NMDA Receptor
NMDA (N-methyl-D-aspartate) receptor is a glutamate-gated cation channels that plays a vital role in regulating synaptic transmission, neuroplasticity and central nervous system development. It is involved in a range of physiological processes such as learning, memory and pain etc.
Products Related to NMDA Receptor(77)
- GC17206DL-AP5CAS: 76326-31-3Purity: >98.00%
DL-AP5 is an racemic form of a selective NMDA (N-methyl-D-aspartate) receptor antagonist. D-AP5 is the active (-) stereoisomer, which can competitively inhibit the glutamate binding site of the NMDA receptor (K d = 1.4μM), while the (+) isomer (L-AP5) shows relatively low NMDA receptor antagonist activity.
- GC17481GavestinelCAS: 153436-38-5Purity: >98%
Gavestinel (GV 150526) is a potent, selective, orally active and non-competitive antagonist of NMDA receptor.
- GC17823L-Cysteinesulfinic acidCAS: 1115-65-7Purity: >98.00%
L-Cysteinesulfinic acid is an endogenous sulfur-containing excitatory amino acid, and an intermediate in the metabolic conversion of cysteine to taurine. L-Cysteinesulfinic acid acts as an agonist of NMDA receptors and mGlu receptors, and is applied in research on glutamatergic neurotransmission, taurine biosynthesis and central cardiovascular regulation.
| Catalog No. | Product Name | CAS No. | Purity | Structure |
|---|---|---|---|---|
| GC17206 | DL-AP5 | 76326-31-3 | >98.00% | |
DL-AP5 is an racemic form of a selective NMDA (N-methyl-D-aspartate) receptor antagonist. D-AP5 is the active (-) stereoisomer, which can competitively inhibit the glutamate binding site of the NMDA receptor (K d = 1.4μM), while the (+) isomer (L-AP5) shows relatively low NMDA receptor antagonist activity. | ||||
| GC17481 | Gavestinel | 153436-38-5 | >98% | |
Gavestinel (GV 150526) is a potent, selective, orally active and non-competitive antagonist of NMDA receptor. | ||||
| GC17652 | N-(4-Hydroxyphenylacetyl)spermine | 130210-32-1 | >98% | |
NMDA receptor antagonist | ||||
| GC17823 | L-Cysteinesulfinic acid | 1115-65-7 | >98.00% | |
L-Cysteinesulfinic acid is an endogenous sulfur-containing excitatory amino acid, and an intermediate in the metabolic conversion of cysteine to taurine. L-Cysteinesulfinic acid acts as an agonist of NMDA receptors and mGlu receptors, and is applied in research on glutamatergic neurotransmission, taurine biosynthesis and central cardiovascular regulation. | ||||
| GC18118 | SDZ 220-581 | 174575-17-8 | >99.00% | |
