GLPBio

Vasorelaxant agent-2

Catalog No.: GC84373
COASDSData Sheet
Vasorelaxant agent-2 (Compound 8h) targets α1A-adrenergic receptor with an affinity of pD2=5.4.

Products are for research use only. Not for human use. We do not sell to patients.

Vasorelaxant agent-2
Cas No.: 53242-88-9
25mgIn Stock
$22.00
1
50mgIn Stock
$36.00
1
100mgIn Stock
$58.00
1
250mgIn Stock
$118.00
1
500mgIn Stock
$189.00
1
1gIn Stock
$304.00
1
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Citations

No citations are currently available for this product. Below are selected publications citing GlpBio products.
  • Nature cover
    Nature
    641, 529–536 (2025)
  • Nature cover
    Nature
    628, 630–638 (2024)
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    Nature
    632, 686–694 (2024)
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    Nature
    618, 1017–1023 (2023)
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    Nature
    610, 366–372 (2022)
  • Cell cover
    Cell
    187(9):2288-2304 (2024)
  • Cell cover
    Cell
    183(7):1867-1883 (2020)
  • Science cover
    Science
    388(6745) (2025)
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    Science
    387(6739) (2025)
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    Science
    387(6734) (2025)
  • Cell Research cover
    Cell Research
    35, 97–116 (2025)
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    Cell Research
    34, 683–706 (2024)
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    Cell Research
    33, 273–287 (2023)
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    Cell Research
    33, 546–561 (2023)
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    Cell Research
    33, 904–922 (2023)
  • Cell Research cover
    Cell Research
    31, 1291–1307 (2021)

Description

Vasorelaxant agent-2 (Compound 8h) targets α1A-adrenergic receptor with an affinity of pD2=5.4. Vasorelaxant agent-2 exhibits vasodilator activity in rats aortic rings with an EC 50 of 0.79 μM [1].

References:
[1]. del Olmo E, et al., Vasorelaxant activity of phthalazinones and related compounds. Bioorg Med Chem Lett. 2006 May 15;16(10):2786-90.

Product Documents

Appearance:A solid
COASDSData Sheet

Chemical Properties

CAS No.
53242-88-9
Molecular Formula
C15H11ClN2O
Molecular Weight
270.71
Storage
Store at RT, protect from light
Shipping Condition
Evaluation samples are shipped with blue ice. Other available sizes are shipped at room temperature or with blue ice upon request.

CalculatorsMolarity / Dilution / Molecular Weight / Unit Conversion / In Vivo Formulation / Solubility

g/mol

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