TT-012-Br (Compound 4) is a ligand for MITF and can be used for the synthesis of PROTACs, such as WZS0347 [1].
References:
[1]. Shen W, et al. Discovery of a first-in-class degrader for microphthalmia-associated transcription factor (MITF). Eur J Med Chem. 2026 Jan 15;302(Pt 3):118367.
References:
[1]. Shen W, et al. Discovery of a first-in-class degrader for microphthalmia-associated transcription factor (MITF). Eur J Med Chem. 2026 Jan 15;302(Pt 3):118367.
















