Pain Research

An α 2D -adrenergic receptor agonist

Salvinorin A carbamate is a potent κ-opioid receptor (KOR) full agonist that is almost as potent as salvinorin A with EC50 values of 6.2 and 4.5 nM, respectively, for activation of the human KOR to enhance binding of [35S]GTPγS.

Salvinorin A propionate is a selective partial agonist at κ1-opioid receptors (KOR) with a Ki value of 32.6 nM.

Salvinorin B mesylate (Mesyl Sal B) is a selective κ-opioid receptor agonist that is more potent than salvinorin A in CHO cells transfected with the human κ-opioid receptor (EC50s = 30 and 40 nM, respectively).

Vapreotide is a peptide neurokinin-1 receptor (NK1) antagonist and analog of somatostatin (IC50 = 330 nM in a radioligand binding assay).

WOBE437 is a potent endocannabinoid uptake inhibitor with IC50 values of 10 and 283 nM for arachidonoyl ethanolamide and 2-arachidonoyl glycerol uptake, respectively, in U937 cells.

Ziconotide is a synthetic version of ω-conopeptide MVIIA, a peptide toxin originally found in the venom of the fish-eating marine snail C.

β-endorphin (1-26) is a neuropeptide found in rat hippocampus, brain stem, and pituitary.

β-Endorphin (1-27) is an endogenous peptide that binds to μ-, δ-, and κ-opioid receptors (Kis = 5.31, 6.17, and 39.82 nM, respectively, in COS-1 cells expressing rat receptors).

An internal standard for the quantification of decanoic acid

Flupirtine-d4 (D 9998-d4) هيدروكلوريد هو الديوتيريوم المسمى Flupirtine.

A neuropeptide with diverse biological activities

An internal standard for the quantification of decanoic acid

Rofecoxib D5 (MK 966 D5) هو الديوتيريوم المسمى Rofecoxib

An internal standard for the quantification of phentolamine

An atypical sphingolipid

An internal standard for the quantification of decanoic acid

An angular pyranocoumarin with diverse biological activities

A neuropeptide with diverse biological activities