GPCR/G protein
- Neuropeptide FF/AF Receptors(40)
- Neuropeptide S Receptor(1)
- GPBA Receptor(1)
- Trace Amine 1 Receptor(2)
- GPCR protein(1)
- FFAR3(1)
- Formyl Peptide Receptors(11)
- 5-HT Receptor(387)
- Acetylcholine(19)
- Adenosine Deaminase(9)
- Adenosine Receptor(116)
- Adenosine Kinase(4)
- Adiponectin Receptor(3)
- Adrenergic Receptor(358)
- Adrenergic Transporters(5)
- Apelin Receptor(9)
- Angiotensin Receptor(96)
- Bombesin Receptors(22)
- Bradykinin Receptors(26)
- Calcitonin and Related Receptors(10)
- Cannabinoid Receptor(127)
- Calcimimetic Agent(2)
- CaSR(18)
- CCK1 Receptors(7)
- CCK2 Receptors(7)
- CCR(61)
- Chemokine Receptors(25)
- CRF1 Receptors(9)
- CRF2 Receptors(3)
- CXCR(64)
- CysLT1 receptor(1)
- Endothelin Receptor(45)
- EP1 Receptor(2)
- EP4 Receptor(3)
- ERRγ(1)
- ETA Receptors(5)
- ETB Receptors(5)
- Free Fatty Acid Receptors(18)
- Galanin Receptors(11)
- Ghrelin Receptors(12)
- GHSR(19)
- GIP Receptor(5)
- Glucagon Receptor(59)
- Glucocorticoid Receptor(80)
- GLUT1(1)
- Gonadotropin-Releasing Hormone Receptors(3)
- GPCR19(12)
- GPR109A(3)
- GPR119(10)
- GPR120(9)
- GPR35(7)
- GPR44(1)
- GPR55(9)
- Hydroxycarboxylic Acid Receptors(5)
- Leukotriene Receptor(54)
- LPA Receptor(13)
- LPL Receptor(49)
- LTD4 Receptor(1)
- mGluR (96)
- Melanin-concentrating Hormone Receptors(7)
- Melanocortin (MC) Receptors(42)
- Melatonin Receptors(21)
- Motilin Receptor(6)
- MT Receptor(1)
- Non-selective CRF(7)
- Neurotensin Receptors(17)
- NK2 Receptors(7)
- NK3 Receptor(6)
- NOP Receptor(21)
- NPY Receptors(27)
- Orexin(3)
- Orphan 7-TM Receptors(6)
- OX Receptor(34)
- Oxytocin Receptors(20)
- P2Y Receptor(53)
- PACAP Receptors(3)
- PAF Receptors(8)
- Peptide Receptors(15)
- PGD2 Receptor(1)
- Prostaglandin Receptor(149)
- Prostanoid Receptors(25)
- Protease-Activated Receptors(10)
- RGS(2)
- S1P receptor(8)
- Secretin Receptors(1)
- Sensory Neuron-Specific Receptors(1)
- Somatostatin Receptor(33)
- Sigma Receptor(52)
- Vasopressin Receptor(28)
- 17,20-lyase(5)
- Ras(89)
- Urotensin-II Receptor(11)
- VIP Receptors(7)
- EBI2/GPR183(4)
- TSH Receptor(8)
- NK Receptor(1)
- GPR81(1)
- C3aR(1)
- CysLT2 receptor(1)
- S1P receptor inhibitor(22)
- CCKB(1)
- FFAR1 (GPR40)(22)
- GPR84(4)
- Neuromedin U Receptors(2)
- Kisspeptin Receptor(4)
- CRFR(19)
- RGS Protein(5)
- Urotensin Receptor(6)
- Cholecystokinin Receptor(23)
- GPR139(1)
- mAChR(160)
- MCHR1 (GPR24)(16)
- Neurokinin Receptor(65)
- cGMP(18)
- GRK(1)
Products for GPCR/G protein
- Cat.No. Product Name Information
-
GC38007
β-Melanocyte Stimulating Hormone (MSH), human TFA
-
GC40105
βARK1 Inhibitor
βARK1 inhibitor is an inhibitor of G protein-coupled receptor kinase 2/β-adrenergic receptor kinase 1 (GRK2/βARK1; IC50 = 126 μM).
