GLPBio

Free Fatty Acid Receptors

FFAR1 (GPR40) is a G protein-coupled receptor for medium and long chain saturated and unsaturated fatty acids. It plays a role in glucose homeostasis, insulin secretion and bone homeostasis etc.

Products Related to Free Fatty Acid Receptors(16)

  • GC10373 structure
    GC10373MEDICA 16
    CAS: 87272-20-6
    Purity: >98%

    Free fatty acid 1 (FFA1/GPR40) receptor agonist

  • GC10922 structure
    GC10922TUG 424
    CAS: 1082058-99-8
    Purity: >98.00%

    FFA1 (GPR40) agonist

  • GC11467 structure
    GC11467AS 2034178
    CAS: 1030846-42-4
    Purity: >98%

    AS 2034178, a specific and orally active GPR40 agonist, exhibits glucose-dependent insulin secretion enhancement.

  • GC16176 structure
    GC16176GSK 137647
    CAS: 349085-82-1
    Purity: >98.00%

    GSK 137647 (GSK 137647) is a potent, selective free fatty acid receptor 4 (FFA4) agonist with pEC50 values of 6.3, 6.2, and 6.1 for human, mouse and rat FFA4, and pEC50 values < 4.5 for all three species for FFA1, FFA2, and FFA3, respectively.

  • GC17149 structure
    GC171494-CMTB
    CAS: 300851-67-6
    Purity: >99.00%

    4-CMTB is a selective free fatty acid receptor 2 (FFA2/GPR43) agonist and a positive allosteric modulator.

  • GC17753 structure
    GC17753AH 7614
    CAS: 6326-06-3
    Purity: >99.50%

    AH 7614 is a selective free fatty acid receptor 4 (FFA4/GPR120) antagonist. AH 7614 exhibits pIC 50 values of 7.1, 8.1, and 8.1 for human, mouse, and rat FFA4, respectively.

  • GC11434 structure
    GC11434GSK1292263
    CAS: 1032823-75-8
    Purity: >99.00%

    Novel GPR119 agonist

  • GC12401 structure
    GC12401GW9508
    CAS: 885101-89-3
    Purity: >98.00%

    FFA1/GPR40 agonist,potent and selective

  • GC14027 structure
    GC14027GW-1100
    CAS: 306974-70-9
    Purity: >98%

    A selective GPR40 antagonist

  • GC16054 structure
    GC16054TUG-770
    CAS: 1402601-82-4
    Purity: >99.50%

    An agonist of FFA1/GPR40

  • GC16555 structure
    GC16555TAK-875
    CAS: 1000413-72-8
    Purity: >98.50%

    TAK-875 is a potent, selective and orally bioavailable GPR40 (G protein-coupled receptor 40) agonist with an EC 50 value of 0.014μM for human GPR40.

  • GC50293 structure
    GC50293CATPB
    CAS: 1322598-09-3
    Purity: >98.00%

    FFA2 (GPR43) inverse agonist

  • GC50313 structure
    GC50313ZQ 16
    CAS: 376616-73-8
    Purity: >98%

    Selective GPR84 agonist

  • GC50333 structure
    GC50333AMG 837 hemicalcium salt
    CAS: 1291087-14-3
    Purity: >98%

    AMG 837 hemicalcium salt is a potent, orally bioavailable and partial agonist of GPR40/FFA1.

  • GC50578 structure
    GC50578AZ 1729
    CAS: 2016864-46-1
    Purity: >98%

    FFA2 allosteric agonist; displays bias for the Gi signaling pathway

  • GC50662 structure
    GC50662DL 175
    CAS: 2487253-25-6
    Purity: >98.00%