MK-0249 |
Katalog-Nr.GC31027 |
MK-0249 (Verbindung 1) ist ein potenter, selektiver und oral aktiver Histamin-H3-Rezeptor-Antagonist mit einem IC50-Wert von 1,7 nM fÜr menschliches H3.
Products are for research use only. Not for human use. We do not sell to patients.
Cas No.: 862309-06-6
Sample solution is provided at 25 µL, 10mM.
MK-0249 is a potent histamine H3 receptor antagonist, with Ki of 1.7 nM for human H3.
[1]. Brioni JD, et al. Discovery of histamine H3 antagonists for the treatment of cognitive disorders and Alzheimer's disease. J Pharmacol Exp Ther. 2011 Jan;336(1):38-46.
Average Rating: 5
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