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NMDA Receptor

NMDA (N-methyl-D-aspartate) receptor is a glutamate-gated cation channels that plays a vital role in regulating synaptic transmission, neuroplasticity and central nervous system development. It is involved in a range of physiological processes such as learning, memory and pain etc.

Products for  NMDA Receptor

  1. Cat.No. Product Name Information
  2. GC10237 (±)-1-(1,2-Diphenylethyl)piperidine maleate NMDA receptor antagonist (±)-1-(1,2-Diphenylethyl)piperidine maleate  Chemical Structure
  3. GC16616 (+)-MK 801 (+)-MK 801  Chemical Structure
  4. GC11025 (+)-MK 801 Maleate (+)-MK 801 Maleate (MK-801 maleate) is a potent, selective and non-competitive NMDA receptor antagonist with Kd of 37.2 nM in rat brain membranes. (+)-MK 801 Maleate  Chemical Structure
  5. GC15270 (-)-MK 801 (-)-MK 801 ((-)-MK-801 maleate) is a less active (-)-enantiomer of Dizocilpine. (-)-MK 801  Chemical Structure
  6. GC16915 (2R,3S)-Chlorpheg NMDA receptor antagonist (2R,3S)-Chlorpheg  Chemical Structure
  7. GC14085 (R)-(+)-HA-966 NMDA receptor antagonist/partial agonist (R)-(+)-HA-966  Chemical Structure
  8. GC10168 (R)-4-Carboxyphenylglycine NMDA receptor antagonist (R)-4-Carboxyphenylglycine  Chemical Structure
  9. GC14236 (R)-CPP NMDA antagonist (R)-CPP  Chemical Structure
  10. GC12488 (RS)-(Tetrazol-5-yl)glycine NMDA receptor agonist (RS)-(Tetrazol-5-yl)glycine  Chemical Structure
  11. GC10476 (RS)-CPP NMDA antagonist (RS)-CPP  Chemical Structure
  12. GC10370 (S)-(-)-HA-966 NMDA receptor antagonist (S)-(-)-HA-966  Chemical Structure
  13. GC16799 5,7-Dichlorokynurenic acid NMDA receptor antagonist 5,7-Dichlorokynurenic acid  Chemical Structure
  14. GC14598 5,7-Dichlorokynurenic acid sodium salt NMDA receptor antagonist 5,7-Dichlorokynurenic acid sodium salt  Chemical Structure
  15. GC11286 ACBC ACBC is a NMDA receptor partial agonist acting at the glycine site, NR1. ACBC  Chemical Structure
  16. GC14470 Arcaine sulfate NMDA antagonist Arcaine sulfate  Chemical Structure
  17. GC12137 CCMQ inhibits [3H]-homoquinolinic acid binding to non-NMDA sensitive sites CCMQ  Chemical Structure
  18. GC10122 CGP 37849 NMDA receptor antagonist CGP 37849  Chemical Structure
  19. GC11027 CGP 39551 NMDA antagonist CGP 39551  Chemical Structure
  20. GC15752 CGP 78608 hydrochloride NMDA antagonist CGP 78608 hydrochloride  Chemical Structure
  21. GC16272 CGS 19755 NMDA receptor antagonist CGS 19755  Chemical Structure
  22. GC14414 CIQ NMDA receptor potentiator CIQ  Chemical Structure
  23. GC11942 cis-ACPD NMDA receptor agonist and group II mGluR agonist cis-ACPD  Chemical Structure
  24. GC10792 Co 101244 hydrochloride NR2B-containing NMDA receptor antagonist Co 101244 hydrochloride  Chemical Structure
  25. GC13714 Conantokin G NR2B-selective NMDA receptor antagonist Conantokin G  Chemical Structure
  26. GC12944 Conantokin-R non-competitive NMDA receptor antagonist Conantokin-R  Chemical Structure
  27. GC15156 Conantokin-T Non-competitive NMDA receptor antagonist Conantokin-T  Chemical Structure
  28. GC16315 D-AP5

    A NMDA antagonist

    D-AP5  Chemical Structure
  29. GC15112 D-AP7 NMDA receptor antagonist D-AP7  Chemical Structure
  30. GC10043 D-CPP-ene NMDA antagonist D-CPP-ene  Chemical Structure
  31. GC17206 DL-AP5 A NMDA antagonist DL-AP5  Chemical Structure
  32. GC14897 DL-AP5 Sodium salt NMDA receptor antagonist DL-AP5 Sodium salt  Chemical Structure
  33. GC11335 DL-AP7 first generation phosphono NMDA antagonist DL-AP7  Chemical Structure
  34. GC10085 DQP 1105