-
GC61462
γ-1-Melanocyte Stimulating Hormone (MSH), amide
-
GC17002
γ1-MSH
melanocortin MC3 receptor agonist
-
GC62708
σ1 Receptor antagonist-1
-
GC15519
α-CGRP (human)
Endogenous calcitonin gene-related peptide receptor (CGRP) agonist
-
GC11346
α-helical CRF 9-41
Antagonist of corticotropin releasing factor receptor
-
GC11577
α-Methyl-5-hydroxytryptamine maleate
5-HT2B receptor agonist
-
GC31237
α1 adrenoceptor-MO-1
-
GC33681
β-Caryophyllene ((−)-trans-Caryophyllene)
-
GC33693
β-Melanocyte Stimulating Hormone (MSH), human (Beta-MSH (1-22) (human))
-
GC31573
β3-AR agonist 2
-
GC34231
γ-1-Melanocyte Stimulating Hormone (MSH), amide
-
GC17413
(±)-5'-Chloro-5'-deoxy-ENBA
adenosine A1 receptor agonist, selective and high-affinity
-
GC17408
(±)-AC 7954 hydrochloride
urotensin-II (UT) receptor agonist
-
GC15045
(±)-AMG 487
CXCR3 antagonist
-
GC41668
(±)-Clopidogrel (hydrochloride)
Clopidogrel is an antithrombic compound whose active metabolite is a selective, irreversible antagonist of the platelet purinergic P2Y12 receptor (IC50 = 100 nM).
-
GC16838
(±)-Cloprostenol sodium salt
prostaglandin F2α (PGF2α) analog,FP receptor agonist
-
GC18090
(±)-J 113397
NOP receptor antagonist
-
GC62727
(±)-Penbutolol-d9 hydrochloride
-
GC15144
(±)-PPCC oxalate
sigma (σ) receptor ligand
-
GC10907
(±)-SLV 319
CB1 receptor antagonist,potent and selective
-
GC12394
(±)-trans-ACPD
metabotropic glutamate receptors agonist
-
GC32523
(±)-Befunolol
-
GC34957
(+)-Cevimeline hydrochloride hemihydrate
-
GC30743
(+)-Cloprostenol (D-Cloprostenol)
-
GC45259
(+)-Cloprostenol (sodium salt)
(+)-Cloprostenol (sodium salt) is a more water soluble, crystalline form of (+)-cloprostenol.
-
GC12750
(+)-Fluprostenol
Prostaglandin F2α (FP) receptor agonist
-
GC18146
(+)-Igmesine hydrochloride
σ1 receptor ligand
-
GC31597
(+)-Penbutolol ((R)-Penbutolol)
-
GC17301
(+)-SK&F 10047 hydrochloride
prototypical σ1 receptor agonist
-
GC10675
(+,-)-Octopamine HCl
adrenoceptor agonist
-
GC50245
(+/-)-ADX 71743
Negative allosteric modulator of mGlu7 receptors; brain penetrant
-
GC50048
(+/-)-PPCC oxalate
Selective sigma (σ) agonist (σ1> σ2)
-
GC61646
(-)-Camphoric acid
-
GC16919
(1R,1'S,3'R/1R,1'R,3'S)-L-054,264
somatostatin sst2 receptor agonist
-
GC34963
(1R,2S)-VU0155041
-
GC34965
(20S)-Protopanaxatriol
-
GC38712
(2R,3R)-E1R
-
GC38713
(2R,3S)-E1R
-
GC38714
(2S,3S)-E1R
-
GC32644
(4E)-SUN9221
-
GA20063
(D-Ala²)-Gastric Inhibitory Polypeptide (human)
GIP receptor agonist.
-
GA20084
(Deamino-Cys¹,β-cyclohexyl-Ala⁴,Arg⁸)-Vasopressin
Studies revealed that this specific vasopressin agonist exhibited a nanomolar affinity for V-1b receptors from various mammalian species (bovine, human, rat). It exhibited high V-1b/V-1a and V-1b/oxytocin selectivity for rat, human, and bovine receptors. Furthermore, it showed a high V-1b/V-2 specificity for both bovine and human vasopressin receptors. Therefore, d(Cha?)-AVP is a promising tool for research of V-1b receptor structure-function relationships.
-
GA20195
(Gly¹,Ser³·²²,Gln⁴·³⁴,Thr⁶,Arg¹⁹,Tyr²¹,Ala²³·³¹,Aib³²)-Pancreatic Polypeptide (human)
This (Ala-Aib)-containing pancreatic peptide/neuropeptide Y chimera is a highly selective neuropeptide Y? receptor agonist. At this receptor this compound turned out to be 25-fold more potent than the derivative H-5084 (0.24 nM vs 6 nM) and three-fold more potent than the native ligand neuropeptide Y (H-6375) (0.24 nM vs 0.6 nM). This analog turned out to increase feeding approximately 2.5-fold more effective than neuropeptide Y.
-
GA20221
(Hyp³)-Bradykinin
Bradykinin antagonist.
-
GA20229
(Leu³¹,Pro³⁴)-Neuropeptide Y (human, rat)
Specific Y? receptor agonist.
