Dopamine Receptor
Dopamine receptors (DR) are members of G protein-coupled receptors superfamily. There are 5 subtypes (D1, D2, D3, D4, D5) of DR which mediate the functions of dopamine in central nervous system for control of locomotion, cognition, and emotion etc.
Products Related to Dopamine Receptor(300)
- GC79286(+)-RazpipadonCAS: 1643489-51-3Purity: >98.00%
(+)-Razpipadon ((+)-PW0464) is a selective D1 dopamine receptor agonist belonging to non-catechol compounds.
- GC79287TAT-D1 peptide acetatePurity: >98.00%
TAT-D1 peptide acetate is a dopamine D1-D2 receptor heterodimer inhibitor.
- GC79288MazapertineCAS: 134208-17-6Purity: >99.00%
Mazapertine is an orally active antipsychotic agent.
- GC79779N-Desmethyl xanomelineCAS: 131986-96-4Purity: >98%
N-Desmethyl xanomeline is a pharmacologically active metabolite of Xanomeline.
- GC80835Didesmethyl cariprazine-d 8CAS: 1308279-08-4Purity: >99.00%
Didesmethyl cariprazine -d 8 is the deuterium labeled Didesmethyl cariprazine.
- GC80837Desmethyl cariprazine-d 8CAS: 1308278-85-4Purity: >99.50%
Desmethyl cariprazine -d 8 is the deuterium labeled Desmethyl cariprazine.
- GC81895RB 101 hydrochloridePurity: >98.00%
RB 101 hydrochloride is a blood-brain barrier-crossing prodrug as well as aminopeptidase N and neutral endopeptidase-24.11 inhibitor.
- GN10607NuciferineCAS: 475-83-2Purity: >98.00%
Nuciferine, un principal composant bioactif issu de la feuille de lotus, est un antagoniste des récepteurs 5-HT 2A , 5-HT 2C et 5-HT 2B avec des valeur d' IC 50 respectives de 0.478μM, 0.131μM et 1μM.
- GC10441CabergolineCAS: 81409-90-7Purity: >98.00%
La cabergoline est un agoniste des récepteurs de type dopamine D2 dérivé de l'ergot qui a une forte affinité pour les récepteurs D2, D3 et 5-HT2B (Ki = 0,7, 1,5 et 1,2, respectivement).
| Catalog No. | Product Name | CAS No. | Purity | Structure |
|---|---|---|---|---|
| GC79286 | (+)-Razpipadon | 1643489-51-3 | >98.00% | |
(+)-Razpipadon ((+)-PW0464) is a selective D1 dopamine receptor agonist belonging to non-catechol compounds. | ||||
| GC79287 | TAT-D1 peptide acetate | - | >98.00% | |
TAT-D1 peptide acetate is a dopamine D1-D2 receptor heterodimer inhibitor. | ||||
| GC79288 | Mazapertine | 134208-17-6 | >99.00% | |
Mazapertine is an orally active antipsychotic agent. | ||||
| GC79779 | N-Desmethyl xanomeline | 131986-96-4 | >98% | |
N-Desmethyl xanomeline is a pharmacologically active metabolite of Xanomeline. | ||||
| GC80835 | Didesmethyl cariprazine-d 8 | 1308279-08-4 | >99.00% | |
Didesmethyl cariprazine -d 8 is the deuterium labeled Didesmethyl cariprazine. | ||||
| GC80837 | Desmethyl cariprazine-d 8 | 1308278-85-4 | >99.50% | |
Desmethyl cariprazine -d 8 is the deuterium labeled Desmethyl cariprazine. | ||||
| GC81895 | RB 101 hydrochloride | - | >98.00% | |
RB 101 hydrochloride is a blood-brain barrier-crossing prodrug as well as aminopeptidase N and neutral endopeptidase-24.11 inhibitor. | ||||
| GN10513 | Tetrahydroberberine,THB | 522-97-4 | >98.00% | |
| GN10607 | Nuciferine | 475-83-2 | >98.00% | |
Nuciferine, un principal composant bioactif issu de la feuille de lotus, est un antagoniste des récepteurs 5-HT 2A , 5-HT 2C et 5-HT 2B avec des valeur d' IC 50 respectives de 0.478μM, 0.131μM et 1μM. | ||||
| GN10740 | Tetrahydropalmatine | 10097-84-4 | >99.00% | |
| GC10441 | Cabergoline | 81409-90-7 | >98.00% | |
La cabergoline est un agoniste des récepteurs de type dopamine D2 dérivé de l'ergot qui a une forte affinité pour les récepteurs D2, D3 et 5-HT2B (Ki = 0,7, 1,5 et 1,2, respectivement). | ||||
| GC14657 | Rotundine | 483-14-7 | >99.50% | |
La rotundine est un antagoniste des récepteurs dopaminergiques D1, D2 et D3 avec des CI50 de 166 nM, 1,4 μM et 3,3 μM, respectivement. | ||||
