Histamine Receptor
Histamine receptor has 4 subtypes (H1,H2,H3 and H4) which mediates various biological fuctions, including allergic reaction, gastric acid secretion and inflammation etc.
Products for Histamine Receptor
- Cat.No. Product Name Information
- GC61256 Rupatadine D4 fumarate Rupatadine D4 fumarate (UR-12592 D4 fumarate) is a deuterium labeled Rupatadine fumarate.
- GC11033 Rupatadine Fumarate Inhibitor of PAF and histamine (H1) receptor
- GC31105 S 38093 S 38093 is a brain-penetrant, orally active antagonist of H3 receptor, with Kis of 8.8, 1.44 and 1.2 ?M for rat, mouse and human H3 receptors, respectively.
- GC64084 Samelisant Samelisant (SUVN-G3031) is a potent and selective histamine H3 receptor (H3R) inverse agonist with good brain penetration and oral bioavailability.
- GC68014 Seliforant
- GC31800 SUN 1334H SUN 1334H is a potent, orally active, highly selective H1 receptor antagonist, with Ki of 9.7 nM.
- GC64545 Tecastemizole Tecastemizole (Norastemizole), a major metabolite of Astemizole, is a potent and selective H1 receptor antagonist.
- GC10978 Terfenadine Histamine H1-receptor antagonist
- GC64934 Thiethylperazine Thiethylperazine, a phenothiazine derivate, is an orally active and potent dopamine D2-receptor and histamine H1-receptor antagonist.
- GC64935 Thiethylperazine dimaleate Thiethylperazine dimaleate, a phenothiazine derivate, is an orally active and potent dopamine D2-receptor and histamine H1-receptor antagonist.
- GC13496 Thioperamide histamine H3 and H4 antagonist/inverse agonist
- GC11330 Tiotidine Potent histamine H2-receptor antagonist
- GC31220 Toreforant (JNJ-38518168) Toreforant (JNJ-38518168) is a potent and selective histamine H4 receptor (H4R) antagonist, with a Ki at the human receptor of 8.4 nM.
- GC13266 trans-Triprolidine hydrochloride trans-Triprolidine hydrochloride is an orally active histamine H1 antagonist.
- GC17488 Trimipramine (maleate) potent antagonist of histamine H1 receptor
- GC12061 Tripelennamine HCl Tripelennamine HCl, an ethylenediamine derivative, is a potent histamine H1-receptor antagonist.
- GC39735 Triprolidine hydrochloride monohydrate Triprolidine hydrochloride monohydrate, a first-generation antihistamine, is an oral active histamine H1 antagonist.
- GC17585 VUF 10460 histamine H4 receptor agonist
- GC16018 VUF 5681 dihydrobromide histamine H3 receptor silent antagonist
- GC17564 VUF 8430 dihydrobromide histamine H4 receptor full agonist
- GC31824 Wy 49051 Wy 49051 is a potent, orally active H1 receptor antagonist, with IC50 of 44 nM.
- GC37959 Zaltidine Zaltidine(CP-57361) is a H2-receptor antagonist, which has the antisecretory action.
- GC13388 Zolantidine dimaleate H2 receptor antagonist