GLPBio

KDM4C-IN-2

Catalog No.: GC79157Purity:>98.00%
COASDSData Sheet
KDM4C-IN-2 is a histone lysine demethylase KDM4C ( JMJD2C ) inhibitor with an IC50 of 147 μM and a K i of 51 μM.

Products are for research use only. Not for human use. We do not sell to patients.

KDM4C-IN-2
Cas No.: 23705-85-3
100mgIn Stock
$18.00
1
250mgIn Stock
$31.00
1
1gIn Stock
$61.00
1
5gIn Stock
$195.00
1
Tel: (909) 407-4943 / (909) 689-7124Email: sales@glpbio.com

Citations

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    632, 686–694 (2024)
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    618, 1017–1023 (2023)
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    Nature
    610, 366–372 (2022)
  • Cell cover
    Cell
    187(9):2288-2304 (2024)
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    Cell
    183(7):1867-1883 (2020)
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    388(6745) (2025)
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    35, 97–116 (2025)
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    34, 683–706 (2024)
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    33, 904–922 (2023)
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    31, 1291–1307 (2021)

Description

KDM4C-IN-2 is a histone lysine demethylase KDM4C ( JMJD2C ) inhibitor with an IC50 of 147 μM and a K i of 51 μM. KDM4C-IN-2 can be used for the research of cancer, such as prostate and breast cancer [1].

In Vitro, KDM4C-IN-2 (Compound 2) (0.01-500 μM) shows no inhibitory effect on FDH[1].

References:
[1]. Leurs U, et al. Inhibitor scaffold for the histone lysine demethylase KDM4C (JMJD2C). Bioorg Med Chem Lett. 2012 Sep 15;22(18):5811-3.

Product Documents

Purity:>98.00%Appearance:A solid
COASDSData Sheet

Chemical Properties

CAS No.
23705-85-3
Molecular Formula
C7H8N2O5
Molecular Weight
200.15
Storage
Store at 4°C, stored under nitrogen
Shipping Condition
Evaluation samples are shipped with blue ice. Other available sizes are shipped at room temperature or with blue ice upon request.

CalculatorsMolarity / Dilution / Molecular Weight / Unit Conversion / In Vivo Formulation / Solubility

g/mol

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