VX-150 |
| Katalog-Nr.GC63259 |
VX-150 ist ein oral aktiver, hochselektiver NaV1.8-Inhibitor.
Products are for research use only. Not for human use. We do not sell to patients.
Cas No.: 1793080-72-4
Sample solution is provided at 25 µL, 10mM.
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VX-150 is an orally active, highly selective NaV1.8 inhibitor. VX-150 has the potential for various pain indications research[1].
VX-150 is an orally bioavailable pro-drug that rapidly converts into its active moiety, which is a highly selective inhibitor of NaV1.8 relative to the other sodium channel subtypes (>400-fold)[1].
[1]. Hemme J Hijma, et al. A Phase 1, Randomized, Double-Blind, Placebo-Controlled, Crossover Study to Evaluate the Pharmacodynamic Effects of VX-150, a Highly Selective NaV1.8 Inhibitor, in Healthy Male Adults. Pain Med. 2021 Aug 6;22(8):1814-1826.
Average Rating: 5 (Based on Reviews and 30 reference(s) in Google Scholar.)
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