Histamine Receptor
Histamine receptor has 4 subtypes (H1,H2,H3 and H4) which mediates various biological fuctions, including allergic reaction, gastric acid secretion and inflammation etc.
Products Related to Histamine Receptor(243)
- GC10127Betahistine 2HClCAS: 5579-84-0Purity: >99.50%
Betahistine 2HCl is an orally active histamine H1 receptor agonist and a H3 receptor antagonist.
- GC10306Hydroxyzine 2HClCAS: 2192-20-3Purity: >99.50%
Hydroxyzine 2HCl, a benzodiazepine antihistamine agent, acts as a orally active histamineH1-receptor and serotonin antagonist.
- GC10369Roxatidine Acetate HClCAS: 93793-83-0Purity: >98.00%
Roxatidine Acetate HCl is a potent, selective, competitive and orally active histamine H2-receptor antagonist.
- GC10400JNJ-7777120CAS: 459168-41-3Purity: >98.00%
JNJ-7777120 is a histamine H 4 receptor (H 4 R: K i = 4.5nM) antagonist.
- GC10511Olopatadine HClCAS: 140462-76-6Purity: >99.50%
Olopatadine HCl (ALO4943A) is a histamine blocker used to treat allergic conjunctivitis.
- GC10966Fexofenadine HClCAS: 153439-40-8Purity: >99.50%
Fexofenadine HCl is an orally active and nonsedative histamine H1 receptor antagonist.
- GC11009Cetirizine DiHClCAS: 83881-52-1Purity: >99.00%
Cetirizine DiHCl, a second-generation antihistamine and the carboxylated metabolite of hydroxyzine, is a specific, orally active and long-acting histamine H1-receptor antagonist.
- GC11033Rupatadine FumarateCAS: 182349-12-8Purity: >99.50%
Inhibitor of PAF and histamine (H1) receptor
- GC12061Tripelennamine HClCAS: 154-69-8Purity: >99.50%
Tripelennamine HCl, an ethylenediamine derivative, is a potent histamine H1-receptor antagonist.
- GC12365Ranitidine hydrochlorideCAS: 66357-59-3Purity: >98.00%
Ranitidine hydrochloride, an inhibitor of gastric acid secretion, competitively antagonizes histamine-induced increases in contraction frequency with a pA2 value of 7.2.
- GC13341Brompheniramine hydrogen maleateCAS: 980-71-2Purity: >99.50%
Brompheniramine ((±)-Brompheniramine) maleate is a potent and orally active antihistamine of the alkylamine class.
- GC14250Bepotastine BesilateCAS: 190786-44-8Purity: >99.50%
Non-sedating, selective antagonist of histamine 1 (H1) receptor
- GC14726Mianserin HClCAS: 21535-47-7Purity: >99.50%
Mianserin HCl (Org GB 94) is a H1 receptor inverse agonist and is a psychoactive agent of the tetracyclic antidepressant.
- GC14892Clemastine FumarateCAS: 14976-57-9Purity: >99.50%
Clemastine Fumarate, the over-the-counter antihistamine and muscarinic receptor blocker, has remyelinating potential in Multiple sclerosis (MS).
- GC15068Buclizine HClCAS: 129-74-8Purity: >98.00%
Buclizine HCl is an orally active antihistamine antiallergic compound.
