Home >> Signaling Pathways >> Tyrosine Kinase

Tyrosine Kinase

  1. Cat.No. Product Name Information
  2. GN10784 Rhoifolin Rhoifolin  Chemical Structure
  3. GN10737 Tanshinone IIA Tanshinone IIA  Chemical Structure
  4. GN10633 Scutellarein Scutellarein  Chemical Structure
  5. GN10603 Sennoside B Sennoside B  Chemical Structure
  6. GN10540 Fumalic acid Fumalic acid  Chemical Structure
  7. GN10527 Formononetin Formononetin  Chemical Structure
  8. GN10503 Piceatannol Piceatannol  Chemical Structure
  9. GN10497 Kaempferitrin Kaempferitrin  Chemical Structure
  10. GN10336 Daphnetin Daphnetin  Chemical Structure
  11. GN10327 Chrysophanol Chrysophanol  Chemical Structure
  12. GN10325 Nobiletin Nobiletin  Chemical Structure
  13. GN10156 Ginsenoside Rb1 Ginsenoside Rb1  Chemical Structure
  14. GC11496 TLQP 21 TLQP 21  Chemical Structure
  15. GC12656 ZM323881 A potent and selective VEGFR2 inhibitor ZM323881  Chemical Structure
  16. GC13102 XL228 A tyrosine kinase inhibitor XL228  Chemical Structure
  17. GC11876 Vandetanib hydrochloride A multi-kinase inhibitor Vandetanib hydrochloride  Chemical Structure
  18. GC10719 Toceranib A multi-targeted receptor tyrosine kinase inhibitor Toceranib  Chemical Structure
  19. GC11622 TG 100801 TG 100801  Chemical Structure
  20. GC15307 SU5416

    A tyrosine kinase inhibitor

    SU5416  Chemical Structure
  21. GC14315 SU14813 maleate A dual VEGFR and PDGFR family kinase inhibitor SU14813 maleate  Chemical Structure
  22. GC11790 SU14813 double bond Z Tyrosine kinase inhibitor SU14813 double bond Z  Chemical Structure
  23. GC14733 SU14813 A dual VEGFR and PDGFR family kinase inhibitor SU14813  Chemical Structure
  24. GC14660 SU 5402 An inhibitor of VEGFR2, FGFR1, and PDGFRβ SU 5402  Chemical Structure
  25. GC12877 SR3335 A selective inverse agonist of RORα SR3335  Chemical Structure
  26. GC16392 SR1078 A selective RORα/RORγ agonist SR1078  Chemical Structure
  27. GC11455 Silvestrol Silvestrol  Chemical Structure
  28. GC12064 SB1317 A multi-kinase inhibitor SB1317  Chemical Structure
  29. GC14534 Regorafenib monohydrate A multi-kinase inhibitor Regorafenib monohydrate  Chemical Structure
  30. GC14606 Regorafenib hydrochloride A multi-kinase inhibitor Regorafenib hydrochloride  Chemical Structure
  31. GC12857 R1530 A multi-kinase inhibitor R1530  Chemical Structure
  32. GC10499 PRT062607 Hydrochloride PRT062607 Hydrochloride  Chemical Structure
  33. GC15164 PND-1186 A potent FAK inhibitor PND-1186  Chemical Structure
  34. GC15733 PF-04217903 methanesulfonate A c-Met inhibitor PF-04217903 methanesulfonate  Chemical Structure
  35. GC16028 NVP-BGJ398 phosphate NVP-BGJ398 phosphate  Chemical Structure
  36. GC14237 Nilotinib monohydrochloride monohydrate A Bcr-Abl inhibitor Nilotinib monohydrochloride monohydrate  Chemical Structure
  37. GC13012 Motesanib Motesanib  Chemical Structure
  38. GC13140 MK-8033 MK-8033  Chemical Structure
  39. GC13424 LY2874455 A pan-FGFR inhibitor LY2874455  Chemical Structure
  40. GC11057 LY2801653 A MET kinase inhibitor LY2801653  Chemical Structure
  41. GC10809 LRRK2-IN-1 A selective LRRK2 inhibitor LRRK2-IN-1  Chemical Structure
  42. GC14931 LDN193189 Hydrochloride An inhibitor of BMP receptors ALK1, ALK2, ALK3, and ALK6 LDN193189 Hydrochloride  Chemical Structure
  43. GC17452 LDK378 dihydrochloride LDK378 dihydrochloride  Chemical Structure
  44. GC13117 Lck Inhibitor A selective inhibitor of lymphocyte-specific protein tyrosine kinase Lck Inhibitor  Chemical Structure
  45. GC10222 KX2-391 dihydrochloride A Src kinase inhibitor KX2-391 dihydrochloride  Chemical Structure
  46. GC10626 KU14R KU14R  Chemical Structure
  47. GC13264 Ki20227 A c-Fms kinase inhibitor Ki20227  Chemical Structure
  48. GC16869 Ixabepilone A broad-spectrum anticancer agent Ixabepilone  Chemical Structure
  49. GC12167 ITK inhibitor