    NMDA receptor antagonist

    DQP 1105  Chemical Structure
  35. GC15343 Eliprodil NMDA receptor antagonist Eliprodil  Chemical Structure
  36. GC10522 Felbamate antagonist at the NMDA-associated glycine binding site Felbamate  Chemical Structure
  37. GC15363 Felbamate hydrate N-methyl-D-aspartate (NMDA) inhibitor Felbamate hydrate  Chemical Structure
  38. GC11470 Flupirtine maleate NMDA receptor antagonist Flupirtine maleate  Chemical Structure
  39. GC17481 Gavestinel Gavestinel (GV 150526) is a potent, selective, orally active and non-competitive antagonist of NMDA receptor. Gavestinel  Chemical Structure
  40. GC14121 GLYX 13 GLYX 13 (GLYX-13) is an N-methyl-D-aspartate receptor (NMDAR) modulator that has characteristics of a glycine site partial agonist. GLYX 13  Chemical Structure
  41. GC10114 Homoquinolinic acid NMDA receptor agonist Homoquinolinic acid  Chemical Structure
  42. GC13074 HU 211 NMDA antagonist, novel and non-competitive HU 211  Chemical Structure
  43. GC11715 Ibotenic acid NMDA and metabotropic glutamate receptor agonist Ibotenic acid  Chemical Structure
  44. GC10471 Ifenprodil hemitartrate Ifenprodil hemitartrate is a typical noncompetitive NMDA receptor antagonist. Ifenprodil hemitartrate  Chemical Structure
  45. GC10696 L-689,560 potent NMDA antagonist L-689,560  Chemical Structure
  46. GC11706 L-701,252 glycine-NMDA site antagonist L-701,252  Chemical Structure
  47. GC14810 L-701,324 NMDA receptor antagonist L-701,324  Chemical Structure
  48. GC12154 L-AP5 NMDA antagonist L-AP5  Chemical Structure
  49. GC17823 L-Cysteinesulfinic acid NMDA and mGlu receptor agonist L-Cysteinesulfinic acid  Chemical Structure
  50. GC11124 Lanicemine

    voltage-dependent NMDA channel blocker

    Lanicemine  Chemical Structure
  51. GC11862 LY 233053 Competitive NMDA receptor antagonist LY 233053  Chemical Structure
  52. GC12873 LY 235959 NMDA receptor antagonist LY 235959  Chemical Structure
  53. GC14039 MDL-29951 Glycine antagonist of NMDA receptor activation MDL-29951  Chemical Structure
  54. GC10688 MNI-caged-D-aspartate Agonist at NMDA receptors and EAAT substrate MNI-caged-D-aspartate  Chemical Structure
  55. GC16240 MNI-caged-NMDA NMDA caged with the photosensitive 4-methoxy-7-nitroindolinyl group MNI-caged-NMDA  Chemical Structure
  56. GC17652 N-(4-Hydroxyphenylacetyl)spermine NMDA receptor antagonist N-(4-Hydroxyphenylacetyl)spermine  Chemical Structure
  57. GC11281 N20C hydrochloride NMDA receptor antagonist N20C hydrochloride  Chemical Structure
  58. GC10574 Norketamine hydrochloride

    Major metabolite of ketamine, NMDA receptor antagonist

    Norketamine hydrochloride  Chemical Structure
  59. GC14357 PMPA (NMDA antagonist) Competitive NMDA receptor antagonist PMPA (NMDA antagonist)  Chemical Structure
  60. GC10247 PPDA Subtype-selective NMDA receptor antagonist PPDA  Chemical Structure
  61. GC11879 PPPA NMDA receptor antagonist PPPA  Chemical Structure
  62. GC16776 QNZ 46 NR2C/NR2D-selective NMDA receptor antagonist QNZ 46  Chemical Structure
  63. GC14547 Quinolinic acid NMDA agonist Quinolinic acid  Chemical Structure
  64. GC16131 Remacemide hydrochloride NMDA receptor antagonist Remacemide hydrochloride  Chemical Structure
  65. GC14782 Ro 04-5595 hydrochloride NR2B-containing NMDA receptors antagonist Ro 04-5595 hydrochloride  Chemical Structure
  66. GC14381 Ro 8-4304 hydrochloride NMDA receptor antagonist Ro 8-4304 hydrochloride  Chemical Structure
  67. GC12816 SDZ 220-040

    NMDA receptor antagonist

    SDZ 220-040  Chemical Structure
  68. GC18118 SDZ 220-581 SDZ 220-581  Chemical Structure
  69. GC16986 SDZ 220-581 hydrochloride NMDA receptor antagonist SDZ 220-581 hydrochloride  Chemical Structure
  70. GC10866 Spermidine trihydrochloride Spermidine trihydrochloride maintains cell membrane stability, increases antioxidant enzymes activities, improving photosystem II (PSII), and relevant gene expression. Spermidine trihydrochloride  Chemical Structure
  71. GC11064 Spermine tetrahydrochloride NMDA receptor modulator Spermine tetrahydrochloride  Chemical Structure
  72. GC15732 Synthalin sulfate NMDA receptor antagonist Synthalin sulfate  Chemical Structure
  73. GC15065 TCN 201 NR1/NR2A selective NMDA receptor antagonist TCN 201  Chemical Structure
  74. GC14770 TCN 213 NR1/NR2A selective NMDA receptor antagonist TCN 213  Chemical Structure
  75. GC11585 TCN 237 dihydrochloride TCN 237 dihydrochloride is a potent and NR2B-selective NMDA antagonist with Ki of 0.85 nM; NR2B Ca2+ influx IC50 is 9.7 nM; no activities on NR2A, NR2C, NR2D, hERG-channel and α1-adrenergic receptor. TCN 237 dihydrochloride  Chemical Structure
  76. GC14442 TCS 46b NR1A/NR2B NMDA receptor antagonist,orally active TCS 46b  Chemical Structure
  77. GC10595 threo Ifenprodil hemitartrate σ receptor agonist and NR2B subunit-selective NMDA receptor antagonist threo Ifenprodil hemitartrate  Chemical Structure
  78. GC12785 ZD 9379 NMDA receptor antagonist ZD 9379  Chemical Structure

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