(+)-BAY-1251152 is a CDK9 inhibitor extracted from patent WO 2014076091 A1, example 1. CDK9
[1]. Ulrich LÜCKING, et al. 5-fluoro-n-(pyridin-2-yl)pyridin-2-amine derivatives containing a sulfoximine group. WO 2014076091 A1.
(+)-BAY-1251152
Catalog No.: GC34953Purity:>99.50%Synonyms: (+)-BAY-1251152; (+)-VIP152
(+)-BAY-1251152 ((+)-BAY-1251152) is an enanthiomer of BAY-1251152 with rotation (+). (+)-BAY-1251152 is a potent and selective CDK9 inhibitor with an IC50 of 3 nM. (+)-BAY-1251152 has anti-tumour activity.
Products are for research use only. Not for human use. We do not sell to patients.
Cas No.: 1610358-56-9
10mM (in 1mL DMSO)In Stock
$183.00
1
2mgIn Stock
$89.00
1
5mgIn Stock
$168.00
1
10mgIn Stock
$268.00
1
25mgIn Stock
$495.00
1
| Pack Size | Price | Availability | Quantity | Action |
|---|---|---|---|---|
| 10mM (in 1mL DMSO) | $183.00 | In Stock | 1 | |
| 2mg | $89.00 | In Stock | 1 | |
| 5mg | $168.00 | In Stock | 1 | |
| 10mg | $268.00 | In Stock | 1 | |
| 25mg | $495.00 | In Stock | 1 |
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Citations
No citations are currently available for this product. Below are selected publications citing GlpBio products.
Nature641, 529–536 (2025)
Nature628, 630–638 (2024)
Nature632, 686–694 (2024)
Nature618, 1017–1023 (2023)
Nature610, 366–372 (2022)
Cell187(9):2288-2304 (2024)
Cell183(7):1867-1883 (2020)
Science388(6745) (2025)
Science387(6739) (2025)
Science387(6734) (2025)
Cell Research35, 97–116 (2025)
Cell Research34, 683–706 (2024)
Cell Research33, 273–287 (2023)
Cell Research33, 546–561 (2023)
Cell Research33, 904–922 (2023)
Cell Research31, 1291–1307 (2021)
Description
Product Documents
Purity:>99.50%Appearance:A solid
Chemical Properties
CAS No.
1610358-56-9
Synonyms
(+)-BAY-1251152; (+)-VIP152
SMILES
N=S(CC1=CC(NC2=NC=C(F)C(C3=CC=C(F)C=C3OC)=C2)=NC=C1)(C)=O.[Rotation(+)]
Molecular Formula
C19H18F2N4O2S
Molecular Weight
404.43
Solubility
DMSO: 113.3 mg/mL (280.15 mM and warming)
Storage
Store at -20°C
General tips
Select a suitable solvent according to the product solubility data. Once prepared, aliquot the stock solution to avoid repeated freeze-thaw cycles.
Use stock solutions within 6 months when stored at -80°C or within 1 month when stored at -20°C.
To improve solubility, warm the tube to 37°C and sonicate it for an appropriate period.
Use stock solutions within 6 months when stored at -80°C or within 1 month when stored at -20°C.
To improve solubility, warm the tube to 37°C and sonicate it for an appropriate period.
Shipping Condition
Evaluation samples are shipped with blue ice. Other available sizes are shipped at room temperature or with blue ice upon request.
CalculatorsMolarity / Dilution / Molecular Weight / Unit Conversion / In Vivo Formulation / Solubility
g/mol
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