PTKs/RTKs

Receptor tyrosine kinases transfer phosphate from ATP to protein. They play a vital role in various cellular processes including regulation of cell growth, proliferation, differentiation and metabolism etc.

Products Related to PTKs/RTKs(13)

GC13902 KRCA 0008
CAS: 1472795-20-2
Purity: >98.50%
Ack1 and anaplastic lymphoma kinase (ALK) dual inhibitor
GC14733 SU14813
CAS: 627908-92-3
Purity: >98.50%
A dual VEGFR and PDGFR family kinase inhibitor
GC16798 LDN-211904
CAS: 1198408-78-4
Purity: >98.00%
LDN-211904 (compound 32) is a potent and selective EphB3 inhibitor with an IC50 of 0.079 μM. LDN-211904 shows good metabolic stability in mouse liver microsomes. LDN-211904 with cetuximab could be effective in inhibiting STAT3-activated CSC stemness and cetuximab resistance in CRC.
GC36898 Phosphocreatine
CAS: 67-07-2
Purity: >90.00%
Phosphocreatine is a high-energy phosphate compound that is abundant in muscle and brain.
GC40927 Tilfrinib
CAS: 1600515-49-8
Purity: >98.00%
Tilfrinib is a selective Brk/PTK6 inhibitor with an IC₅₀ value of 3.15nM for Brk.
GC72930 XMU-MP-2
CAS: 2031152-10-8
Purity: >99.00%
XMU-MP-2 is a BRK inhibitor with significant inhibitory activity on BRK-positive cells.
GC72974 Entrectinib-d8
CAS: 2251773-94-9
Purity: >99.00%
Entrectinib-d8 (NMS-E628-d8; RXDX-101-d8) is a deuterated version of Entrectinib.
GC73232 PRDX1-IN-1
Purity: >98.00%
PRDX1-IN-1 is a selective inhibtor of PRDX1 with an IC50 value of 0.164 μM.
GC73482 PF-07284892
CAS: 2498597-94-5
Purity: >99.00%
PF-07284892 (ARRY-558) is a potent and orally active SHP2 inhibitor with an IC50 value of 21 nM.
GC73980 GGTI-2417
CAS: 501010-05-5
Purity: >98.00%
GGTI-2417 is a potent and selective inhibitor of GGTase I.
GC74371 Pinealon
CAS: 175175-23-2
Purity: >99.00%
Pinealon is a 3-amino acid peptide and shows neuroprotective properties.
GC81326 Tyrosine ethyl ester
CAS: 34081-17-9
Purity: >98%
Tyrosine ethyl ester exhibits antioxidant activity [1] .
GC81731 Hericene A
CAS: 157207-54-0
Purity: >98.50%
Hericene A is an orally active aromatic hericene derivative.

Category Product List
Catalog No.	Product Name	CAS No.	Purity
GC13902	KRCA 0008	1472795-20-2	>98.50%
GC13902	Ack1 and anaplastic lymphoma kinase (ALK) dual inhibitor
GC14733	SU14813	627908-92-3	>98.50%
GC14733	A dual VEGFR and PDGFR family kinase inhibitor
GC16798	LDN-211904	1198408-78-4	>98.00%
GC16798	LDN-211904 (compound 32) is a potent and selective EphB3 inhibitor with an IC50 of 0.079 μM. LDN-211904 shows good metabolic stability in mouse liver microsomes. LDN-211904 with cetuximab could be effective in inhibiting STAT3-activated CSC stemness and cetuximab resistance in CRC.
GC36898	Phosphocreatine	67-07-2	>90.00%
GC36898	Phosphocreatine is a high-energy phosphate compound that is abundant in muscle and brain.
GC40927	Tilfrinib	1600515-49-8	>98.00%
GC40927	Tilfrinib is a selective Brk/PTK6 inhibitor with an IC₅₀ value of 3.15nM for Brk.
GC72930	XMU-MP-2	2031152-10-8	>99.00%
GC72930	XMU-MP-2 is a BRK inhibitor with significant inhibitory activity on BRK-positive cells.
GC72974	Entrectinib-d8	2251773-94-9	>99.00%
GC72974	Entrectinib-d8 (NMS-E628-d8; RXDX-101-d8) is a deuterated version of Entrectinib.
GC73232	PRDX1-IN-1	-	>98.00%
GC73232	PRDX1-IN-1 is a selective inhibtor of PRDX1 with an IC50 value of 0.164 μM.
GC73482	PF-07284892	2498597-94-5	>99.00%
GC73482	PF-07284892 (ARRY-558) is a potent and orally active SHP2 inhibitor with an IC50 value of 21 nM.
GC73980	GGTI-2417	501010-05-5	>98.00%
GC73980	GGTI-2417 is a potent and selective inhibitor of GGTase I.
GC74371	Pinealon	175175-23-2	>99.00%
GC74371	Pinealon is a 3-amino acid peptide and shows neuroprotective properties.
GC81326	Tyrosine ethyl ester	34081-17-9	>98%
GC81326	Tyrosine ethyl ester exhibits antioxidant activity [1] .
GC81731	Hericene A	157207-54-0	>98.50%
GC81731	Hericene A is an orally active aromatic hericene derivative.