCR2 antagonist
-
GC10207
INCB3344
An antagonist of CCR2
-
GC14821
INCB 3284 dimesylate
An antagonist of the MCP-1 receptor CCR2
-
GC10287
Ibutamoren Mesylate
A growth hormone secretagogue and ghrelin receptor agonist
-
GC12243
HOKU-81
-
GC14027
GW-1100
A selective GPR40 antagonist
-
GC12132
Guanfacine hydrochloride
An α2-adrenergic receptor agonist
-
GC16016
GPR120 modulator 2
-
GC14836
GPR120 modulator 1
-
GC11399
Glucocorticoid receptor agonist
-
GC13512
glucagon receptor antagonists 3
-
GC12569
glucagon receptor antagonists 2
-
GC15486
glucagon receptor antagonists 1
-
GC13391
Exendin-4
-
GC10394
DY131
An ERRβ/γ agonist
-
GC16073
Dronedarone
An antiarrhythmic agent
-
GC16523
Dipraglurant
-
GC11265
Desmopressin Acetate
-
GC12303
Desmopressin
A vasopressin receptor agonist
-
GC13076
Deltarasin
A KRAS inhibitor
-
GC13426
CPPHA
A positive allosteric modulator of the mGluR5
-
GC10822
Clozapine N-oxide (CNO)
A metabolite of clozapine and muscarinic DREADD agonist
-
GC13518
Cinacalcet
-
GC10172
CGS 21680
A selective agonist of the adenosine A2A receptor
-
GC17157
Cevimeline hydrochloride hemihydrate
-
GC14215
Cevimeline
A muscarinic receptor agonist
-
GC14412
CCG-63808
-
GC10658
CCG-63802
-
GC14935
Capadenoson
A partial adenosine receptor agonist
-
GC17244
Calcium-Sensing Receptor Antagonists I
-
GC14491
B-HT 920
A potent agonist of D2 receptors
-
GC15926
BAN ORL 24
A nociceptin receptor antagonist
-
GC11405
Avosentan
-
GC11783
Atrasentan hydrochloride
-
GC13253
Anamorelin
A small molecule agonist of GHS-R1a
-
GC17018
AMD-070 hydrochloride
CXCR4 antagonist,potent and selective