| Catalog No. | Product Name | CAS No. | Purity | Structure |
|---|---|---|---|---|
| GC10127 | Betahistine 2HCl | 5579-84-0 | >99.50% | |
Betahistine 2HCl is an orally active histamine H1 receptor agonist and a H3 receptor antagonist. | ||||
| GC10306 | Hydroxyzine 2HCl | 2192-20-3 | >99.50% | |
Hydroxyzine 2HCl, a benzodiazepine antihistamine agent, acts as a orally active histamineH1-receptor and serotonin antagonist. | ||||
| GC10369 | Roxatidine Acetate HCl | 93793-83-0 | >98.00% | |
Roxatidine Acetate HCl is a potent, selective, competitive and orally active histamine H2-receptor antagonist. | ||||
| GC10400 | JNJ-7777120 | 459168-41-3 | >98.00% | |
JNJ-7777120 is a histamine H 4 receptor (H 4 R: K i = 4.5nM) antagonist. | ||||
| GC10478 | Mizolastine dihydrochloride | 1056596-82-7 | >98% | |
Histamine H1-receptor antagonist | ||||
| GC10511 | Olopatadine HCl | 140462-76-6 | >99.50% | |
Olopatadine HCl (ALO4943A) is a histamine blocker used to treat allergic conjunctivitis. | ||||
| GC10806 | Histamine 2HCl | 56-92-8 | >98.00% | |
Histamine 2HCl is an endogenous metabolite. | ||||
| GC10966 | Fexofenadine HCl | 153439-40-8 | >99.50% | |
Fexofenadine HCl is an orally active and nonsedative histamine H1 receptor antagonist. | ||||
| GC11009 | Cetirizine DiHCl | 83881-52-1 | >99.00% | |
Cetirizine DiHCl, a second-generation antihistamine and the carboxylated metabolite of hydroxyzine, is a specific, orally active and long-acting histamine H1-receptor antagonist. | ||||
| GC11033 | Rupatadine Fumarate | 182349-12-8 | >99.50% | |
Inhibitor of PAF and histamine (H1) receptor | ||||
| GC12039 | Cyclizine 2HCl | 5897-18-7 | >98% | |
Histamine H1 receptor antagonist | ||||
| GC12061 | Tripelennamine HCl | 154-69-8 | >99.50% | |
Tripelennamine HCl, an ethylenediamine derivative, is a potent histamine H1-receptor antagonist. | ||||
| GC12365 | Ranitidine hydrochloride | 66357-59-3 | >98.00% | |
Ranitidine hydrochloride, an inhibitor of gastric acid secretion, competitively antagonizes histamine-induced increases in contraction frequency with a pA2 value of 7.2. | ||||
| GC12549 | Mizolastine | 108612-45-9 | >98.00% | |
Histamine H1-receptor antagonist | ||||
| GC12794 | Nizatidine | 76963-41-2 | >99.00% | |
Histamine H2 receptor antagonist | ||||
| GC12924 | Ciproxifan | 184025-18-1 | >98% | |
Histamine H3-receptor antagonist | ||||
| GC13341 | Brompheniramine hydrogen maleate | 980-71-2 | >99.50% | |
Brompheniramine ((±)-Brompheniramine) maleate is a potent and orally active antihistamine of the alkylamine class. | ||||
| GC13486 | Cimetidine | 51481-61-9 | >98.00% | |
H2 receptor antagonist | ||||
| GC14070 | Azatadine | 3964-81-6 | >98% | |
Histamine and cholinergic inhibitor | ||||
| GC14250 | Bepotastine Besilate | 190786-44-8 | >99.50% | |
Non-sedating, selective antagonist of histamine 1 (H1) receptor | ||||
| GC14726 | Mianserin HCl | 21535-47-7 | >99.50% | |
Mianserin HCl (Org GB 94) is a H1 receptor inverse agonist and is a psychoactive agent of the tetracyclic antidepressant. | ||||
| GC14892 | Clemastine Fumarate | 14976-57-9 | >99.50% | |
Clemastine Fumarate, the over-the-counter antihistamine and muscarinic receptor blocker, has remyelinating potential in Multiple sclerosis (MS). | ||||
| GC15068 | Buclizine HCl | 129-74-8 | >98.00% | |
Buclizine HCl is an orally active antihistamine antiallergic compound. | ||||
| GC15214 | Levodropropizine | 99291-25-5 | >99.50% | |
Histamine receptor inhibitor,cough suppressant | ||||