GLPBio

Histamine Receptor

Histamine receptor has 4 subtypes (H1,H2,H3 and H4) which mediates various biological fuctions, including allergic reaction, gastric acid secretion and inflammation etc.

Products Related to Histamine Receptor(243)

  • GC13537 structure
    GC13537A 331440 dihydrochloride
    CAS: 1049740-32-0
    Purity: >98%

    H3 receptor antagonist,non-imidazole,high affinity

  • GC13757 structure
    GC13757CarbinoxaMine Maleate
    CAS: 3505-38-2
    Purity: >99.00%

    CarbinoxaMine Maleate는 히스타민 H1 수용체 길항제입니다.

  • GC13899 structure
    GC13899Antazoline HCl
    CAS: 2508-72-7
    Purity: >99.00%

    Antazoline HCl은 1세대 항히스타민제로 항콜린성 특성을 가지고 있어 비강 충혈 및 점안액을 완화하는 데 사용됩니다.

  • GC13995 structure
    GC13995Carcinine ditrifluoroacetate
    CAS: 56897-53-1
    Purity: >98%

    H3 receptor antagonist

  • GC14051 structure
    GC14051Doxylamine Succinate
    CAS: 562-10-7
    Purity: >99.50%

    1세대 항히스타민제인 독실아민(숙시네이트)은 히스타민(H1) 수용체 길항제입니다.

  • GC14260 structure
    GC14260Immethridine dihydrobromide
    CAS: 699020-93-4
    Purity: >98%

    histamine H3 receptor agonist

  • GC14429 structure
    GC14429JNJ 10191584 maleate
    CAS: 869497-75-6
    Purity: >98%

    histamine H4 receptor silent antagonist

  • GC14742 structure
    GC14742DPPE fumarate
    CAS: 1185241-83-1
    Purity: >99.50%

    H1C 수용체 길항제인 DPPE 푸마레이트(DPPE 푸마레이트)는 광범위한 세포독성 물질을 강화하고 심지어 정상 세포를 어느 정도 보호합니다.

  • GC14984 structure
    GC14984Diphenylpyraline HCl
    CAS: 132-18-3
    Purity: >99.00%

    디페닐피랄린 HCl은 강력한 히스타민 H1수용체 길항제입니다.

  • GC15713 structure
    GC15713Ebastine
    CAS: 90729-43-4
    Purity: >98.00%

    Ebastine(LAS-W 090)은 경구 활성 2세대 히스타민 H1 수용체 길항제입니다.

  • GC15723 structure
    GC15723Dimebolin
    CAS: 3613-73-8
    Purity: >98%

    antihistamine, orally-available

  • GC15957 structure
    GC15957Proxyfan oxalate
    CAS: 177708-09-7
    Purity: >98%

    histamine H3 receptor ligand

  • GC16018 structure
    GC16018VUF 5681 dihydrobromide
    CAS: 639089-06-8
    Purity: >98%

    histamine H3 receptor silent antagonist

  • GC16052 structure
    GC16052Aminopotentidine
    CAS: 140873-26-3
    Purity: >98%

    H2 antagonist

  • GC16089 structure
    GC16089Ebrotidine
    CAS: 100981-43-9
    Purity: >99.00%
  • GC16162 structure
    GC16162ICI 162,846
    CAS: 84545-30-2
    Purity: >98%

    histamine H2 receptor antagonist

  • GC16180 structure
    GC16180GT 2016
    CAS: 152241-24-2
    Purity: >98%

    GT 2016은 Ki가 43.8nM인 강력하고 선택적인 뇌 침투 히스타민 H3 수용체 길항제입니다.

  • GC16487 structure
    GC16487Nα-Methylhistamine dihydrochloride
    CAS: 16503-22-3
    Purity: >98%

    histamine H3 receptor agonist

  • GC16787 structure
    GC16787Pheniramine Maleate
    CAS: 132-20-7
    Purity: >99.50%

    Histamine receptor antagonist

  • GC16945 structure
    GC16945Astemizole
    CAS: 68844-77-9
    Purity: >99.50%

    Astemizole은 IC50 값이 4nM인 강력한 항히스타민 화합물로 히스타민 H1-수용체를 길항한다.

  • GC17000 structure
    GC17000Nedocromil
    CAS: 69049-73-6
    Purity: >98.50%

    Nedocromil은 히스타민, 류코트리엔 C4(LTC4) 및 프로스타글란딘 D2(PGD2)를 포함한 여러 매개체의 작용 또는 형성을 억제합니다.

  • GC17010 structure
    GC17010Methimepip dihydrobromide
    CAS: 817636-54-7
    Purity: >98%

    histamine H3 receptor agonist

  • GC17429 structure
    GC17429HTMT dimaleate
    CAS: 195867-54-0
    Purity: >98%

    HTMT(디말레에이트)는 강력한 히스타민 H1 및 H2 수용체 작용제입니다.

  • GC17488 structure
    GC17488Trimipramine (maleate)
    CAS: 521-78-8
    Purity: >98.00%

    트리미프라민(말레에이트)은 5-HT 수용체 길항제이며, 5-HT1C, 5-HT2 및 5-HT1A에 대해 각각 pKi 결합 값이 6.39, 8.10, 4.66입니다.