-
GC11952
(R)-(+)-Atenolol
less active enantiomer of the racemic β1-adrenergic receptor antagonist, (R,S)-atenolol.
-
GC10608
(R)-(+)-Propranolol hydrochloride
β-adrenoceptor antagonist
-
GC11219
(R)-(+)-Tolterodine
Muscarinic receptor antagonists
-
GC12144
(R)-(-)-Niguldipine hydrochloride
L-type Ca2+ channel blocker and α1A-adrenoceptor antagonist
-
GC34985
(R)-ADX-47273
-
GC60001
(R)-Carvedilol
-
GC10028
(R)-SLV 319
CB1 receptor antagonist
-
GC39298
(R)-Terazosin
-
GC50426
(R)-ZINC 3573
MRGPRX2 agonist
-
GC62588
(R,R)-CXCR2-IN-2
-
GC34995
(R,R)-Palonosetron Hydrochloride
-
GC12823
(R,S)-Atenolol
β1-adrenergic receptor antagonist
-
GC63452
(Rac)-5-Hydroxymethyl Tolterodine
-
GC19541
(rac)-Antineoplaston A10
(rac)-Antineoplaston A10 is the racemate of Antineoplaston A10
-
GC62642
(rac)-Dobutamine-d6 hydrochloride
-
GC38721
(Rac)-E1R
-
GC63410
(Rac)-MRI-1867
-
GC62228
(rac)-Nebivolol-d4
-
GC34367
(RS)-Butyryltimolol
-
GC12279
(RS)-MCPG
mGluR antagonist
-
GC15292
(S)-(+)-Niguldipine hydrochloride
L-type Ca2+ channel blocker and α1A-adrenoceptor antagonist
-
GC12463
(S)-(-)-Atenolol
β-adrenergic blocker
-
GC15039
(S)-(-)-Pindolol
beta-adrenergic antagonist
-
GC16637
(S)-(-)-Propranolol hydrochloride
β-adrenoceptor antagonist
-
GC60006
(S)-Carvedilol
-
GC35002
(S)-Mapracorat
-
GC16349
(S)-MCPG
mGluR antagonist
-
GC10753
(S)-SLV 319
CB1 receptor antagonist
-
GC39249
(S)-Terazosin
-
GC60425
(S)-Verapamil D7 hydrochloride
-
GC60008
(S)-Verapamil hydrochloride
-
GA20291
(Sar¹)-Angiotensin II
The substitution with Sar at position 1 of angiotensin II resulted in a partial agonistic activity.
-
GC35011
(Z)-Thiothixene
-
GC16663
(±)-4-hydroxy Propranolol (hydrochloride)
β1- and β2-adrenergic receptors inhibitor
-
GC15087
(±)-Talinolol
β1-selective adrenoceptor antagonist
-
GC15528
(±)trans-2,5-bis-(3,4,5-Trimethoxyphenyl)-1,3-dioxolane
PAF receptor antagonist
-
GC10600
1,3-Dipropyl-8-phenylxanthine
A1 adenosine antagonist
-
GC12587
1-(1-Naphthyl) piperazine (hydrochloride)
ligand for 5-HT receptors
-
GC17913
1-Deazaadenosine
adenosine deaminase inhibitor
-
GC14607
1-Methylpsilocin
5-HT2C agonist,potent and selective
-
GC42011
1-Oleoyl Lysophosphatidic Acid
A potent LPA receptor agonist
-
GC15140
1-Oleoyl lysophosphatidic acid sodium salt
Activates LPA receptor
-
GC16876
1-Phenylbiguanide hydrochloride
5-HT3 receptor agonist
-
GC10821
11-keto-β-Boswellic Acid
leukotriene synthesis inhibitor via 5-lipoxygenase
-
GC41883
12(S)-HHTrE
12(S)-HHTrE is a product of the cyclooxygenase (COX) pathway and one of the primary arachidonic acid metabolites of human platelets.
-
GC16693
13Z,16Z-Docosadienoic Acid
FFAR4(GPR120) agonist
-
GC11133
16,16-Dimethyl Prostaglandin E2
derivative of prostaglandin E2
-
GC32770
1A-116
-
GC17757
1H-1-ethyl Candesartan Cilexetil
selective angiotensin II type 1 receptor (AT1) antagonist
-
GC11112
2'-MeCCPA
A1 adenosine receptor agonist
-
GC30561
2-(E-2-decenoylamino)ethyl 2-(cyclohexylethyl) sulfide
-
GC16403
2-Arachidonoyl Glycerol
An endogenous agonist of the cannabinoid (CB) receptors CB1 and CB2
-
GC10116
2-chloro-3-Deazaadenosine
adenosine receptors agonist