Endothelin Receptor
Endothelin receptors are members of rhodopsin-like g-protein coupled receptor (GPCRA) with 4 types (ETA, ETB1, ETB2 and ETC), which mediate various physiological processes including vasoconstriction, vasodilation, and neurotransmission etc.
Products Related to Endothelin Receptor(53)
- GC70458BMS 182874CAS: 153042-42-3Purity: >99.00%
BMS 182874 is an orallyactive, highly selective endothelin receptor (ETA receptor) antagonist, with IC50 value of 0.150 μM, Ki of 0.055 μM.
- GC72107BQ-3020 ammoniumPurity: >99.00%
BQ-3020 ammonium is a selective endothelin receptor (ETB receptor) agonist.
| Catalog No. | Product Name | CAS No. | Purity | Structure |
|---|---|---|---|---|
| GC70458 | BMS 182874 | 153042-42-3 | >99.00% | |
BMS 182874 is an orallyactive, highly selective endothelin receptor (ETA receptor) antagonist, with IC50 value of 0.150 μM, Ki of 0.055 μM. | ||||
| GC71536 | SB-209670 | 157659-79-5 | - | |
SB-209670 is an extremely potent and highly specific non-peptide, subnanomolar endothelin (ET) receptor antagonist. | ||||
| GC72107 | BQ-3020 ammonium | - | >99.00% | |
BQ-3020 ammonium is a selective endothelin receptor (ETB receptor) agonist. | ||||
| GC72942 | PD-156707 | 162412-70-6 | >99.00% | |
PD-156707 is an orally active, nonpeptide and selective Endothelin-A receptor antagonist. | ||||
| GC79668 | RES-701-3 peptide TFA | - | >98.00% | |
RES-701-3 peptide TFA is a class II lasso peptide. | ||||