    Potent ITK inhibitor

    ITK inhibitor  Chemical Structure
  50. GC15999 IRAK-1-4 Inhibitor I A benzimidazole IRAK-1-4 Inhibitor I  Chemical Structure
  51. GC17371 IRAK inhibitor 6 An IRAK4 inhibitor IRAK inhibitor 6  Chemical Structure
  52. GC16264 IRAK inhibitor 4 IRAK inhibitor 4  Chemical Structure
  53. GC11103 IRAK inhibitor 3 IRAK inhibitor 3  Chemical Structure
  54. GC12651 IRAK inhibitor 2 IRAK inhibitor 2  Chemical Structure
  55. GC17158 IRAK inhibitor 1 An IRAK4 inhibitor IRAK inhibitor 1  Chemical Structure
  56. GC15263 Imatinib hydrochloride V-Abl/c-Kit/PDGFR inhibitor Imatinib hydrochloride  Chemical Structure
  57. GC16244 Icotinib Hydrochloride An EGFR inhibitor Icotinib Hydrochloride  Chemical Structure
  58. GC14295 Gefitinib hydrochloride An EGFR inhibitor Gefitinib hydrochloride  Chemical Structure
  59. GC10627 Erlotinib An EGFR tyrosine kinase inhibitor Erlotinib  Chemical Structure
  60. GC10466 EMD-1214063

    EMD-1214063 (Tepotinib, MSC2156119J) is a novel potent and highly selective reversible, ATP-competitive small molecule c-Met inhibitor .

    EMD-1214063  Chemical Structure
  61. GC12149 E-3810 E-3810  Chemical Structure
  62. GC11171 DCC-2618 A dual inhibitor of c-Kit and c-MET DCC-2618  Chemical Structure
  63. GC14695 CO-1686 (AVL-301) A selective inhibitor of mutant EGFR CO-1686 (AVL-301)  Chemical Structure
  64. GC14650 CGP60474 A CDK inhibitor CGP60474  Chemical Structure
  65. GC12087 Canertinib dihydrochloride A pan-ErbB tyrosine kinase inhibitor Canertinib dihydrochloride  Chemical Structure
  66. GC11063 BMX-IN-1 A selective BMX and BTK inhibitor BMX-IN-1  Chemical Structure
  67. GC13873 BMS-690514 BMS-690514  Chemical Structure
  68. GC10606 BMS-599626 Hydrochloride BMS-599626 Hydrochloride  Chemical Structure
  69. GC10455 BMS-509744 BMS-509744  Chemical Structure
  70. GC10087 BIBX 1382 An EGFR inhibitor BIBX 1382  Chemical Structure
  71. GC12136 BAY 61-3606 dihydrochloride BAY 61-3606 dihydrochloride  Chemical Structure
  72. GC16389 BAY 61-3606 A Syk inhibitor BAY 61-3606  Chemical Structure
  73. GC17045 AXL1717 A potent and selective inhibitor of IGF-1R AXL1717  Chemical Structure
  74. GC10914 AST 487 A multi-kinase inhibitor AST 487  Chemical Structure
  75. GC14446 ASP3026 An ALK inhibitor ASP3026  Chemical Structure
  76. GC11134 ALW-II-41-27

