Idelalisib D5 (Synonyms: CAL-101 D5; GS-1101 D5) |
カタログ番号GC62465 |
イデラリシブ D5 は、イデラリシブとラベル付けされた重水素です。イデラリシブは、選択性が高く、経口で生物学的に利用可能な p110δ 阻害剤です。
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Cas No.: 1830330-31-8
Sample solution is provided at 25 µL, 10mM.
Idelalisib D5 is a deuterium labeled Idelalisib. Idelalisib is a highly selective and orally bioavailable p110δ inhibitor[1].
[1]. Lannutti BJ, et al. CAL-101, a p110delta selective phosphatidylinositol-3-kinase inhibitor for the treatment of B-cell malignancies, inhibits PI3K signaling and cellular viability. Blood, 2011, 117(2), 591-594.
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