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Pain Research

Products Related to Pain Research(225)

  • GC18181 structure
    GC18181GW 405833
    CAS: 180002-83-9
    Purity: >98%

    GW 405833 (L768242) هو ناهض قوي وانتقائي لمستقبلات القنب 2 (CB2) مع EC50 يبلغ 50.7 نانومتر.

  • GC18231 structure
    GC18231Urocortin II (human) (trifluoroacetate salt)
    CAS: 398001-88-2
    Purity: >98%

    Urocortin II is a neuropeptide hormone and member of the corticotropin-releasing factor (CRF) family which includes mammalian CRF , urocortin , urocortin III , frog sauvagine, and piscine urotensin I.

  • GC18369 structure
    GC18369Cimicoxib
    CAS: 265114-23-6
    Purity: >98%

    Cimicoxib (CX) هو مثبط فعال عن طريق الفم وانتقائي COX-2 (سيكلو أوكسيجيناز -2)

  • GC18397 structure
    GC18397R-(-)-α-Methylhistamine (hydrochloride)
    CAS: 75614-89-0
    Purity: >98.00%

    R - (-) - α ؛ -Methylhistamine (هيدروكلوريد) هو ناهض قوي وانتقائي واختراق الدماغ لمستقبلات الهيستامين H3 ، مع Kd 50.3 نانومتر.

  • GC18506 structure
    GC18506N-Arachidonoyl Dopamine
    CAS: 199875-69-9
    Purity: >98.50%

    N-Arachidonoyl Dopamine هو ناهض قوي وانتقائي لمستقبلات CB1 الذاتية مع Ki من 250 نانومتر.

  • GC18582 structure
    GC185825'-hydroxy Meloxicam
    CAS: 130262-92-9
    Purity: >98%

    A metabolite of meloxicam

  • GC18650 structure
    GC18650S-(5'-Adenosyl)-L-methionine (tosylate)
    CAS: 52248-03-0
    Purity: >98.00%

    S-Adenosyl-L-methionine tosylate (S-Adenosyl methionine tosylate) is produced endogenously from methionine and ATP by action of the enzyme methionine adenosyltransferase and is an important orally active methyl group donor.

  • GC18728 structure
    GC18728CJ-13610
    CAS: 179420-17-8
    Purity: >98%

    CJ-13610 ، مثبط 5-LO من النوع nonredox ، تمنع الجرعة بشكل يعتمد على تكوين منتج 5-LO في PMNL المحفز الأيوني A23187 في غياب AA خارجي مع IC 50 بحوالي 70 نانومتر.

  • GC18783 structure
    GC1878313,14-dihydro-15-keto Prostaglandin E1
    CAS: 5094-14-4
    Purity: >98.00%

    13,14-dihydro-15-keto Prostaglandin E1 (PGE1) is a metabolite of PGE1 with much reduced biological activity.

  • GC18866 structure
    GC18866MCHB-1
    CAS: 1046140-32-2

    A CB 2 receptor agonist

  • GC18867 structure
    GC18867SER-601
    CAS: 1048038-90-9

    A selective CB 2 receptor agonist

  • GC18923 structure
    GC18923URB937
    CAS: 1357160-72-5
    Purity: >98.00%

    URB937 هو مثبط FAAH نشط عن طريق الفم ومقيد محيطيًا (IC50 = 26.8 نانومتر) ويزيد من مستويات أنانداميد

  • GC19449 structure
    GC19449ML221
    CAS: 877636-42-5
    Purity: >98%

    ML221 is a potent apelin (APJ) functional antagonist

  • GC19686 structure
    GC19686DL-Pyroglutamic acid
    CAS: 149-87-1
    Purity: >98%
  • GC19706 structure
    GC19706Propacetamol hydrochloride
    CAS: 66532-86-3
    Purity: >98%
  • GC19903 structure
    GC19903HISPOLON(P)
    CAS: 173933-40-9
    Purity: >95.00%
  • GC26144 structure
    GC26144Menthol
    CAS: 1490-04-6

    Menthol is a natural painkiller. Menthol stimulates the cold receptors by inhibiting the Ca++ current in the cell membrane of neurons, thus producing a cold feeling.

  • GC39256 structure
    GC39256LP-935509
    CAS: 1454555-29-3
    Purity: >99.50%

    LP-935509 هو مثبط فعال عن طريق الفم وانتقائي ومنافس للأدينوزين ثلاثي الفوسفات (ATP) وذو قدرة اختراق للدماغ، لبروتين المحول المهاجر 2 المرتبط بالأدابتور كيناز 1 (AAK1) بـ IC50 يبلغ 3.3 نانومتر و Ki يبلغ 0.9 نانومتر على التوالي.

  • GC39344 structure
    GC39344BAY-1797
    CAS: 2055602-83-8
    Purity: >98.50%

    BAY-1797 هو مضاد P2X4 فعال وفعال عن طريق الفم وانتقائي ، مع IC50 من 211 نانومتر ضد الإنسان P2X4

  • GC40184 structure
    GC40184Probenecid-d14
    CAS: 1189657-87-1
    Purity: >99.00%

    Probenecid-d14 is intended for use as an internal standard for the quantification of probenecid by GC- or LC-MS.

  • GC40594 structure
    GC40594(R)-AM1241
    CAS: 444912-51-0
    Purity: >98.00%

    (R)-AM1241 binds to cannabinoid (CB) receptors and has greater than 100-fold selectivity for the CB2 over the CB1 receptor (Kis = 15 and 5,000 nM, respectively, in a membrane assay using human receptors).

  • GC40595 structure
    GC40595(S)-AM1241
    CAS: 444912-53-2
    Purity: >98.00%

    (S)-AM1241 binds to cannabinoid (CB) receptors and is selective for the CB2 over the CB1 receptor (Kis = 658 and >10,000 nM, respectively, in a membrane assay using human receptors).

  • GC40759 structure
    GC407598-methyl Nonanoic Acid
    CAS: 5963-14-4
    Purity: >98.00%

    8-methyl Nonanoic Acid is the precursor of 8-methyl-nonenoic acid and is involved in the synthesis of capsaicin.

  • GC41151 structure
    GC41151Decursinol angelate
    CAS: 130848-06-5
    Purity: >98.00%

    Decursinol angelate is a pyranocoumarin that has been found in the Korean medicinal herb A.