NTRC 824 |
Katalog-Nr.GC50164 |
NTRC 824 (Verbindung 5) ist ein potenter, selektiver und Neurotensin-ähnlicher Antagonist des nichtpeptidischen Neurotensinrezeptors Typ 2 (NTS2) mit einem IC50 von 38 nM und einem Ki von 202 nM.
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Cas No.: 1623002-61-8
Sample solution is provided at 25 µL, 10mM.
Potent and selective non-peptide neurotensin (NTS) type-2 receptor antagonist (IC50 = 38 nM). Exhibits >150-fold selectivity for NTS2 over NTS1.
Thomas et al (2014) Identification of N-[(5-{[(4-methylphenyl)sulfonyl]amino}-3-(trifluoroacetyl)-1H-indol-1-yl)acetyl]-L-leucine (NTRC-824), a neurotensin-like nonpeptide compound selective for the neurotensin receptor type 2. J.Med.Chem. 57 7472 PMID:25157640
Average Rating: 5
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