Histamine Receptor
Histamine receptor has 4 subtypes (H1,H2,H3 and H4) which mediates various biological fuctions, including allergic reaction, gastric acid secretion and inflammation etc.
Products Related to Histamine Receptor(243)
- GC11291Mepyramine maleateCAS: 59-33-6Purity: >99.50%
Mepyramine maleate is mainly used as H 1 antagonists, which has a high affinity pK d of 9.4.
- GC11382Pitolisant hydrochlorideCAS: 903576-44-3Purity: >99.50%
A histamine H 3 receptor antagonist and inverse agonist
- GC11809(R)-(-)-α-Methylhistamine dihydrobromideCAS: 868698-49-1Purity: >98.00%
(R)-(-)-α-Methylhistamine dihydrobromide is a potent, selective and brain-penetrant agonist of H3 histamine receptor, with a Kd of 50.3 nM.
- GC11883Dimaprit dihydrochlorideCAS: 23256-33-9Purity: >98%
Dimaprit dihydrochloride is a highly specific histamine H2-receptor agonist, with an IC 50 value of 49μM for nitric oxide synthase (NOS).
- GC12030Epinastine HClCAS: 108929-04-0Purity: >99.00%
Epinastine HCl (WAL801 hydrochloride) is an antihistamine and mast cell stabilizer.
- GC12085ROS 234 dioxalateCAS: 184576-87-2Purity: >98%
ROS 234 dioxalate is a potent H3 antagonist, with a pKB of 9.46 for Guinea-pig ileum H3-receptor, a pKi of 8.90 for Rat cerebral cortex H3-receptor, and a ED50 of 19.12 mg/kg (ip) in ex vivo of Rat cerebral cortex.
- GC12892Doxepin (hydrochloride)CAS: 1229-29-4Purity: >98.00%
histamine, serotonin, adrenergic, and muscarinic receptors antagonist
- GC12966Immepip dihydrobromideCAS: 164391-47-3Purity: >98.00%
Immepip dihydrobromide is a potent and specific H3 agonist.
- GC13266trans-Triprolidine hydrochlorideCAS: 550-70-9Purity: >98%
trans-Triprolidine hydrochloride is an orally active histamine H1 antagonist.
- GC13465Chlorcyclizine (hydrochloride)CAS: 14362-31-3Purity: >99.50%
histamine H1 receptor antagonist and inhibits HCV
| Catalog No. | Product Name | CAS No. | Purity | Structure |
|---|---|---|---|---|
| GC11220 | Imetit dihydrobromide | 32385-58-3 | >95.00% | |
H3 and H4 receptors agonist | ||||
| GC11291 | Mepyramine maleate | 59-33-6 | >99.50% | |
Mepyramine maleate is mainly used as H 1 antagonists, which has a high affinity pK d of 9.4. | ||||
| GC11330 | Tiotidine | 69014-14-8 | >98.50% | |
Potent histamine H2-receptor antagonist | ||||
| GC11382 | Pitolisant hydrochloride | 903576-44-3 | >99.50% | |
A histamine H 3 receptor antagonist and inverse agonist | ||||
| GC11695 | Cinnarizine | 298-57-7 | >99.50% | |
antihistamine and calcium channel blocker | ||||
| GC11809 | (R)-(-)-α-Methylhistamine dihydrobromide | 868698-49-1 | >98.00% | |
(R)-(-)-α-Methylhistamine dihydrobromide is a potent, selective and brain-penetrant agonist of H3 histamine receptor, with a Kd of 50.3 nM. | ||||
| GC11883 | Dimaprit dihydrochloride | 23256-33-9 | >98% | |
Dimaprit dihydrochloride is a highly specific histamine H2-receptor agonist, with an IC 50 value of 49μM for nitric oxide synthase (NOS). | ||||
| GC12030 | Epinastine HCl | 108929-04-0 | >99.00% | |
Epinastine HCl (WAL801 hydrochloride) is an antihistamine and mast cell stabilizer. | ||||
| GC12085 | ROS 234 dioxalate | 184576-87-2 | >98% | |
ROS 234 dioxalate is a potent H3 antagonist, with a pKB of 9.46 for Guinea-pig ileum H3-receptor, a pKi of 8.90 for Rat cerebral cortex H3-receptor, and a ED50 of 19.12 mg/kg (ip) in ex vivo of Rat cerebral cortex. | ||||
| GC12238 | Oxomemazine | 3689-50-7 | >98% | |
NULL | ||||
| GC12265 | Iodophenpropit dihydrobromide | 145196-87-8 | >98% | |
H3 antagonist | ||||
| GC12293 | Perphenazine | 58-39-9 | >99.50% | |
dopamine antagonist | ||||
| GC12371 | JNJ 10181457 dihydrochloride | 544707-19-9 | >98% | |
Histamine H3 receptor antagonist | ||||
| GC12444 | Clemizole | 442-52-4 | >98% | |
An antihistamine and TRPC5 channel blocker | ||||
| GC12472 | Amthamine dihydrobromide | 142457-00-9 | >98% | |
H2 agonist | ||||
| GC12737 | 4-Methylhistamine dihydrochloride | 36376-47-3 | >95.00% | |
H4 receptor agonist | ||||
| GC12749 | Conessine | 546-06-5 | >98% | |
Conessine is a steroidal alkaloid and a potent, selective histamine H3 receptor antagonist (pK i =8.27). | ||||
| GC12892 | Doxepin (hydrochloride) | 1229-29-4 | >98.00% | |
histamine, serotonin, adrenergic, and muscarinic receptors antagonist | ||||
| GC12966 | Immepip dihydrobromide | 164391-47-3 | >98.00% | |
Immepip dihydrobromide is a potent and specific H3 agonist. | ||||
| GC13024 | Metiamide | 34839-70-8 | >98% | |
| GC13266 | trans-Triprolidine hydrochloride | 550-70-9 | >98% | |
trans-Triprolidine hydrochloride is an orally active histamine H1 antagonist. | ||||
| GC13388 | Zolantidine dimaleate | 104076-39-3 | >98% | |
H2 receptor antagonist | ||||
| GC13465 | Chlorcyclizine (hydrochloride) | 14362-31-3 | >99.50% | |
histamine H1 receptor antagonist and inhibits HCV | ||||
| GC13496 | Thioperamide | 106243-16-7 | >98% | |
histamine H3 and H4 antagonist/inverse agonist | ||||