    A multi-kinase inhibitor

    ALW-II-41-27  Chemical Structure
  77. GC17376 ALK inhibitor 2 An inhibitor of TSSK2 ALK inhibitor 2  Chemical Structure
  78. GC16228 AIM-100 An ACK1/TNK2 inhibitor AIM-100  Chemical Structure
  79. GC10707 Afatinib dimaleate An inhibitor of EGFR and ErbB2 Afatinib dimaleate  Chemical Structure
  80. GC16391 Amuvatinib (MP-470, HPK 56) A multi-targeted RTK inhibitor Amuvatinib (MP-470, HPK 56)  Chemical Structure
  81. GC18074 PF-03814735 An inhibitor of Aurora A and B kinases PF-03814735  Chemical Structure
  82. GC14592 KW 2449 A multi-kinase inhibitor KW 2449  Chemical Structure
  83. GC10638 AT9283 A broad spectrum kinase inhibitor AT9283  Chemical Structure
  84. GC15217 Danusertib (PHA-739358) A pan-Aurora kinase and Abl inhibitor Danusertib (PHA-739358)  Chemical Structure
  85. GC16519 ENMD-2076 A multi-kinase inhibitor ENMD-2076  Chemical Structure
  86. GC12145 ENMD-2076 L-(+)-Tartaric acid ENMD-2076 L-(+)-Tartaric acid  Chemical Structure
  87. GC15589 WHI-P154 A JAK3 inhibitor WHI-P154  Chemical Structure
  88. GC13848 LY2784544 Potent inhibitor of JAK2 LY2784544  Chemical Structure
  89. GC10035 TG101209 An inhibitor of JAK2, FLT3, RET, and JAK3 TG101209  Chemical Structure
  90. GC16008 CUDC-101 A multi-target inhibitor of HDACs, EGFR, and HER2 CUDC-101  Chemical Structure
  91. GC16327 Pazopanib (GW-786034) A multi-kinase inhibitor Pazopanib (GW-786034)  Chemical Structure
  92. GC14729 (R)-Crizotinib A c-MET and ALK receptor tyrosine kinase inhibitor (R)-Crizotinib  Chemical Structure
  93. GC15568 Dasatinib (BMS-354825) An inhibitor of Abl and Src Dasatinib (BMS-354825)  Chemical Structure
  94. GC10055 BGJ398 An FGFR inhibitor BGJ398  Chemical Structure
  95. GC17369 Sorafenib

    A multi-kinase inhibitor

    Sorafenib  Chemical Structure
  96. GC15983 PD 153035 hydrochloride A highly potent EGFR inhibitor PD 153035 hydrochloride  Chemical Structure
  97. GC12837 Compound 56 A potent EGFR inhibitor Compound 56  Chemical Structure
  98. GC15299 Staurosporine(CGP 41251) A potent inhibitor of protein kinase C Staurosporine(CGP 41251)  Chemical Structure
  99. GC26063 WAY-340935 WAY-340935 (VEGFR2-IN-2) can inhibit the function of VEGFR2 and the anti-proliferative activity against the H460 cell line is produced partly by interaction of VEGFR protein. WAY-340935  Chemical Structure
  100. GC26021 UNC2025 HCl UNC2025 HCl is a potent and orally bioavailable dual MER/FLT3 inhibitor with IC50 of 0.74 nM and 0.8 nM, respectively, about 20-fold selectivity over Axl and Tyro3. UNC2025 HCl  Chemical Structure
  101. GC26001 TPX-0046 TPX-0046  Chemical Structure

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